AU2011269989B2 - Novel fused pyrimidine derivatives for inhibition of tyrosine kinase activity - Google Patents
Novel fused pyrimidine derivatives for inhibition of tyrosine kinase activity Download PDFInfo
- Publication number
- AU2011269989B2 AU2011269989B2 AU2011269989A AU2011269989A AU2011269989B2 AU 2011269989 B2 AU2011269989 B2 AU 2011269989B2 AU 2011269989 A AU2011269989 A AU 2011269989A AU 2011269989 A AU2011269989 A AU 2011269989A AU 2011269989 B2 AU2011269989 B2 AU 2011269989B2
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- Prior art keywords
- phenyl
- thieno
- acrylamide
- pyrimidin
- yloxy
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- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2014202057A AU2014202057B2 (en) | 2010-06-23 | 2014-04-11 | Novel Fused Pyrimidine Derivatives for Inhibition of Tyrosine Kinase Activity |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20100059686 | 2010-06-23 | ||
| KR10-2010-0059686 | 2010-06-23 | ||
| PCT/KR2011/004482 WO2011162515A2 (en) | 2010-06-23 | 2011-06-20 | Novel fused pyrimidine derivatives for inhd3ition of tyrosine kinase activity |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2014202057A Division AU2014202057B2 (en) | 2010-06-23 | 2014-04-11 | Novel Fused Pyrimidine Derivatives for Inhibition of Tyrosine Kinase Activity |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| AU2011269989A1 AU2011269989A1 (en) | 2013-02-07 |
| AU2011269989A8 AU2011269989A8 (en) | 2013-02-28 |
| AU2011269989B2 true AU2011269989B2 (en) | 2014-12-11 |
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