AR075498A1 - Metodos para la preparacion de arilamidas - Google Patents
Metodos para la preparacion de arilamidasInfo
- Publication number
- AR075498A1 AR075498A1 ARP090105105A ARP090105105A AR075498A1 AR 075498 A1 AR075498 A1 AR 075498A1 AR P090105105 A ARP090105105 A AR P090105105A AR P090105105 A ARP090105105 A AR P090105105A AR 075498 A1 AR075498 A1 AR 075498A1
- Authority
- AR
- Argentina
- Prior art keywords
- catalyst
- methods
- compound
- formula
- arilamids
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/28—Halogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
- C07C25/18—Polycyclic aromatic halogenated hydrocarbons
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C251/72—Hydrazones
- C07C251/82—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to carbon atoms of rings other than six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C43/00—Ethers; Compounds having groups, groups or groups
- C07C43/02—Ethers
- C07C43/18—Ethers having an ether-oxygen atom bound to a carbon atom of a ring other than a six-membered aromatic ring
- C07C43/192—Ethers having an ether-oxygen atom bound to a carbon atom of a ring other than a six-membered aromatic ring containing halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
- C07C49/687—Unsaturated compounds containing a keto groups being part of a ring containing halogen
- C07C49/693—Unsaturated compounds containing a keto groups being part of a ring containing halogen polycyclic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Catalysts (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
La presente solicitud se refiere a métodos para iniciar una reaccion representada por el esquema 1 Q-X + P-C(=O)(NHR)catalizador PC(=O)N-(Q)(R), donde Q es arilo opcionalmente sustituido o heteroarilo opcionalmente sustituido; X es halogeno o un sulfonato; P es un radical orgánico; R es H o un radical orgánico; donde el catalizador comprende cobre y un ligando; que comprende proveer el compuesto de la formula (3) en forma líquida antes de poner en contacto el compuesto de la formula (3) con el catalizador.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US14065008P | 2008-12-24 | 2008-12-24 | |
EP09163256 | 2009-06-19 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR075498A1 true AR075498A1 (es) | 2011-04-06 |
Family
ID=42286925
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP090105105A AR075498A1 (es) | 2008-12-24 | 2009-12-23 | Metodos para la preparacion de arilamidas |
ARP090105106A AR074982A1 (es) | 2008-12-24 | 2009-12-23 | Metodos para la preparacion de fungicidas |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP090105106A AR074982A1 (es) | 2008-12-24 | 2009-12-23 | Metodos para la preparacion de fungicidas |
Country Status (10)
Country | Link |
---|---|
US (3) | US20110257410A1 (es) |
EP (2) | EP2373625B1 (es) |
JP (2) | JP2012513961A (es) |
CN (2) | CN102300850A (es) |
AR (2) | AR075498A1 (es) |
BR (2) | BRPI0923401B1 (es) |
IL (2) | IL213351A0 (es) |
MX (2) | MX2011006425A (es) |
TW (2) | TW201023742A (es) |
WO (2) | WO2010072631A1 (es) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0923401B1 (pt) * | 2008-12-24 | 2021-11-23 | Syngenta Limited | Método para o preparo de aril amidas e composto |
CN102906072B (zh) * | 2010-04-20 | 2014-07-02 | 先正达参股股份有限公司 | 吡唑羧酸酰胺的制备方法 |
EP2560960B1 (en) * | 2010-04-20 | 2014-02-26 | Syngenta Participations AG | Process for the preparation of pyrazole carboxylic acid amides |
