AR245445A1 - Procedimiento para la preparacion de cis-1-aril-2-(fluormetil)oxiranos,compuestos asi obtenidos y preparacion de (treo)-1-aril-2-acilamido-3-fluor-1-propanoles utilizando dichos compuestos. - Google Patents

Procedimiento para la preparacion de cis-1-aril-2-(fluormetil)oxiranos,compuestos asi obtenidos y preparacion de (treo)-1-aril-2-acilamido-3-fluor-1-propanoles utilizando dichos compuestos.

Info

Publication number
AR245445A1
AR245445A1 AR85301633A AR30163385A AR245445A1 AR 245445 A1 AR245445 A1 AR 245445A1 AR 85301633 A AR85301633 A AR 85301633A AR 30163385 A AR30163385 A AR 30163385A AR 245445 A1 AR245445 A1 AR 245445A1
Authority
AR
Argentina
Prior art keywords
aryl
preparation
propanols
acylamido
threo
Prior art date
Application number
AR85301633A
Other languages
English (en)
Spanish (es)
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Application granted granted Critical
Publication of AR245445A1 publication Critical patent/AR245445A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D301/00—Preparation of oxiranes
    • C07D301/02—Synthesis of the oxirane ring
    • C07D301/03—Synthesis of the oxirane ring by oxidation of unsaturated compounds, or of mixtures of unsaturated and saturated compounds
    • C07D301/14—Synthesis of the oxirane ring by oxidation of unsaturated compounds, or of mixtures of unsaturated and saturated compounds with organic peracids, or salts, anhydrides or esters thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/34—Compounds containing oxirane rings with hydrocarbon radicals, substituted by sulphur, selenium or tellurium atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
AR85301633A 1984-09-19 1985-09-17 Procedimiento para la preparacion de cis-1-aril-2-(fluormetil)oxiranos,compuestos asi obtenidos y preparacion de (treo)-1-aril-2-acilamido-3-fluor-1-propanoles utilizando dichos compuestos. AR245445A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/651,980 US4582918A (en) 1984-09-19 1984-09-19 Preparation of intermediates for (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols

Publications (1)

Publication Number Publication Date
AR245445A1 true AR245445A1 (es) 1994-01-31

Family

ID=24615030

Family Applications (1)

Application Number Title Priority Date Filing Date
AR85301633A AR245445A1 (es) 1984-09-19 1985-09-17 Procedimiento para la preparacion de cis-1-aril-2-(fluormetil)oxiranos,compuestos asi obtenidos y preparacion de (treo)-1-aril-2-acilamido-3-fluor-1-propanoles utilizando dichos compuestos.

Country Status (18)

