CY1109242T1 - Θεραπευτικοι παραγοντες χρησιμοι για θεραπεια πονου - Google Patents

Θεραπευτικοι παραγοντες χρησιμοι για θεραπεια πονου

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Publication number
CY1109242T1
CY1109242T1 CY20091100095T CY091100095T CY1109242T1 CY 1109242 T1 CY1109242 T1 CY 1109242T1 CY 20091100095 T CY20091100095 T CY 20091100095T CY 091100095 T CY091100095 T CY 091100095T CY 1109242 T1 CY1109242 T1 CY 1109242T1
Authority
CY
Cyprus
Prior art keywords
therapeutic agents
agents useful
pain treatment
compound
animal
Prior art date
Application number
CY20091100095T
Other languages
English (en)
Inventor
Qun Sun
Original Assignee
Euro-Celtique S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Euro-Celtique S.A. filed Critical Euro-Celtique S.A.
Publication of CY1109242T1 publication Critical patent/CY1109242T1/el

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79Acids; Esters
    • C07D213/80Acids; Esters in position 3
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    • C07DHETEROCYCLIC COMPOUNDS
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    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81Amides; Imides

Abstract

Η παρούσα εφεύρεση αποκαλύπτει μία ένωση του τύπου:
CY20091100095T 2003-09-22 2009-01-27 Θεραπευτικοι παραγοντες χρησιμοι για θεραπεια πονου CY1109242T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US50473003P 2003-09-22 2003-09-22
EP04784627A EP1664016B9 (en) 2003-09-22 2004-09-21 Therapeutic agents useful for treating pain

Publications (1)

Publication Number Publication Date
CY1109242T1 true CY1109242T1 (el) 2014-07-02

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Family Applications (1)

Application Number Title Priority Date Filing Date
CY20091100095T CY1109242T1 (el) 2003-09-22 2009-01-27 Θεραπευτικοι παραγοντες χρησιμοι για θεραπεια πονου

Country Status (17)

Country Link
US (3) US7772254B2 (el)
EP (1) EP1664016B9 (el)
JP (1) JP4630871B2 (el)
CN (1) CN1863790A (el)
AT (1) ATE412646T1 (el)
AU (1) AU2004276252B2 (el)
CA (1) CA2537004A1 (el)
CY (1) CY1109242T1 (el)
DE (1) DE602004017481D1 (el)
DK (1) DK1664016T3 (el)
ES (1) ES2317052T3 (el)
HK (1) HK1091481A1 (el)
MX (1) MXPA06003123A (el)
PL (1) PL1664016T3 (el)
PT (1) PT1664016E (el)
SI (1) SI1664016T1 (el)
WO (1) WO2005030753A2 (el)

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JP5876423B2 (ja) 2010-06-22 2016-03-02 塩野義製薬株式会社 Trpv1阻害活性を有する化合物とその使用
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TWI453205B (zh) 2011-06-22 2014-09-21 Purdue Pharma Lp 包含二羥基取代基之trpv1拮抗劑及其用途
AU2012293417A1 (en) 2011-08-10 2013-05-02 Purdue Pharma L.P. TRPV1 antagonists including dihydroxy substituent and uses thereof
TWI572597B (zh) 2012-06-29 2017-03-01 美國禮來大藥廠 二甲基-苯甲酸化合物
WO2014121033A1 (en) 2013-02-04 2014-08-07 Fl Therapeutics Llc Soluble complexes of drug analogs and albumin
ES2729642T3 (es) * 2013-09-24 2019-11-05 Purdue Pharma Lp Tratamiento del dolor por quemaduras mediante moduladores de TRPV1
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DE102022104759A1 (de) 2022-02-28 2023-08-31 SCi Kontor GmbH Co-Kristall-Screening Verfahren, insbesondere zur Herstellung von Co-Kristallen

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MXPA06003123A (es) 2006-05-31
ATE412646T1 (de) 2008-11-15
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PL1664016T3 (pl) 2009-04-30
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US20060241117A1 (en) 2006-10-26
US20100317670A1 (en) 2010-12-16
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