AU2003298571B2 - Pyrazolo[1,5-a]pyrimidines compounds as cyclin dependent kinase inhibitors - Google Patents

Pyrazolo[1,5-a]pyrimidines compounds as cyclin dependent kinase inhibitors Download PDF

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Publication number
AU2003298571B2
AU2003298571B2 AU2003298571A AU2003298571A AU2003298571B2 AU 2003298571 B2 AU2003298571 B2 AU 2003298571B2 AU 2003298571 A AU2003298571 A AU 2003298571A AU 2003298571 A AU2003298571 A AU 2003298571A AU 2003298571 B2 AU2003298571 B2 AU 2003298571B2
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cycloalkyl
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AU2003298571A1 (en
Inventor
Carmen S. Alvarez
Tin-Yau Chan
Lawrence W. Dillard
Ronald J. Doll
Michael P. Dwyer
Thierry O. Fischmann
Viyyoor Moopil Girijavallabhan
Timothy J. Guzi
Zhen Min He
Ray Anthony James
Chad Knutson
Vincent Madison
Haengsoon Park
Kamil Paruch
Vinh D. Tran
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Merck Sharp and Dohme LLC
Pharmacopeia LLC
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Merck Sharp and Dohme Ltd
Pharmacopeia Inc
Merck Sharp and Dohme LLC
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Assigned to SCHERING CORPORATION, PHARMACOPEIA, INC. reassignment SCHERING CORPORATION Request for Assignment Assignors: PHARMACOPEIA DRUG DISCOVERY, INC., SCHERING CORPORATION
Assigned to MERCK SHARP & DOHME CORP., PHARMACOPEIA, INC. reassignment MERCK SHARP & DOHME CORP. Request to Amend Deed and Register Assignors: PHARMACOPEIA, INC., SCHERING CORPORATION
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Virology (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Heart & Thoracic Surgery (AREA)
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  • Diabetes (AREA)
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AU2003298571A 2002-09-04 2003-09-03 Pyrazolo[1,5-a]pyrimidines compounds as cyclin dependent kinase inhibitors Ceased AU2003298571B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40802902P 2002-09-04 2002-09-04
US60/408,029 2002-09-04
PCT/US2003/027491 WO2004026229A2 (en) 2002-09-04 2003-09-03 Pyrazolo[1,5-a]pyrimidines compounds as cyclin dependent kinase inhibitors

Publications (2)

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AU2003298571A1 AU2003298571A1 (en) 2004-04-08
AU2003298571B2 true AU2003298571B2 (en) 2006-10-19

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AU2003298571A Ceased AU2003298571B2 (en) 2002-09-04 2003-09-03 Pyrazolo[1,5-a]pyrimidines compounds as cyclin dependent kinase inhibitors

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US (2) US7067661B2 (enExample)
EP (1) EP1534712B1 (enExample)
JP (2) JP4790265B2 (enExample)
KR (1) KR20050033659A (enExample)
CN (1) CN1701073B (enExample)
AR (1) AR041133A1 (enExample)
AT (1) ATE362474T1 (enExample)
AU (1) AU2003298571B2 (enExample)
CA (1) CA2497544C (enExample)
DE (1) DE60313872T2 (enExample)
ES (1) ES2283868T3 (enExample)
MX (1) MXPA05002572A (enExample)
MY (2) MY145332A (enExample)
NZ (1) NZ539161A (enExample)
PE (1) PE20041000A1 (enExample)
TW (1) TWI329645B (enExample)
WO (1) WO2004026229A2 (enExample)
ZA (1) ZA200501846B (enExample)

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