BR112012026752B1 (pt) * | 2010-04-20 | 2018-02-06 | Syngenta Participations Ag | Processo para a preparação de amidas do ácido pirazol carboxílico e compostos intermediários assim obtidos |
EP2560957B1 (en) * | 2010-04-20 | 2014-05-07 | Syngenta Participations AG | Process for the preparation of pyrazole carboxylic acid amides |
EP2632901B1 (en) * | 2010-10-27 | 2018-09-12 | Solvay Sa | Process for the preparation of pyrazole-4-carboxamides |
TWI534126B (zh) * | 2011-01-25 | 2016-05-21 | 先正達合夥公司 | 用於製備吡唑羧酸醯胺之方法 |
GB201104203D0 (en) | 2011-03-11 | 2011-04-27 | Syngenta Ltd | Chemical process |
CN105047164B (zh) * | 2015-08-27 | 2017-09-29 | 深圳市华星光电技术有限公司 | 一种灰阶调整方法及装置 |
CN107935930A (zh) * | 2017-12-01 | 2018-04-20 | 浙江工业大学 | 一种1‑甲基‑3‑二氟甲基‑1h‑吡唑‑4‑酰胺衍生物及其制备方法与应用 |
CN111138364A (zh) * | 2018-11-01 | 2020-05-12 | 东莞市东阳光菌阳氢专利农药有限公司 | 一种氟苯醚酰胺的制备方法 |
CN110922285B (zh) * | 2019-12-06 | 2022-08-23 | 上海合全药业股份有限公司 | 一种金属催化一锅法制备芳基伯酰胺的方法 |
WO2023044364A1 (en) | 2021-09-15 | 2023-03-23 | Enko Chem, Inc. | Protoporphyrinogen oxidase inhibitors |
WO2024077487A1 (en) * | 2022-10-11 | 2024-04-18 | Syngenta Crop Protection Ag | Process for the preparation of pyrazole carboxylic acid amides |
Family Cites Families (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5747518A (en) | 1995-04-11 | 1998-05-05 | Mitsui Toatsu Chemicals, Inc. | Substituted thiophene derivative and agricultural and horticultural fungicide containing the same as active ingredient |
US20020173475A1 (en) | 2001-04-16 | 2002-11-21 | Asim Dasgupta | Methods to inhibit viral replication |
CN1266112C (zh) | 2001-04-24 | 2006-07-26 | 麻省理工学院 | 铜-催化的碳-杂原子键和碳-碳键的形成 |
DE10215292A1 (de) | 2002-02-19 | 2003-08-28 | Bayer Cropscience Ag | Disubstitutierte Pyrazolylcarbocanilide |
SI1480955T1 (sl) | 2002-03-05 | 2007-12-31 | Syngenta Participations Ag | O-ciklopropil-karboksanilidi in njihova uporaba kot fungicidi |
US7202367B2 (en) | 2002-05-31 | 2007-04-10 | Rhodia Chimie | Process for arylating or vinylating or alkynating a nucleophilic compound |
EP1509502A1 (fr) * | 2002-05-31 | 2005-03-02 | Rhodia Chimie | Procede de formation d une liaison carbone-carbone ou carbone-heteroatome |
GB0224316D0 (en) | 2002-10-18 | 2002-11-27 | Syngenta Participations Ag | Chemical compounds |
GB0319949D0 (en) * | 2003-08-26 | 2003-09-24 | Univ Strathclyde | Nucleic acid sequence identification |
TW200526626A (en) * | 2003-09-13 | 2005-08-16 | Astrazeneca Ab | Chemical compounds |
AU2005233430B2 (en) * | 2004-04-12 | 2010-11-25 | Eisai R & D Management Co., Ltd. | Process for production of pyrazole-fused ring derivatives |
JP2008540656A (ja) | 2005-05-18 | 2008-11-20 | ワイス | Tpl2キナーゼの3−シアノキノリン阻害物質ならびにそれを製造および使用する方法 |
CA2621228C (en) | 2005-09-02 | 2014-05-27 | Nissan Chemical Industries, Ltd. | Isoxazoline-substituted benzamide compound and pesticide |
CN101979375A (zh) * | 2005-09-16 | 2011-02-23 | 先正达参股股份有限公司 | 酰胺的制备方法 |
GT200600468A (es) * | 2005-10-25 | 2007-06-08 | Nuevos microbiocidas | |
AU2006314825B2 (en) | 2005-11-15 | 2011-11-10 | Syngenta Participations Ag | Process for the production of carboxanilides |
AR058302A1 (es) | 2005-12-12 | 2008-01-30 | Syngenta Participations Ag | Proceso para la preparacion de aminas |
FR2896503B1 (fr) * | 2006-01-23 | 2012-07-13 | Aventis Pharma Sa | Nouveaux derives soufres d'uree cyclique, leur preparation et leur utilisation pharmaceutique comme inhibiteurs de kinases |
