ATE44735T1 - Verfahren zur herstellung von (threo)-1-aryl-2acylamido-3-fluoro-1-propanole. - Google Patents
Verfahren zur herstellung von (threo)-1-aryl-2acylamido-3-fluoro-1-propanole.Info
- Publication number
- ATE44735T1 ATE44735T1 AT85904734T AT85904734T ATE44735T1 AT E44735 T1 ATE44735 T1 AT E44735T1 AT 85904734 T AT85904734 T AT 85904734T AT 85904734 T AT85904734 T AT 85904734T AT E44735 T1 ATE44735 T1 AT E44735T1
- Authority
- AT
- Austria
- Prior art keywords
- 2acylamido
- propanols
- threo
- fluoro
- aryl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D301/00—Preparation of oxiranes
- C07D301/02—Synthesis of the oxirane ring
- C07D301/03—Synthesis of the oxirane ring by oxidation of unsaturated compounds, or of mixtures of unsaturated and saturated compounds
- C07D301/14—Synthesis of the oxirane ring by oxidation of unsaturated compounds, or of mixtures of unsaturated and saturated compounds with organic peracids, or salts, anhydrides or esters thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/34—Compounds containing oxirane rings with hydrocarbon radicals, substituted by sulphur, selenium or tellurium atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Epoxy Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/651,980 US4582918A (en) | 1984-09-19 | 1984-09-19 | Preparation of intermediates for (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols |
EP85904734A EP0200739B1 (de) | 1984-09-19 | 1985-09-17 | Verfahren zur herstellung von (threo)-1-aryl-2-acylamido-3-fluoro-1-propanole |
PCT/US1985/001753 WO1986001799A1 (en) | 1984-09-19 | 1985-09-17 | Preparation of (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE44735T1 true ATE44735T1 (de) | 1989-08-15 |
Family
ID=24615030
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT85904734T ATE44735T1 (de) | 1984-09-19 | 1985-09-17 | Verfahren zur herstellung von (threo)-1-aryl-2acylamido-3-fluoro-1-propanole. |
Country Status (18)
Country | Link |
---|---|
US (1) | US4582918A (de) |
EP (1) | EP0200739B1 (de) |
JP (1) | JPS62500519A (de) |
KR (1) | KR900001509B1 (de) |
AR (1) | AR245445A1 (de) |
AT (1) | ATE44735T1 (de) |
AU (1) | AU577622B2 (de) |
CA (1) | CA1262553A (de) |
DE (1) | DE3571613D1 (de) |
DK (1) | DK173703B1 (de) |
ES (1) | ES8702339A1 (de) |
HU (1) | HU196198B (de) |
IE (1) | IE58491B1 (de) |
IL (1) | IL76432A (de) |
NZ (1) | NZ213508A (de) |
SG (1) | SG39092G (de) |
WO (1) | WO1986001799A1 (de) |
ZA (1) | ZA857132B (de) |
Families Citing this family (33)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4973750A (en) * | 1984-09-19 | 1990-11-27 | Schering Corporation | Preparation of (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols |
DE3543021A1 (de) * | 1985-12-05 | 1987-06-11 | Boehringer Mannheim Gmbh | Verbesserte verfahren zur herstellung von d-threo-1-(p-methylsulfonylphenyl) -2-dichloracetamido-propandiol-1,3-(thiamphenicol) sowie verwendung geeigneter zwischenprodukte |
US5084583A (en) * | 1989-10-12 | 1992-01-28 | E. I. Du Pont De Nemours And Company | Epoxidation of fluorine containing olefins |
IT1249048B (it) | 1991-02-21 | 1995-02-11 | Zambon Spa | Processo per la preparazione di trans-(5r)-2-ossazoline -2,4,5, trisostituite |
US5346828A (en) * | 1991-03-27 | 1994-09-13 | Celgene Corporation | Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenylpropionic acids using d-threonine aldolase |
