ATE412646T1 - Zur behandlung von schmerzen geeignete therapeutische mittel - Google Patents

Zur behandlung von schmerzen geeignete therapeutische mittel

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Publication number
ATE412646T1
ATE412646T1 AT04784627T AT04784627T ATE412646T1 AT E412646 T1 ATE412646 T1 AT E412646T1 AT 04784627 T AT04784627 T AT 04784627T AT 04784627 T AT04784627 T AT 04784627T AT E412646 T1 ATE412646 T1 AT E412646T1
Authority
AT
Austria
Prior art keywords
pain
treatment
therapeutic agents
agents suitable
compound
Prior art date
Application number
AT04784627T
Other languages
English (en)
Inventor
Qun Sun
Original Assignee
Euro Celtique Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Euro Celtique Sa filed Critical Euro Celtique Sa
Application granted granted Critical
Publication of ATE412646T1 publication Critical patent/ATE412646T1/de

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C07D213/80—Acids; Esters in position 3
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Ophthalmology & Optometry (AREA)
  • Diabetes (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Virology (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Obesity (AREA)
  • Reproductive Health (AREA)
  • Rheumatology (AREA)
AT04784627T 2003-09-22 2004-09-21 Zur behandlung von schmerzen geeignete therapeutische mittel ATE412646T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US50473003P 2003-09-22 2003-09-22

Publications (1)

Publication Number Publication Date
ATE412646T1 true ATE412646T1 (de) 2008-11-15

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
AT04784627T ATE412646T1 (de) 2003-09-22 2004-09-21 Zur behandlung von schmerzen geeignete therapeutische mittel

Country Status (16)

Country Link
US (3) US7772254B2 (de)
EP (1) EP1664016B9 (de)
JP (1) JP4630871B2 (de)
CN (1) CN1863790A (de)
AT (1) ATE412646T1 (de)
AU (1) AU2004276252B2 (de)
CA (1) CA2537004A1 (de)
CY (1) CY1109242T1 (de)
DE (1) DE602004017481D1 (de)
DK (1) DK1664016T3 (de)
ES (1) ES2317052T3 (de)
MX (1) MXPA06003123A (de)
PL (1) PL1664016T3 (de)
PT (1) PT1664016E (de)
SI (1) SI1664016T1 (de)
WO (1) WO2005030753A2 (de)

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DE60234812D1 (de) 2001-01-29 2010-02-04 Shionogi & Co Arzneipräparat, das als wirkstoff 5-methyl-1-phenyl-2-(1h)-pyridon enthält
US7582635B2 (en) 2002-12-24 2009-09-01 Purdue Pharma, L.P. Therapeutic agents useful for treating pain
PT2017276E (pt) * 2003-09-22 2011-04-05 Euro Celtique Sa Compostos de fenilcarboxamida úteis para o tratamento da dor
WO2005073193A1 (en) * 2004-01-23 2005-08-11 Amgen Inc. Vanilloid receptor ligands and their use in treatments
EP1959944A1 (de) * 2005-12-15 2008-08-27 Shionogi Co., Ltd. Pharmazeutische zusammensetzung mit einem amin-derivat
US20080051380A1 (en) 2006-08-25 2008-02-28 Auerbach Alan H Methods and compositions for treating cancer
BRPI0810195A2 (pt) * 2007-04-13 2014-12-30 Novartis Ag Moduladores de gpbar1
NZ581614A (en) 2007-05-03 2011-06-30 Pfizer Ltd 2-pyridine carboxamide derivatives as sodium channel modulators
US20100249941A1 (en) * 2007-05-15 2010-09-30 Fell Barry M Surgically implantable knee prosthesis with captured keel
US8759362B2 (en) * 2008-10-24 2014-06-24 Purdue Pharma L.P. Bicycloheteroaryl compounds and their use as TRPV1 ligands
US8703962B2 (en) * 2008-10-24 2014-04-22 Purdue Pharma L.P. Monocyclic compounds and their use as TRPV1 ligands
CN102030771B (zh) * 2009-09-30 2013-07-17 孙群 作为trpv1阻断剂的化合物、药物组合物及其医药用途
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JP4630871B2 (ja) 2011-02-09
US7772254B2 (en) 2010-08-10
EP1664016B9 (de) 2009-07-08
CY1109242T1 (el) 2014-07-02
HK1091481A1 (en) 2007-01-19
CA2537004A1 (en) 2005-04-07
DE602004017481D1 (de) 2008-12-11
US20100317670A1 (en) 2010-12-16
US7994177B2 (en) 2011-08-09
CN1863790A (zh) 2006-11-15
PL1664016T3 (pl) 2009-04-30
ES2317052T3 (es) 2009-04-16
EP1664016B1 (de) 2008-10-29
US20110288100A1 (en) 2011-11-24
AU2004276252A1 (en) 2005-04-07
US20060241117A1 (en) 2006-10-26
DK1664016T3 (da) 2009-02-23
SI1664016T1 (sl) 2009-04-30
PT1664016E (pt) 2008-12-29
AU2004276252B2 (en) 2007-11-22
EP1664016A2 (de) 2006-06-07

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