AU2012273365A1 - Glucagon/glp-1 receptor co-agonists - Google Patents
Glucagon/glp-1 receptor co-agonists Download PDFInfo
- Publication number
- AU2012273365A1 AU2012273365A1 AU2012273365A AU2012273365A AU2012273365A1 AU 2012273365 A1 AU2012273365 A1 AU 2012273365A1 AU 2012273365 A AU2012273365 A AU 2012273365A AU 2012273365 A AU2012273365 A AU 2012273365A AU 2012273365 A1 AU2012273365 A1 AU 2012273365A1
- Authority
- AU
- Australia
- Prior art keywords
- amino acid
- peptide
- glucagon
- receptor
- acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/605—Glucagons
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
- A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
- A61K47/60—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
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-
2012
- 2012-06-12 BR BR112013032717A patent/BR112013032717A2/pt not_active IP Right Cessation
- 2012-06-12 AU AU2012273365A patent/AU2012273365A1/en not_active Abandoned
- 2012-06-12 JP JP2014517015A patent/JP6184404B2/ja not_active Expired - Fee Related
- 2012-06-12 KR KR1020147001710A patent/KR20140043793A/ko not_active Withdrawn
- 2012-06-12 US US13/494,480 patent/US8729017B2/en not_active Expired - Fee Related
- 2012-06-12 EP EP12803439.4A patent/EP2723766A4/en not_active Withdrawn
- 2012-06-12 WO PCT/US2012/042085 patent/WO2012177444A2/en not_active Ceased
- 2012-06-12 CN CN201280040883.8A patent/CN103748109A/zh active Pending
- 2012-06-12 MX MX2013015168A patent/MX2013015168A/es not_active Application Discontinuation
- 2012-06-12 RU RU2014101697/10A patent/RU2014101697A/ru not_active Application Discontinuation
- 2012-06-12 US US14/127,469 patent/US9309301B2/en not_active Expired - Fee Related
- 2012-06-12 CA CA2839867A patent/CA2839867A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| RU2014101697A (ru) | 2015-07-27 |
| US20140206607A1 (en) | 2014-07-24 |
| BR112013032717A2 (pt) | 2017-01-24 |
| EP2723766A2 (en) | 2014-04-30 |
| US20120329707A1 (en) | 2012-12-27 |
| US9309301B2 (en) | 2016-04-12 |
| JP6184404B2 (ja) | 2017-08-23 |
| US8729017B2 (en) | 2014-05-20 |
| WO2012177444A3 (en) | 2013-04-25 |
| MX2013015168A (es) | 2014-03-31 |
| JP2014524908A (ja) | 2014-09-25 |
| EP2723766A4 (en) | 2015-05-20 |
| CN103748109A (zh) | 2014-04-23 |
| CA2839867A1 (en) | 2012-12-27 |
| KR20140043793A (ko) | 2014-04-10 |
| WO2012177444A2 (en) | 2012-12-27 |
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