IL134144A (en) * | 1999-02-19 | 2004-02-08 | Akzo Nobel Nv | Process for the preparation of a-droxy organic acids |
EP1487785A2 (de) * | 2002-03-08 | 2004-12-22 | Schering-Plough Ltd. | Neue florfenicol-ähnliche antibiotika |
US20040202762A1 (en) * | 2003-04-08 | 2004-10-14 | Ducharme Paul E | Smoked nonfibrous casing |
US7126005B2 (en) | 2003-10-06 | 2006-10-24 | Aurobindo Pharma Limited | Process for preparing florfenicol |
PT1776109E (pt) * | 2004-08-13 | 2009-03-25 | Schering Plough Ltd | Formulação farmacêutica que compreende um antibiótico, um triazol e um corticosteróide |
BRPI0515917A (pt) | 2004-09-23 | 2008-08-12 | Schering Plough Ltd | controle de parasitas em animais pelo uso de novos derivados de éter de oxima de trifluorometanossulfonanilida |
JP4750126B2 (ja) * | 2004-11-19 | 2011-08-17 | シェーリング−プラウ・リミテッド | 殺寄生虫薬2−フェニル−3−(1h−ピロール−2−イル)アクリロニトリル誘導体の使用による動物における寄生虫の制御 |
PT1830885E (pt) * | 2004-12-21 | 2008-12-22 | Intervet Int Bv | Composição veterinária injectável |
AR054380A1 (es) * | 2005-06-09 | 2007-06-20 | Schering Plough Ltd | Control de parasitos en animales con derivados de n- ((feniloxi) fenil) -1,1,1-trifluorometansulfonamida y de n-(fenilsulfanil) fenil) -1,1,1-trifluorometansulfonamida |
US8119667B2 (en) * | 2005-12-29 | 2012-02-21 | Schering-Plough Animal Health Corporation | Carbonates of fenicol antibiotics |
US7518017B2 (en) | 2006-02-17 | 2009-04-14 | Idexx Laboratories | Fenicol compounds and methods synthesizing 2-trifluoroacetamido-3-substituted propiophenone compounds |
MX2009006282A (es) * | 2006-12-13 | 2009-06-23 | Schering Plough Ltd | Profarmacos solubles en agua de florfenicol y sus analogos. |
US8044230B2 (en) * | 2006-12-13 | 2011-10-25 | Intervet Inc. | Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof |
US20090062397A1 (en) * | 2007-04-27 | 2009-03-05 | Schering-Plough Animal Health Corporation | Compounds and methods for enhancing solubility of florfenicol and structurally-related antibiotics using cyclodextrins |
TWI430995B (zh) | 2007-06-26 | 2014-03-21 | Du Pont | 萘異唑啉無脊椎有害動物控制劑 |
ES2666187T3 (es) | 2007-06-27 | 2018-05-03 | E. I. Du Pont De Nemours And Company | Procedimiento de control de plagas en animales |
CN101909600A (zh) * | 2007-11-09 | 2010-12-08 | 英特维特国际股份有限公司 | 速释固体制剂、其制备及其应用 |
TWI468407B (zh) | 2008-02-06 | 2015-01-11 | Du Pont | 中離子農藥 |
EP2321269B1 (de) * | 2008-07-30 | 2018-09-19 | Intervet International B.V. | Verfahren zur herstellung von als zwischenprodukte für florfenicol geeigneten oxazolingeschützten aminodiolverbindungen |
UA110924C2 (uk) | 2009-08-05 | 2016-03-10 | Е. І. Дю Пон Де Немур Енд Компані | Мезоіонні пестициди |
AU2010279587A1 (en) | 2009-08-05 | 2012-02-09 | E. I. Du Pont De Nemours And Company | Mesoionic pesticides |
UA107804C2 (en) | 2009-08-05 | 2015-02-25 | Du Pont | Mixtures of pesticides mezoionnyh |
EP2461684A2 (de) | 2009-08-05 | 2012-06-13 | E. I. du Pont de Nemours and Company | Mesoionische pestizide |
BRPI1002023A2 (pt) | 2010-03-01 | 2011-10-25 | Nanocore Biotecnologia S A | forma farmacêutica sólida de dissolução rápida para tratamento de infecções bacterianas |
MY156670A (en) | 2010-05-27 | 2016-03-15 | Du Pont | Crystalline form of 4-[5-[3-chloro-5-(trifluoromethly)phenyl]-4,5-dihydro-5-(trifluoromethyl)-3-isoxazolyl]-n-[2-oxo-2-[(2,2,2-trifluoroethyl) amino]ethyl]-1-naphthalenecarboxamide |
JP5716349B2 (ja) * | 2010-10-22 | 2015-05-13 | 住友化学株式会社 | エポキシアルコール化合物の取得方法、並びにエポキシアルコール化合物及びトリアゾール化合物の製造方法 |
WO2012087630A1 (en) | 2010-12-20 | 2012-06-28 | E.I. Du Pont De Nemours And Company | Pyridine and pyrimidine compounds for controlling invertebrate |
WO2013158422A1 (en) | 2012-04-17 | 2013-10-24 | E. I. Du Pont De Nemours And Company | Heterocyclic compounds for controlling invertebrate pests |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DD83161A (de) * | ||||
US3849482A (en) * | 1967-10-30 | 1974-11-19 | Merck & Co Inc | Amine salts of cis-propenylphosphonic acid |
LU79970A1 (fr) * | 1978-07-13 | 1980-02-14 | Continental Pharma | Procede de preparation de derives de 1-phenyl-1-propanol |
ES8104203A1 (es) * | 1979-02-05 | 1981-04-16 | Schering Corp | Un procedimiento para la preparacion de un compuesto d-(treo-1-aril-2-acilamido-3-fluor-1-propanol |
US4235892A (en) * | 1979-02-05 | 1980-11-25 | Schering Corporation, Patent Dept. | 1-Aryl-2-acylamido-3-fluoro-1-propanols, methods for their use as antibacterial agents and compositions useful therefor |
-
1984
- 1984-09-19 US US06/651,980 patent/US4582918A/en not_active Expired - Lifetime
-
1985
- 1985-09-17 EP EP85904734A patent/EP0200739B1/de not_active Expired
- 1985-09-17 JP JP60504073A patent/JPS62500519A/ja active Granted
- 1985-09-17 WO PCT/US1985/001753 patent/WO1986001799A1/en active IP Right Grant
- 1985-09-17 AR AR85301633A patent/AR245445A1/es active
- 1985-09-17 AT AT85904734T patent/ATE44735T1/de not_active IP Right Cessation
- 1985-09-17 DE DE8585904734T patent/DE3571613D1/de not_active Expired
- 1985-09-17 IE IE229685A patent/IE58491B1/en not_active IP Right Cessation
- 1985-09-17 KR KR1019860700277A patent/KR900001509B1/ko not_active IP Right Cessation
- 1985-09-17 AU AU48097/85A patent/AU577622B2/en not_active Expired
- 1985-09-17 HU HU853894A patent/HU196198B/hu unknown
- 1985-09-17 NZ NZ213508A patent/NZ213508A/xx unknown
- 1985-09-17 ZA ZA857132A patent/ZA857132B/xx unknown
- 1985-09-18 CA CA000490974A patent/CA1262553A/en not_active Expired
- 1985-09-18 ES ES547083A patent/ES8702339A1/es not_active Expired
- 1985-09-19 IL IL76432A patent/IL76432A/xx not_active IP Right Cessation
-
1986
- 1986-05-14 DK DK198602240A patent/DK173703B1/da not_active IP Right Cessation
-
1992
- 1992-04-07 SG SG390/92A patent/SG39092G/en unknown
Also Published As
Publication number | Publication date |
---|---|
IL76432A (en) | 1989-02-28 |
DK224086D0 (da) | 1986-05-14 |
AR245445A1 (es) | 1994-01-31 |
HU196198B (en) | 1988-10-28 |
EP0200739A1 (de) | 1986-11-12 |
AU4809785A (en) | 1986-04-08 |
IE58491B1 (en) | 1993-09-22 |
KR900001509B1 (ko) | 1990-03-12 |
ES547083A0 (es) | 1986-12-16 |
JPS62500519A (ja) | 1987-03-05 |
ZA857132B (en) | 1986-05-28 |
DE3571613D1 (en) | 1989-08-24 |
ES8702339A1 (es) | 1986-12-16 |
CA1262553A (en) | 1989-10-31 |
DK173703B1 (da) | 2001-07-09 |
IL76432A0 (en) | 1986-01-31 |
WO1986001799A1 (en) | 1986-03-27 |
IE852296L (en) | 1986-03-19 |
SG39092G (en) | 1992-05-22 |
AU577622B2 (en) | 1988-09-29 |
EP0200739B1 (de) | 1989-07-19 |
KR870700614A (ko) | 1987-12-30 |
US4582918A (en) | 1986-04-15 |
NZ213508A (en) | 1989-05-29 |
HUT45243A (en) | 1988-06-28 |
JPH0529216B2 (de) | 1993-04-28 |
DK224086A (da) | 1986-05-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
UEP | Publication of translation of european patent specification | ||
EELA | Cancelled due to lapse of time |