UA84710C2 - Пиперидиновые производные, фармацевтическая композиция, которая их содержит, и способ лечения - Google Patents

Пиперидиновые производные, фармацевтическая композиция, которая их содержит, и способ лечения

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Publication number
UA84710C2
UA84710C2 UAA200601979A UAA200601979A UA84710C2 UA 84710 C2 UA84710 C2 UA 84710C2 UA A200601979 A UAA200601979 A UA A200601979A UA A200601979 A UAA200601979 A UA A200601979A UA 84710 C2 UA84710 C2 UA 84710C2
Authority
UA
Ukraine
Prior art keywords
piperidine compound
piperidine compounds
animal
pharmaceutical compositions
treatment method
Prior art date
Application number
UAA200601979A
Other languages
English (en)
Ukrainian (uk)
Inventor
Квун Сун
Кейт Вен
Ксяоминг Жоу
Original Assignee
Евро-Селтик С.А.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Евро-Селтик С.А. filed Critical Евро-Селтик С.А.
Publication of UA84710C2 publication Critical patent/UA84710C2/ru

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P27/02Ophthalmic agents
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    • AHUMAN NECESSITIES
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Addiction (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Psychology (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Communicable Diseases (AREA)
  • Transplantation (AREA)
  • Endocrinology (AREA)
UAA200601979A 2003-07-24 2004-07-23 Пиперидиновые производные, фармацевтическая композиция, которая их содержит, и способ лечения UA84710C2 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US48951503P 2003-07-24 2003-07-24

Publications (1)

Publication Number Publication Date
UA84710C2 true UA84710C2 (ru) 2008-11-25

Family

ID=34102892

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Application Number Title Priority Date Filing Date
UAA200601979A UA84710C2 (ru) 2003-07-24 2004-07-23 Пиперидиновые производные, фармацевтическая композиция, которая их содержит, и способ лечения

Country Status (29)

Country Link
US (2) US7572812B2 (ru)
EP (2) EP2067776A1 (ru)
JP (1) JP4686456B2 (ru)
KR (2) KR100977242B1 (ru)
CN (2) CN1829708A (ru)
AT (1) ATE430741T1 (ru)
AU (1) AU2004259357B2 (ru)
BR (1) BRPI0412808A (ru)
CA (1) CA2533509C (ru)
CY (1) CY1109273T1 (ru)
DE (1) DE602004020994D1 (ru)
DK (1) DK1648878T3 (ru)
EA (1) EA010852B1 (ru)
ES (1) ES2326979T3 (ru)
GE (1) GEP20094676B (ru)
HK (1) HK1089755A1 (ru)
HR (1) HRP20090404T1 (ru)
IL (3) IL173343A (ru)
IS (1) IS2684B (ru)
MA (1) MA27983A1 (ru)
MX (1) MXPA06000941A (ru)
NO (1) NO20060910L (ru)
NZ (1) NZ545506A (ru)
PL (1) PL1648878T3 (ru)
PT (1) PT1648878E (ru)
SI (1) SI1648878T1 (ru)
UA (1) UA84710C2 (ru)
WO (1) WO2005009987A1 (ru)
ZA (1) ZA200509562B (ru)

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JP4521777B2 (ja) 2003-07-24 2010-08-11 ユーロ−セルティーク エス.エイ. 疼痛治療または予防に有用な4−ヘテロアリール−テトラヒドロピペリジル化合物
EP1812439B2 (en) 2004-10-15 2017-12-06 Takeda Pharmaceutical Company Limited Kinase inhibitors
US20060281718A1 (en) * 2005-05-12 2006-12-14 Bannon Anthony W Treatment of VR1-antagonist-induced increase in body temperature with an antipyretic agent
DE102005023943A1 (de) 2005-05-20 2006-11-23 Grünenthal GmbH Pentafluorsulfanyl-substituierte Verbindung und deren Verwendung zur Herstellung von Arzneimitteln
US8119655B2 (en) 2005-10-07 2012-02-21 Takeda Pharmaceutical Company Limited Kinase inhibitors
EA200970361A1 (ru) 2006-10-09 2010-02-26 Такеда Фармасьютикал Компани Лимитед Ингибиторы киназы
NZ579820A (en) 2007-04-27 2011-01-28 Purdue Pharma Lp Therapeutic agents useful for treating pain
AU2011226773C1 (en) * 2007-04-27 2012-07-26 Purdue Pharma L.P. TRPV1 antagonists and uses thereof
PT2142529E (pt) * 2007-04-27 2014-03-20 Purdue Pharma Lp Antagonistas de trpv1 e as respectivas utilizações
US8084616B2 (en) 2007-10-24 2011-12-27 Abbott Laboratories TRPV1 antagonists
US11969501B2 (en) 2008-04-21 2024-04-30 Dompé Farmaceutici S.P.A. Auris formulations for treating otic diseases and conditions
CA2721927C (en) 2008-04-21 2014-01-28 Otonomy, Inc. Auris formulations for treating otic diseases and conditions
US10092580B2 (en) 2008-07-21 2018-10-09 Otonomy, Inc. Controlled-release otic structure modulating and innate immune system modulating compositions and methods for the treatment of otic disorders
US8703962B2 (en) * 2008-10-24 2014-04-22 Purdue Pharma L.P. Monocyclic compounds and their use as TRPV1 ligands
US8759362B2 (en) * 2008-10-24 2014-06-24 Purdue Pharma L.P. Bicycloheteroaryl compounds and their use as TRPV1 ligands
WO2010064597A1 (ja) * 2008-12-01 2010-06-10 武田薬品工業株式会社 ピペリジン誘導体
CN102098080B (zh) * 2009-12-09 2014-07-02 京信通信系统(中国)有限公司 数字微波射频拉远覆盖系统及方法
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