IL76432A - Cis-1-aryl-2-(fluoromethyl)oxiranes,their preparation and their use as starting materials in the preparation of(threo)-1-aryl-2-acylamino-3-fluoro-1-propanols - Google Patents
Cis-1-aryl-2-(fluoromethyl)oxiranes,their preparation and their use as starting materials in the preparation of(threo)-1-aryl-2-acylamino-3-fluoro-1-propanolsInfo
- Publication number
- IL76432A IL76432A IL76432A IL7643285A IL76432A IL 76432 A IL76432 A IL 76432A IL 76432 A IL76432 A IL 76432A IL 7643285 A IL7643285 A IL 7643285A IL 76432 A IL76432 A IL 76432A
- Authority
- IL
- Israel
- Prior art keywords
- aryl
- preparation
- propanols
- oxiranes
- threo
- Prior art date
Links
- 150000002924 oxiranes Chemical class 0.000 title 1
- 239000007858 starting material Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D301/00—Preparation of oxiranes
- C07D301/02—Synthesis of the oxirane ring
- C07D301/03—Synthesis of the oxirane ring by oxidation of unsaturated compounds, or of mixtures of unsaturated and saturated compounds
- C07D301/14—Synthesis of the oxirane ring by oxidation of unsaturated compounds, or of mixtures of unsaturated and saturated compounds with organic peracids, or salts, anhydrides or esters thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/34—Compounds containing oxirane rings with hydrocarbon radicals, substituted by sulphur, selenium or tellurium atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Epoxy Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/651,980 US4582918A (en) | 1984-09-19 | 1984-09-19 | Preparation of intermediates for (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols |
Publications (2)
Publication Number | Publication Date |
---|---|
IL76432A0 IL76432A0 (en) | 1986-01-31 |
IL76432A true IL76432A (en) | 1989-02-28 |
Family
ID=24615030
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL76432A IL76432A (en) | 1984-09-19 | 1985-09-19 | Cis-1-aryl-2-(fluoromethyl)oxiranes,their preparation and their use as starting materials in the preparation of(threo)-1-aryl-2-acylamino-3-fluoro-1-propanols |
Country Status (18)
Country | Link |
---|---|
US (1) | US4582918A (xx) |
EP (1) | EP0200739B1 (xx) |
JP (1) | JPS62500519A (xx) |
KR (1) | KR900001509B1 (xx) |
AR (1) | AR245445A1 (xx) |
AT (1) | ATE44735T1 (xx) |
AU (1) | AU577622B2 (xx) |
CA (1) | CA1262553A (xx) |
DE (1) | DE3571613D1 (xx) |
DK (1) | DK173703B1 (xx) |
ES (1) | ES8702339A1 (xx) |
HU (1) | HU196198B (xx) |
IE (1) | IE58491B1 (xx) |
IL (1) | IL76432A (xx) |
NZ (1) | NZ213508A (xx) |
SG (1) | SG39092G (xx) |
WO (1) | WO1986001799A1 (xx) |
ZA (1) | ZA857132B (xx) |
Families Citing this family (33)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4973750A (en) * | 1984-09-19 | 1990-11-27 | Schering Corporation | Preparation of (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols |
DE3543021A1 (de) * | 1985-12-05 | 1987-06-11 | Boehringer Mannheim Gmbh | Verbesserte verfahren zur herstellung von d-threo-1-(p-methylsulfonylphenyl) -2-dichloracetamido-propandiol-1,3-(thiamphenicol) sowie verwendung geeigneter zwischenprodukte |
US5084583A (en) * | 1989-10-12 | 1992-01-28 | E. I. Du Pont De Nemours And Company | Epoxidation of fluorine containing olefins |
IT1249048B (it) | 1991-02-21 | 1995-02-11 | Zambon Spa | Processo per la preparazione di trans-(5r)-2-ossazoline -2,4,5, trisostituite |
