AU2016361428A1 - Triazole ACC inhibitors and uses thereof - Google Patents
Triazole ACC inhibitors and uses thereof Download PDFInfo
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- AU2016361428A1 AU2016361428A1 AU2016361428A AU2016361428A AU2016361428A1 AU 2016361428 A1 AU2016361428 A1 AU 2016361428A1 AU 2016361428 A AU2016361428 A AU 2016361428A AU 2016361428 A AU2016361428 A AU 2016361428A AU 2016361428 A1 AU2016361428 A1 AU 2016361428A1
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Classifications
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
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- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
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- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
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Landscapes
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- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
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| RU2016134947A (ru) | 2014-01-31 | 2018-03-01 | Дана-Фарбер Кансер Институт, Инк. | Производные диаминопиримидин бензолсульфона и их применение |
| US10793571B2 (en) | 2014-01-31 | 2020-10-06 | Dana-Farber Cancer Institute, Inc. | Uses of diazepane derivatives |
| BR112018004618A2 (pt) | 2015-09-11 | 2018-09-25 | Dana-Farber Cancer Institute, Inc. | ciano tienotriazoldiazepinas e usos das mesmas |
| CA2996977A1 (en) | 2015-09-11 | 2017-03-16 | Dana-Farber Cancer Institute, Inc. | Acetamide thienotriazolodiazepines and uses thereof |
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| SI3379933T1 (sl) | 2015-11-25 | 2023-07-31 | Gilead Apollo, Llc | Fungicidni sestavki, ki vsebujejo derivate 2,4-diokso-1,4-dihidrotieno (2,3-d)pirimidina |
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| US10913752B2 (en) | 2015-11-25 | 2021-02-09 | Dana-Farber Cancer Institute, Inc. | Bivalent bromodomain inhibitors and uses thereof |
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| CN108341830B (zh) | 2017-01-22 | 2021-03-02 | 广东东阳光药业有限公司 | 噻吩并嘧啶衍生物及其在药物中的应用 |
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| MX2018006288A (es) | 2015-11-25 | 2018-09-07 | Gilead Apollo Llc | Inhibidores de acc tipo ester y usos de los mismos. |
| US20170166582A1 (en) | 2015-11-25 | 2017-06-15 | Gilead Apollo, Llc | Pyrazole acc inhibitors and uses thereof |
| AU2016361428A1 (en) | 2015-11-25 | 2018-05-24 | Gilead Apollo, Llc | Triazole ACC inhibitors and uses thereof |
| US10913752B2 (en) | 2015-11-25 | 2021-02-09 | Dana-Farber Cancer Institute, Inc. | Bivalent bromodomain inhibitors and uses thereof |
| EP3888658B1 (en) | 2015-11-25 | 2023-12-27 | Effector Therapeutics, Inc. | Eif4-a-inhibiting compounds and methods related thereto |
| SI3379933T1 (sl) | 2015-11-25 | 2023-07-31 | Gilead Apollo, Llc | Fungicidni sestavki, ki vsebujejo derivate 2,4-diokso-1,4-dihidrotieno (2,3-d)pirimidina |
| RU2753056C2 (ru) | 2016-12-16 | 2021-08-11 | Систик Файбросис Фаундейшн | Бициклические гетероарильные производные в качестве стимуляторов cftr |
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2016
- 2016-11-22 AU AU2016361428A patent/AU2016361428A1/en not_active Abandoned
- 2016-11-22 BR BR112018010453-1A patent/BR112018010453B1/pt active IP Right Grant
- 2016-11-22 US US15/359,414 patent/US20170166584A1/en not_active Abandoned
- 2016-11-22 KR KR1020187016698A patent/KR20180082557A/ko not_active Withdrawn
- 2016-11-22 PT PT168092724T patent/PT3380479T/pt unknown
- 2016-11-22 CA CA3005900A patent/CA3005900C/en active Active
- 2016-11-22 EP EP16809272.4A patent/EP3380479B1/en active Active
- 2016-11-22 WO PCT/US2016/063410 patent/WO2017091617A1/en not_active Ceased
- 2016-11-22 JP JP2018525706A patent/JP2018536661A/ja active Pending
- 2016-11-22 ES ES16809272T patent/ES2939977T3/es active Active
- 2016-11-22 MX MX2018006287A patent/MX2018006287A/es unknown
- 2016-11-22 PL PL16809272.4T patent/PL3380479T3/pl unknown
- 2016-11-22 CN CN201680067505.7A patent/CN108349994B/zh active Active
- 2016-11-22 EA EA201890926A patent/EA201890926A1/ru unknown
- 2016-11-22 SI SI201631672T patent/SI3380479T1/sl unknown
- 2016-11-24 AR ARP160103601A patent/AR106806A1/es active IP Right Grant
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2018
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- 2018-05-23 CO CONC2018/0005369A patent/CO2018005369A2/es unknown
- 2018-08-20 US US15/999,505 patent/US20190241582A1/en not_active Abandoned
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2019
- 2019-04-24 US US16/393,454 patent/US10800791B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| KR20180082557A (ko) | 2018-07-18 |
| PT3380479T (pt) | 2023-03-13 |
| BR112018010453A8 (pt) | 2019-02-26 |
| US20170166584A1 (en) | 2017-06-15 |
| WO2017091617A1 (en) | 2017-06-01 |
| JP2018536661A (ja) | 2018-12-13 |
| CL2018001360A1 (es) | 2018-08-24 |
| BR112018010453A2 (pt) | 2018-11-21 |
| EA201890926A1 (ru) | 2018-12-28 |
| ES2939977T3 (es) | 2023-04-28 |
| EP3380479B1 (en) | 2022-12-07 |
| MX2018006287A (es) | 2018-09-07 |
| US10800791B2 (en) | 2020-10-13 |
| CA3005900C (en) | 2023-10-31 |
| AR106806A1 (es) | 2018-02-21 |
| SI3380479T1 (sl) | 2023-04-28 |
| CA3005900A1 (en) | 2017-06-01 |
| CN108349994A (zh) | 2018-07-31 |
| CN108349994B (zh) | 2021-06-22 |
| BR112018010453B1 (pt) | 2022-06-14 |
| EP3380479A1 (en) | 2018-10-03 |
| CO2018005369A2 (es) | 2018-05-31 |
| PL3380479T3 (pl) | 2023-05-08 |
| US20190241582A1 (en) | 2019-08-08 |
| US20200017519A1 (en) | 2020-01-16 |
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