Country Link
US (1) US4582918A (enExample)
EP (1) EP0200739B1 (enExample)
JP (1) JPS62500519A (enExample)
KR (1) KR900001509B1 (enExample)
AR (1) AR245445A1 (enExample)
AT (1) ATE44735T1 (enExample)
AU (1) AU577622B2 (enExample)
CA (1) CA1262553A (enExample)
DE (1) DE3571613D1 (enExample)
DK (1) DK173703B1 (enExample)
ES (1) ES8702339A1 (enExample)
HU (1) HU196198B (enExample)
IE (1) IE58491B1 (enExample)
IL (1) IL76432A (enExample)
NZ (1) NZ213508A (enExample)
SG (1) SG39092G (enExample)
WO (1) WO1986001799A1 (enExample)
ZA (1) ZA857132B (enExample)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4973750A (en) * 1984-09-19 1990-11-27 Schering Corporation Preparation of (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols
DE3543021A1 (de) * 1985-12-05 1987-06-11 Boehringer Mannheim Gmbh Verbesserte verfahren zur herstellung von d-threo-1-(p-methylsulfonylphenyl) -2-dichloracetamido-propandiol-1,3-(thiamphenicol) sowie verwendung geeigneter zwischenprodukte
US5084583A (en) * 1989-10-12 1992-01-28 E. I. Du Pont De Nemours And Company Epoxidation of fluorine containing olefins
IT1249048B (it) 1991-02-21 1995-02-11 Zambon Spa Processo per la preparazione di trans-(5r)-2-ossazoline -2,4,5, trisostituite
US5346828A (en) * 1991-03-27 1994-09-13 Celgene Corporation Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenylpropionic acids using d-threonine aldolase
IL134144A (en) * 1999-02-19 2004-02-08 Akzo Nobel Nv Process for the preparation of a-droxy organic acids
BR0308289A (pt) * 2002-03-08 2005-01-11 Schering Plough Ltd Antibióticos do tipo florfenicol
US20040202762A1 (en) * 2003-04-08 2004-10-14 Ducharme Paul E Smoked nonfibrous casing
US7126005B2 (en) 2003-10-06 2006-10-24 Aurobindo Pharma Limited Process for preparing florfenicol
DE602005012107D1 (de) * 2004-08-13 2009-02-12 Schering Plough Ltd Pharmazeutische formulierungen mit einem antibioti
ES2314724T3 (es) 2004-09-23 2009-03-16 Schering-Plough Ltd. Control de parasitos en animales mediante el uso de nuevos derivados de eter de trifluorometanosulfonanilida oxima.
CA2587495A1 (en) * 2004-11-19 2006-05-26 Schering-Plough Ltd. Control of parasites in animals by the use of parasiticidal 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitrile derivatives
DK1830885T3 (da) * 2004-12-21 2009-01-05 Intervet Int Bv Injicerbar veterinærmedicinsk sammensætning omfattende florfenicol
JP2008545788A (ja) * 2005-06-09 2008-12-18 シェーリング−プラウ・リミテッド Ｎ−［（フェニルオキシ）フェニル］−１，１，１−トリフルオロメタンスルホンアミドおよびｎ−［（フェニルスルファニル）フェニル）］−１，１，１−トリフルオロメタンスルホンアミド誘導体による動物中の寄生生物の制御
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
US7518017B2 (en) 2006-02-17 2009-04-14 Idexx Laboratories Fenicol compounds and methods synthesizing 2-trifluoroacetamido-3-substituted propiophenone compounds
US8084643B2 (en) * 2006-12-13 2011-12-27 Intervet Inc. Water-soluble prodrugs of florfenicol and its analogs
CA2672795A1 (en) * 2006-12-13 2008-06-26 Schering-Plough Ltd. Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof
AR066265A1 (es) * 2007-04-27 2009-08-05 Schering Plough Ltd Compuestos y metodos para mejorar la solubilidad de florfenicol y antibioticos estructuralmente relacionados por medio del uso de ciclodextrinas. composicion. complejo. kit. metodo de tratamiento.
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
SI2182945T1 (sl) 2007-06-27 2015-12-31 E.I. Du Pont De Nemours And Company Metoda za zatiranje škodljivcev pri živalih
PL2217207T3 (pl) * 2007-11-09 2019-05-31 Intervet Int Bv Preparat o szybkim uwalnianiu w postaci stałej, jego przygotowanie i zastosowanie
TWI468407B (zh) 2008-02-06 2015-01-11 Du Pont 中離子農藥
CA2732017A1 (en) * 2008-07-30 2010-02-04 Intervet International B.V. Process for preparing oxazoline-protected aminodiol compounds useful as intermediates to florfenicol
WO2011017347A2 (en) 2009-08-05 2011-02-10 E. I. Du Pont De Nemours And Company Mesoionic pesticides
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
WO2011017334A2 (en) 2009-08-05 2011-02-10 E. I. Du Pont De Nemours And Company Mesoionic pesticides
BRPI1002023A2 (pt) 2010-03-01 2011-10-25 Nanocore Biotecnologia S A forma farmacêutica sólida de dissolução rápida para tratamento de infecções bacterianas
DK2576523T3 (en) 2010-05-27 2016-04-18 Du Pont A crystalline form of 4- [5- [3-chloro-5- (trifluoromethyl) phenyl] -4,5-dihydro-5- (trifluoromethyl) -3-isoxazolyl] -N- [2-oxo-2 - [( 2,2,2-trifluoroethyl) amino] ethyl] - 1-naphthalenecarboxamide
JP5716349B2 (ja) * 2010-10-22 2015-05-13 住友化学株式会社 エポキシアルコール化合物の取得方法、並びにエポキシアルコール化合物及びトリアゾール化合物の製造方法
WO2012087630A1 (en) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Pyridine and pyrimidine compounds for controlling invertebrate
WO2013158422A1 (en) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Heterocyclic compounds for controlling invertebrate pests

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DD83161A (enExample) *
US3849482A (en) * 1967-10-30 1974-11-19 Merck & Co Inc Amine salts of cis-propenylphosphonic acid
LU79970A1 (fr) * 1978-07-13 1980-02-14 Continental Pharma Procede de preparation de derives de 1-phenyl-1-propanol
ES8104203A1 (es) * 1979-02-05 1981-04-16 Schering Corp Un procedimiento para la preparacion de un compuesto d-(treo-1-aril-2-acilamido-3-fluor-1-propanol
US4235892A (en) * 1979-02-05 1980-11-25 Schering Corporation, Patent Dept. 1-Aryl-2-acylamido-3-fluoro-1-propanols, methods for their use as antibacterial agents and compositions useful therefor

Also Published As

Publication number Publication date
US4582918A (en) 1986-04-15
NZ213508A (en) 1989-05-29
DK224086A (da) 1986-05-14
ES547083A0 (es) 1986-12-16
DK173703B1 (da) 2001-07-09
IL76432A0 (en) 1986-01-31
SG39092G (en) 1992-05-22
DE3571613D1 (en) 1989-08-24
DK224086D0 (da) 1986-05-14
AU4809785A (en) 1986-04-08
ZA857132B (en) 1986-05-28
EP0200739A1 (en) 1986-11-12
HUT45243A (en) 1988-06-28
IE58491B1 (en) 1993-09-22
EP0200739B1 (en) 1989-07-19
HU196198B (en) 1988-10-28
WO1986001799A1 (en) 1986-03-27
ES8702339A1 (es) 1986-12-16
AU577622B2 (en) 1988-09-29
IE852296L (en) 1986-03-19
JPH0529216B2 (enExample) 1993-04-28
CA1262553A (en) 1989-10-31
JPS62500519A (ja) 1987-03-05
ATE44735T1 (de) 1989-08-15
IL76432A (en) 1989-02-28
KR870700614A (ko) 1987-12-30
KR900001509B1 (ko) 1990-03-12

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