US5346828A (en) * | 1991-03-27 | 1994-09-13 | Celgene Corporation | Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenylpropionic acids using d-threonine aldolase |
IL134144A (en) * | 1999-02-19 | 2004-02-08 | Akzo Nobel Nv | Process for the preparation of a-droxy organic acids |
CN1649829A (zh) * | 2002-03-08 | 2005-08-03 | 先灵-普劳有限公司 | 新型氟苯尼考类抗生素 |
US20040202762A1 (en) * | 2003-04-08 | 2004-10-14 | Ducharme Paul E | Smoked nonfibrous casing |
US7126005B2 (en) | 2003-10-06 | 2006-10-24 | Aurobindo Pharma Limited | Process for preparing florfenicol |
CN102499928A (zh) | 2004-08-13 | 2012-06-20 | 先灵-普劳有限公司 | 包含抗菌素、三唑和皮质类固醇的药物制剂 |
MX2007003378A (es) | 2004-09-23 | 2007-05-10 | Schering Plough Ltd | Control de parasitos en animales mediante el uso de nuevos derivados de trifluorometansulfonanilida oxima eter. |
WO2006055565A2 (en) * | 2004-11-19 | 2006-05-26 | Schering-Plough Ltd. | Control of parasites in animals by the use of parasiticidal 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitrile derivatives |
AU2005318187B2 (en) * | 2004-12-21 | 2010-12-16 | Intervet International B.V. | Injectable veterinary composition |
JP2008545788A (ja) * | 2005-06-09 | 2008-12-18 | シェーリング−プラウ・リミテッド | N−[(フェニルオキシ)フェニル]−1,1,1−トリフルオロメタンスルホンアミドおよびn−[(フェニルスルファニル)フェニル)]−1,1,1−トリフルオロメタンスルホンアミド誘導体による動物中の寄生生物の制御 |
US8119667B2 (en) * | 2005-12-29 | 2012-02-21 | Schering-Plough Animal Health Corporation | Carbonates of fenicol antibiotics |
US7518017B2 (en) | 2006-02-17 | 2009-04-14 | Idexx Laboratories | Fenicol compounds and methods synthesizing 2-trifluoroacetamido-3-substituted propiophenone compounds |
CA2672586A1 (en) * | 2006-12-13 | 2008-06-26 | Schering-Plough Ltd. | Water-soluble prodrugs of florfenicol and its analogs |
US8044230B2 (en) * | 2006-12-13 | 2011-10-25 | Intervet Inc. | Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof |
AR066265A1 (es) * | 2007-04-27 | 2009-08-05 | Schering Plough Ltd | Compuestos y metodos para mejorar la solubilidad de florfenicol y antibioticos estructuralmente relacionados por medio del uso de ciclodextrinas. composicion. complejo. kit. metodo de tratamiento. |
TWI430995B (zh) | 2007-06-26 | 2014-03-21 | Du Pont | 萘異唑啉無脊椎有害動物控制劑 |
CN101743000A (zh) | 2007-06-27 | 2010-06-16 | 杜邦公司 | 动物虫害控制方法 |
KR20100085162A (ko) * | 2007-11-09 | 2010-07-28 | 인터벳 인터내셔널 비.브이. | 속방성 고체 제형, 제조 및 이의 용도 |
TWI401023B (zh) | 2008-02-06 | 2013-07-11 | Du Pont | 中離子農藥 |
WO2010014566A2 (en) * | 2008-07-30 | 2010-02-04 | Intervet International B.V. | Process for preparing oxazoline-protected aminodiol compounds useful as intermediates to florfenicol |
JP2013501063A (ja) | 2009-08-05 | 2013-01-10 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | メソイオン性殺虫剤 |
UA110924C2 (uk) | 2009-08-05 | 2016-03-10 | Е. І. Дю Пон Де Немур Енд Компані | Мезоіонні пестициди |
UA107804C2 (xx) | 2009-08-05 | 2015-02-25 | Du Pont | Суміші мезоіонних пестицидів |
AU2010279574A1 (en) | 2009-08-05 | 2012-02-09 | E. I. Du Pont De Nemours And Company | Mesoionic pesticides |
BRPI1002023A2 (pt) | 2010-03-01 | 2011-10-25 | Nanocore Biotecnologia S A | forma farmacêutica sólida de dissolução rápida para tratamento de infecções bacterianas |
ES2566402T3 (es) | 2010-05-27 | 2016-04-12 | E. I. Du Pont De Nemours And Company | Forma cristalina de 4-[5-[3-cloro-5-(trifluorometil)fenil]-4,5-dihidro-5-(trifluorometil)-3-isoxazolil]-N-[2-oxo-2-[(2,2,2-trifluoroetil)amino]etil]-1-naftalenocarboxamida |