EP2001476A4 (en) * | 2006-03-20 | 2010-12-22 | Synta Pharmaceuticals Corp | BENZOIMIDAZOLYL-PARAZINE-BASED COMPOUNDS FOR INFLAMMATION USES AND IMMUNE DISORDERS |
NZ563488A (en) * | 2006-04-19 | 2010-04-30 | Boehringer Ingelheim Int | Dihydrothienopyrimidines for the treatment of inflammatory diseases |
CA2652385A1 (en) * | 2006-06-08 | 2007-12-21 | Eli Lilly And Company | Novel mch receptor antagonists |
ES2392104T3 (es) * | 2006-06-16 | 2012-12-04 | Syngenta Participations Ag | Derivados de carboxamida etenílica útiles como microbiocidas |
DE102006033090A1 (de) | 2006-07-14 | 2008-01-24 | Bayer Cropscience Ag | Verfahren zum Herstellen von Alkylaniliden aus Halogenbenzolderivaten |
US8044049B2 (en) | 2006-08-04 | 2011-10-25 | Takeda Pharmaceutical Company Limited | Fused heterocyclic derivative and use thereof |
AU2007321719B2 (en) | 2006-11-15 | 2013-11-21 | Ym Biosciences Australia Pty Ltd | Inhibitors of kinase activity |
BRPI0923401B1 (pt) * | 2008-12-24 | 2021-11-23 | Syngenta Limited | Método para o preparo de aril amidas e composto |
-
2009
- 2009-12-16 BR BRPI0923401-2A patent/BRPI0923401B1/pt active IP Right Grant
- 2009-12-16 MX MX2011006425A patent/MX2011006425A/es unknown
- 2009-12-16 WO PCT/EP2009/067283 patent/WO2010072631A1/en active Application Filing
- 2009-12-16 CN CN2009801556464A patent/CN102300850A/zh active Pending
- 2009-12-16 US US13/142,084 patent/US20110257410A1/en not_active Abandoned
- 2009-12-16 JP JP2011542773A patent/JP2012513961A/ja active Pending
- 2009-12-16 MX MX2011006426A patent/MX2011006426A/es active IP Right Grant
- 2009-12-16 JP JP2011542774A patent/JP5727381B2/ja active Active
- 2009-12-16 BR BRPI0923527A patent/BRPI0923527A2/pt not_active IP Right Cessation
- 2009-12-16 WO PCT/EP2009/067286 patent/WO2010072632A1/en active Application Filing
- 2009-12-16 US US13/142,110 patent/US8637678B2/en active Active
- 2009-12-16 EP EP09768405.4A patent/EP2373625B1/en not_active Not-in-force
- 2009-12-16 EP EP09768403A patent/EP2370412A1/en not_active Withdrawn
- 2009-12-16 CN CN2009801520087A patent/CN102264705A/zh active Pending
- 2009-12-23 AR ARP090105105A patent/AR075498A1/es not_active Application Discontinuation
- 2009-12-23 TW TW098144403A patent/TW201023742A/zh unknown
- 2009-12-23 TW TW098144401A patent/TW201026647A/zh unknown
- 2009-12-23 AR ARP090105106A patent/AR074982A1/es not_active Application Discontinuation
-
2011
- 2011-06-02 IL IL213351A patent/IL213351A0/en unknown
- 2011-06-02 IL IL213344A patent/IL213344A/en active IP Right Grant
-
2013
- 2013-12-17 US US14/108,885 patent/US9169233B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
JP2012513962A (ja) | 2012-06-21 |
CN102264705A (zh) | 2011-11-30 |
MX2011006425A (es) | 2011-07-20 |
US9169233B2 (en) | 2015-10-27 |
JP2012513961A (ja) | 2012-06-21 |
US20110257410A1 (en) | 2011-10-20 |
EP2373625B1 (en) | 2014-10-08 |
BRPI0923527A2 (pt) | 2016-08-09 |
EP2373625A1 (en) | 2011-10-12 |
IL213351A0 (en) | 2011-07-31 |
TW201023742A (en) | 2010-07-01 |
IL213344A (en) | 2016-07-31 |
US20140107348A1 (en) | 2014-04-17 |
BRPI0923401A2 (pt) | 2015-07-28 |
CN102300850A (zh) | 2011-12-28 |
EP2370412A1 (en) | 2011-10-05 |
US20110263869A1 (en) | 2011-10-27 |
WO2010072631A1 (en) | 2010-07-01 |
AR074982A1 (es) | 2011-03-02 |
MX2011006426A (es) | 2011-07-20 |
JP5727381B2 (ja) | 2015-06-03 |
BRPI0923401B1 (pt) | 2021-11-23 |
WO2010072632A1 (en) | 2010-07-01 |
US8637678B2 (en) | 2014-01-28 |
TW201026647A (en) | 2010-07-16 |
IL213344A0 (en) | 2011-07-31 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |