AU2007269060B2 - Hydroxylated and methoxylated cyclopenta [D] pyrimidines as AKT protein kinase inhibitors - Google Patents

Hydroxylated and methoxylated cyclopenta [D] pyrimidines as AKT protein kinase inhibitors Download PDF

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Publication number
AU2007269060B2
AU2007269060B2 AU2007269060A AU2007269060A AU2007269060B2 AU 2007269060 B2 AU2007269060 B2 AU 2007269060B2 AU 2007269060 A AU2007269060 A AU 2007269060A AU 2007269060 A AU2007269060 A AU 2007269060A AU 2007269060 B2 AU2007269060 B2 AU 2007269060B2
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Australia
Prior art keywords
methyl
cyclopenta
dihydro
hydroxy
piperazin
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Active
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AU2007269060A
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AU2007269060A1 (en
Inventor
Anna L. Banka
Josef R. Bencsik
James F. Blake
Christine Chabot
Steven Do
Nicholas C. Kallan
Jun Liang
Ian S. Mitchell
Brian Safina
Stephen T. Schlachter
Keith Lee Spencer
Eli M. Wallace
Dengming Xiao
Rui Xu
Birong Zhang
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Genentech Inc
Array Biopharma Inc
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Genentech Inc
Array Biopharma Inc
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Application filed by Genentech Inc, Array Biopharma Inc filed Critical Genentech Inc
Publication of AU2007269060A1 publication Critical patent/AU2007269060A1/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
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AU2007269060A 2006-07-06 2007-07-05 Hydroxylated and methoxylated cyclopenta [D] pyrimidines as AKT protein kinase inhibitors Active AU2007269060B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2014201211A AU2014201211B2 (en) 2006-07-06 2014-03-05 Hydroxylated and methoxylated cyclopenta [d] pyrimidines as akt protein kinase inhibitors

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US81871806P 2006-07-06 2006-07-06
US60/818,718 2006-07-06
PCT/US2007/072885 WO2008006040A1 (en) 2006-07-06 2007-07-05 Hydroxylated and methoxylated cyclopenta [d] pyrimidines as akt protein kinase inhibitors

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AU2007269060A1 AU2007269060A1 (en) 2008-01-10
AU2007269060B2 true AU2007269060B2 (en) 2014-02-20

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UA99597C2 (ru) 2006-07-06 2012-09-10 Еррей Біофарма Інк. Пиримидилциклопентаны как ингибиторы акт протеинкиназ
US8063050B2 (en) 2006-07-06 2011-11-22 Array Biopharma Inc. Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors
CN101516891B (zh) 2006-07-06 2013-06-05 阵列生物制药公司 作为akt蛋白激酶抑制剂的二氢噻吩并嘧啶
UA95641C2 (xx) * 2006-07-06 2011-08-25 Эррей Биофарма Инк. Гідроксильовані піримідильні циклопентани як інгібітори акт протеїнкінази$гидроксилированные пиримидильные циклопентаны как ингибиторы акт протеинкиназы
WO2008006025A1 (en) * 2006-07-06 2008-01-10 Array Biopharma Inc. Dihydrofuro pyrimidines as akt protein kinase inhibitors
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