AU2008321046B2 - 4-pyrazolyl-N-arylpyrimidin-2-amines and 4-pyrazolyl-N-heteroarylpyrimidin-2-amines as janus kinase inhibitors - Google Patents

4-pyrazolyl-N-arylpyrimidin-2-amines and 4-pyrazolyl-N-heteroarylpyrimidin-2-amines as janus kinase inhibitors Download PDF

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AU2008321046B2
AU2008321046B2 AU2008321046A AU2008321046A AU2008321046B2 AU 2008321046 B2 AU2008321046 B2 AU 2008321046B2 AU 2008321046 A AU2008321046 A AU 2008321046A AU 2008321046 A AU2008321046 A AU 2008321046A AU 2008321046 B2 AU2008321046 B2 AU 2008321046B2
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pyrazol
pyrim
ino
cya
pyra
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AU2008321046A1 (en
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Yun-Long Li
James D. Rodgers
Wenqing Yao
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Incyte Holdings Corp
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Incyte Holdings Corp
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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AU2008321046A 2007-11-16 2008-11-13 4-pyrazolyl-N-arylpyrimidin-2-amines and 4-pyrazolyl-N-heteroarylpyrimidin-2-amines as janus kinase inhibitors Active AU2008321046B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US98860607P 2007-11-16 2007-11-16
US60/988,606 2007-11-16
PCT/US2008/083319 WO2009064835A1 (en) 2007-11-16 2008-11-13 4-pyrazolyl-n-arylpyrimidin-2-amines and 4-pyrazolyl-n-heteroarylpyrimidin-2-amines as janus kinase inhibitors

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AU2008321046A1 AU2008321046A1 (en) 2009-05-22
AU2008321046B2 true AU2008321046B2 (en) 2013-10-24

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US (1) US8309718B2 (https=)
EP (1) EP2220068B1 (https=)
JP (1) JP5480813B2 (https=)
KR (1) KR101580482B1 (https=)
CN (1) CN101910152B (https=)
AU (1) AU2008321046B2 (https=)
BR (1) BRPI0820544A2 (https=)
CA (1) CA2704599C (https=)
CO (1) CO6280420A2 (https=)
CR (1) CR11430A (https=)
EA (1) EA020777B1 (https=)
EC (1) ECSP10010263A (https=)
ES (1) ES2569528T3 (https=)
IL (1) IL205571A (https=)
MX (1) MX2010005300A (https=)
MY (1) MY152948A (https=)
NZ (1) NZ585139A (https=)
UA (1) UA104849C2 (https=)
WO (1) WO2009064835A1 (https=)
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Families Citing this family (113)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005105814A1 (en) * 2004-04-28 2005-11-10 Incyte Corporation Tetracyclic inhibitors of janus kinases
EP2455382B1 (en) 2005-12-13 2016-10-26 Incyte Holdings Corporation Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors
EP2121692B1 (en) * 2006-12-22 2013-04-10 Incyte Corporation Substituted heterocycles as janus kinase inhibitors
EP3070090B1 (en) 2007-06-13 2018-12-12 Incyte Holdings Corporation Use of salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h- pyrazol-1-yl)-3- cyclopentylpropanenitrile
CL2008001709A1 (es) 2007-06-13 2008-11-03 Incyte Corp Compuestos derivados de pirrolo [2,3-b]pirimidina, moduladores de quinasas jak; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, psoriasis, artritis reumatoide, entre otras.
FR2938537B1 (fr) 2008-11-14 2012-10-26 Sanofi Aventis Derives de carbamates d'alkyl-heterocycles, leur preparation et leur application en therapeutique.
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UA104849C2 (uk) 2014-03-25
IL205571A (en) 2015-09-24
IL205571A0 (en) 2010-12-30
ES2569528T3 (es) 2016-05-11
KR20100095582A (ko) 2010-08-31
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CA2704599C (en) 2015-05-12
JP5480813B2 (ja) 2014-04-23
EA201070618A1 (ru) 2010-12-30
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AU2008321046A1 (en) 2009-05-22
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WO2009064835A1 (en) 2009-05-22
HK1147476A1 (zh) 2011-08-12
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