JP5716349B2 (ja) * | 2010-10-22 | 2015-05-13 | 住友化学株式会社 | エポキシアルコール化合物の取得方法、並びにエポキシアルコール化合物及びトリアゾール化合物の製造方法 |
WO2012087630A1 (en) | 2010-12-20 | 2012-06-28 | E.I. Du Pont De Nemours And Company | Pyridine and pyrimidine compounds for controlling invertebrate |
WO2013158422A1 (en) | 2012-04-17 | 2013-10-24 | E. I. Du Pont De Nemours And Company | Heterocyclic compounds for controlling invertebrate pests |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DD83161A (xx) * | ||||
US3849482A (en) * | 1967-10-30 | 1974-11-19 | Merck & Co Inc | Amine salts of cis-propenylphosphonic acid |
LU79970A1 (fr) * | 1978-07-13 | 1980-02-14 | Continental Pharma | Procede de preparation de derives de 1-phenyl-1-propanol |
US4235892A (en) * | 1979-02-05 | 1980-11-25 | Schering Corporation, Patent Dept. | 1-Aryl-2-acylamido-3-fluoro-1-propanols, methods for their use as antibacterial agents and compositions useful therefor |
ES488154A0 (es) * | 1979-02-05 | 1981-04-16 | Schering Corp | Un procedimiento para la preparacion de un compuesto d-(treo-1-aril-2-acilamido-3-fluor-1-propanol |
-
1984
- 1984-09-19 US US06/651,980 patent/US4582918A/en not_active Expired - Lifetime
-
1985
- 1985-09-17 IE IE229685A patent/IE58491B1/en not_active IP Right Cessation
- 1985-09-17 NZ NZ213508A patent/NZ213508A/xx unknown
- 1985-09-17 KR KR1019860700277A patent/KR900001509B1/ko not_active IP Right Cessation
- 1985-09-17 JP JP60504073A patent/JPS62500519A/ja active Granted
- 1985-09-17 HU HU853894A patent/HU196198B/hu unknown
- 1985-09-17 AU AU48097/85A patent/AU577622B2/en not_active Expired
- 1985-09-17 AR AR85301633A patent/AR245445A1/es active
- 1985-09-17 EP EP85904734A patent/EP0200739B1/en not_active Expired
- 1985-09-17 DE DE8585904734T patent/DE3571613D1/de not_active Expired
- 1985-09-17 ZA ZA857132A patent/ZA857132B/xx unknown
- 1985-09-17 WO PCT/US1985/001753 patent/WO1986001799A1/en active IP Right Grant
- 1985-09-17 AT AT85904734T patent/ATE44735T1/de not_active IP Right Cessation
- 1985-09-18 CA CA000490974A patent/CA1262553A/en not_active Expired
- 1985-09-18 ES ES547083A patent/ES8702339A1/es not_active Expired
- 1985-09-19 IL IL76432A patent/IL76432A/xx not_active IP Right Cessation
-
1986
- 1986-05-14 DK DK198602240A patent/DK173703B1/da not_active IP Right Cessation
-
1992
- 1992-04-07 SG SG390/92A patent/SG39092G/en unknown
Also Published As
Publication number | Publication date |
---|---|
IE58491B1 (en) | 1993-09-22 |
US4582918A (en) | 1986-04-15 |
HUT45243A (en) | 1988-06-28 |
EP0200739B1 (en) | 1989-07-19 |
DK224086A (da) | 1986-05-14 |
ATE44735T1 (de) | 1989-08-15 |
DK224086D0 (da) | 1986-05-14 |
ZA857132B (en) | 1986-05-28 |
IL76432A0 (en) | 1986-01-31 |
AU4809785A (en) | 1986-04-08 |
EP0200739A1 (en) | 1986-11-12 |
NZ213508A (en) | 1989-05-29 |
KR870700614A (ko) | 1987-12-30 |
ES547083A0 (es) | 1986-12-16 |
JPS62500519A (ja) | 1987-03-05 |
SG39092G (en) | 1992-05-22 |
AR245445A1 (es) | 1994-01-31 |
CA1262553A (en) | 1989-10-31 |
KR900001509B1 (ko) | 1990-03-12 |
ES8702339A1 (es) | 1986-12-16 |
DE3571613D1 (en) | 1989-08-24 |
HU196198B (en) | 1988-10-28 |
WO1986001799A1 (en) | 1986-03-27 |
AU577622B2 (en) | 1988-09-29 |
DK173703B1 (da) | 2001-07-09 |
JPH0529216B2 (xx) | 1993-04-28 |
IE852296L (en) | 1986-03-19 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
KB | Patent renewed | ||
KB | Patent renewed | ||
EXP | Patent expired |