DK1648878T3 - Piperidinforbindelser og farmaceutiske sammensætninger, som indeholder dem - Google Patents

Piperidinforbindelser og farmaceutiske sammensætninger, som indeholder dem

Info

Publication number
DK1648878T3
DK1648878T3 DK04779120T DK04779120T DK1648878T3 DK 1648878 T3 DK1648878 T3 DK 1648878T3 DK 04779120 T DK04779120 T DK 04779120T DK 04779120 T DK04779120 T DK 04779120T DK 1648878 T3 DK1648878 T3 DK 1648878T3
Authority
DK
Denmark
Prior art keywords
piperidine compound
animal
disclosed
piperidine compounds
piperidine
Prior art date
Application number
DK04779120T
Other languages
English (en)
Inventor
Qun Sun
Xiaoming Zhou
Kate Wen
Original Assignee
Euro Celtique Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Euro Celtique Sa filed Critical Euro Celtique Sa
Application granted granted Critical
Publication of DK1648878T3 publication Critical patent/DK1648878T3/da

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • AHUMAN NECESSITIES
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    • AHUMAN NECESSITIES
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
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    • AHUMAN NECESSITIES
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    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P7/12Antidiuretics, e.g. drugs for diabetes insipidus
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    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Communicable Diseases (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Transplantation (AREA)
  • Vascular Medicine (AREA)
DK04779120T 2003-07-24 2004-07-23 Piperidinforbindelser og farmaceutiske sammensætninger, som indeholder dem DK1648878T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US48951503P 2003-07-24 2003-07-24
PCT/US2004/023912 WO2005009987A1 (en) 2003-07-24 2004-07-23 Piperidine compounds and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
DK1648878T3 true DK1648878T3 (da) 2009-08-10

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Family Applications (1)

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DK04779120T DK1648878T3 (da) 2003-07-24 2004-07-23 Piperidinforbindelser og farmaceutiske sammensætninger, som indeholder dem

Country Status (29)

Country Link
US (2) US7572812B2 (da)
EP (2) EP2067776A1 (da)
JP (1) JP4686456B2 (da)
KR (2) KR100954415B1 (da)
CN (2) CN101914088A (da)
AT (1) ATE430741T1 (da)
AU (1) AU2004259357B2 (da)
BR (1) BRPI0412808A (da)
CA (1) CA2533509C (da)
CY (1) CY1109273T1 (da)
DE (1) DE602004020994D1 (da)
DK (1) DK1648878T3 (da)
EA (1) EA010852B1 (da)
ES (1) ES2326979T3 (da)
GE (1) GEP20094676B (da)
HK (1) HK1089755A1 (da)
HR (1) HRP20090404T1 (da)
IL (3) IL173343A (da)
IS (1) IS2684B (da)
MA (1) MA27983A1 (da)
MX (1) MXPA06000941A (da)
NO (1) NO20060910L (da)
NZ (1) NZ545506A (da)
PL (1) PL1648878T3 (da)
PT (1) PT1648878E (da)
SI (1) SI1648878T1 (da)
UA (1) UA84710C2 (da)
WO (1) WO2005009987A1 (da)
ZA (1) ZA200509562B (da)

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MY142655A (en) * 2003-06-12 2010-12-15 Euro Celtique Sa Therapeutic agents useful for treating pain
EA009480B1 (ru) 2003-07-24 2008-02-28 Еуро-Селтик С. А. Гетероарил-тетрагидропиридины и их применение для лечения или профилактики боли
US7713973B2 (en) 2004-10-15 2010-05-11 Takeda Pharmaceutical Company Limited Kinase inhibitors
AU2006247487A1 (en) * 2005-05-12 2006-11-23 Amgen Inc. Antipyretic agents against VR1-antagonist-induced increases in body temperature
DE102005023943A1 (de) 2005-05-20 2006-11-23 Grünenthal GmbH Pentafluorsulfanyl-substituierte Verbindung und deren Verwendung zur Herstellung von Arzneimitteln
US8119655B2 (en) 2005-10-07 2012-02-21 Takeda Pharmaceutical Company Limited Kinase inhibitors
SG158147A1 (en) 2006-10-09 2010-01-29 Takeda Pharmaceutical Kinase inhibitors
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CA2833209C (en) 2007-04-27 2016-06-28 Purdue Pharma L.P. Piperidine and piperazine compounds as trpv1 antagonists
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US8084616B2 (en) 2007-10-24 2011-12-27 Abbott Laboratories TRPV1 antagonists
US11969501B2 (en) 2008-04-21 2024-04-30 Dompé Farmaceutici S.P.A. Auris formulations for treating otic diseases and conditions
CN104491864A (zh) 2008-04-21 2015-04-08 奥德纳米有限公司 用于治疗耳部疾病和病况的耳用调配物及方法
EP2306975A4 (en) 2008-07-21 2012-10-31 Otonomy Inc CONTROLLED RELEASE COMPOSITIONS MODULATING THE OTIC STRUCTURE AND MODULATING THE NATURAL IMMUNE SYSTEM AND METHODS OF TREATING OTIC DISORDERS
US8703962B2 (en) * 2008-10-24 2014-04-22 Purdue Pharma L.P. Monocyclic compounds and their use as TRPV1 ligands
US8759362B2 (en) * 2008-10-24 2014-06-24 Purdue Pharma L.P. Bicycloheteroaryl compounds and their use as TRPV1 ligands
WO2010064597A1 (ja) * 2008-12-01 2010-06-10 武田薬品工業株式会社 ピペリジン誘導体
CN102098080B (zh) * 2009-12-09 2014-07-02 京信通信系统(中国)有限公司 数字微波射频拉远覆盖系统及方法
EA201290505A1 (ru) 2009-12-15 2013-01-30 Ньюроп, Инк. Соединения для лечения неврологических расстройств
US8921373B2 (en) 2010-06-22 2014-12-30 Shionogi & Co., Ltd. Compounds having TRPV1 antagonistic activity and uses thereof
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