AU2002254567B2 - Amino acid complexes of C-aryl glucosides for treatment of diabetes and method - Google Patents

Amino acid complexes of C-aryl glucosides for treatment of diabetes and method Download PDF

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Publication number
AU2002254567B2
AU2002254567B2 AU2002254567A AU2002254567A AU2002254567B2 AU 2002254567 B2 AU2002254567 B2 AU 2002254567B2 AU 2002254567 A AU2002254567 A AU 2002254567A AU 2002254567 A AU2002254567 A AU 2002254567A AU 2002254567 B2 AU2002254567 B2 AU 2002254567B2
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AU
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Prior art keywords
agent
inhibitor
compounds
compound
alkyl
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Ceased
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AU2002254567A
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AU2002254567A1 (en
Inventor
Jack Z. Gougoutas
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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Publication of AU2002254567A1 publication Critical patent/AU2002254567A1/en
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Publication of AU2002254567B2 publication Critical patent/AU2002254567B2/en
Priority to AU2008200159A priority Critical patent/AU2008200159A1/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
AU2002254567A 2001-04-11 2002-04-08 Amino acid complexes of C-aryl glucosides for treatment of diabetes and method Ceased AU2002254567B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2008200159A AU2008200159A1 (en) 2001-04-11 2008-01-11 Amino acid complexes of C-aryl glucosides for treatment of diabetes and method

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28309701P 2001-04-11 2001-04-11
US60/283,097 2001-04-11
PCT/US2002/011066 WO2002083066A2 (en) 2001-04-11 2002-04-08 Amino acid complexes of c-aryl glucosides for treatment of diabetes and method

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU2008200159A Division AU2008200159A1 (en) 2001-04-11 2008-01-11 Amino acid complexes of C-aryl glucosides for treatment of diabetes and method

Publications (2)

Publication Number Publication Date
AU2002254567A1 AU2002254567A1 (en) 2003-04-17
AU2002254567B2 true AU2002254567B2 (en) 2007-10-11

Family

ID=23084500

Family Applications (1)

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AU2002254567A Ceased AU2002254567B2 (en) 2001-04-11 2002-04-08 Amino acid complexes of C-aryl glucosides for treatment of diabetes and method

Country Status (12)

Country Link
US (1) US6774112B2 (https=)
EP (1) EP1385856B1 (https=)
JP (1) JP2004536047A (https=)
AT (1) ATE318272T1 (https=)
AU (1) AU2002254567B2 (https=)
CA (1) CA2444481A1 (https=)
CY (1) CY1105038T1 (https=)
DE (1) DE60209343T2 (https=)
DK (1) DK1385856T3 (https=)
ES (1) ES2258141T3 (https=)
HU (1) HUP0600232A2 (https=)
WO (1) WO2002083066A2 (https=)

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US20030064935A1 (en) 2003-04-03
JP2004536047A (ja) 2004-12-02
DE60209343T2 (de) 2006-10-26
CY1105038T1 (el) 2010-03-03
HUP0600232A2 (en) 2006-08-28
US6774112B2 (en) 2004-08-10
CA2444481A1 (en) 2002-10-24
DE60209343D1 (de) 2006-04-27
DK1385856T3 (da) 2006-05-15
EP1385856B1 (en) 2006-02-22
ES2258141T3 (es) 2006-08-16
WO2002083066A2 (en) 2002-10-24
WO2002083066A3 (en) 2003-03-06
EP1385856A4 (en) 2005-05-11
ATE318272T1 (de) 2006-03-15

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