AR058302A1 - Proceso para la preparacion de aminas - Google Patents

Proceso para la preparacion de aminas

Info

Publication number
AR058302A1
AR058302A1 ARP060105445A ARP060105445A AR058302A1 AR 058302 A1 AR058302 A1 AR 058302A1 AR P060105445 A ARP060105445 A AR P060105445A AR P060105445 A ARP060105445 A AR P060105445A AR 058302 A1 AR058302 A1 AR 058302A1
Authority
AR
Argentina
Prior art keywords
compound
formula
compounds
preparation
precursors
Prior art date
Application number
ARP060105445A
Other languages
English (en)
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of AR058302A1 publication Critical patent/AR058302A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/24—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds
    • C07C209/28—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds by reduction with other reducing agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/62—Preparation of compounds containing amino groups bound to a carbon skeleton by cleaving carbon-to-nitrogen, sulfur-to-nitrogen, or phosphorus-to-nitrogen bonds, e.g. hydrolysis of amides, N-dealkylation of amines or quaternary ammonium compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/23—Preparation of halogenated hydrocarbons by dehalogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/30—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by a Diels-Alder synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/35—Preparation of halogenated hydrocarbons by reactions not affecting the number of carbon or of halogen atoms in the reaction
    • C07C17/354—Preparation of halogenated hydrocarbons by reactions not affecting the number of carbon or of halogen atoms in the reaction by hydrogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/04—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups
    • C07C209/06—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms
    • C07C209/10—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms with formation of amino groups bound to carbon atoms of six-membered aromatic rings or from amines having nitrogen atoms bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/24—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds
    • C07C209/26—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds by reduction with hydrogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/68—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton
    • C07C209/70—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton by reduction of unsaturated amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/57—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton
    • C07C211/60—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton containing a ring other than a six-membered aromatic ring forming part of at least one of the condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/57—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton
    • C07C211/61—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton with at least one of the condensed ring systems formed by three or more rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/18—Polycyclic aromatic halogenated hydrocarbons
    • C07C25/22—Polycyclic aromatic halogenated hydrocarbons with condensed rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/24—Halogenated aromatic hydrocarbons with unsaturated side chains
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/09—Geometrical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/56—Ring systems containing bridged rings
    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/60—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Catalysts (AREA)

Abstract

La presente se refiere a un nuevo proceso para la preparacion del compuesto de la formula general (1) en donde R1 y R2 son independientemente H o alquilo C1-6, el cual comprende tratar con un agente de reduccion o bien un compuesto de la formula general (2); en donde R1 y R2 poseen los significados proporcionados para e compuesto de la formula (1), R3 es H o alquilo C1-4 y Ph es fenilo, o un compuesto de la formula general (3) en donde R1, R2, R3 y Ph poseen los significados proporcionados para el compuesto de la formula (2), siendo el agente de reduccion efectivo para escindir el resto bencilo Ph-CH(R3)- del resto bencilamino PhCH(R3)NH- en el compuesto de la formula (2) o en el compuesto de la formula (3) para dejar un grupo amino y, además, en el caso del compuesto de la formula (3), para reducir tanto el enlace 2,3-doble como el enlace doble que une el resto R1R2C- a la posicion 9 del anillo benzonorborneno a enlaces simples. Ésta también se refiere a procesos para la preparacion de los compuestos (2) y (3) y sus precursores y a los compuestos (2) y (3) en sí mismos y a ciertos de sus precursores, los cuales son nuevos compuestos. Los compuestos (1) son utiles para la preparacion de varias benzonorbornen-5-il- amidas de ácido heterociclil-carboxílico fungicidas.
ARP060105445A 2005-12-12 2006-12-11 Proceso para la preparacion de aminas AR058302A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05027072 2005-12-12
EP06008248 2006-04-21

Publications (1)

Publication Number Publication Date
AR058302A1 true AR058302A1 (es) 2008-01-30

Family

ID=37946810

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060105445A AR058302A1 (es) 2005-12-12 2006-12-11 Proceso para la preparacion de aminas

Country Status (21)

Country Link
US (1) US7781615B2 (es)
EP (5) EP1963251B1 (es)
JP (1) JP5144533B2 (es)
KR (1) KR101364220B1 (es)
CN (3) CN104151132B (es)
AR (1) AR058302A1 (es)
AU (1) AU2006326289B2 (es)
BR (1) BRPI0619629B1 (es)
CA (1) CA2631973C (es)
CL (2) CL2010000015A1 (es)
CR (1) CR10052A (es)
DK (1) DK1963251T3 (es)
EA (1) EA014275B1 (es)
EC (1) ECSP088525A (es)
EG (1) EG25547A (es)
ES (1) ES2391904T3 (es)
IL (3) IL191760A (es)
IN (1) IN2015DN00818A (es)
PL (1) PL1963251T3 (es)
TW (1) TWI396676B (es)
WO (1) WO2007068417A2 (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2006326289B2 (en) * 2005-12-12 2011-12-22 Syngenta Participations Ag Process for the preparation of amines
HUE048086T2 (hu) 2007-09-20 2020-05-28 Bayer Cropscience Lp Fungicid törzset és legalább egy további fungicidet tartalmazó kombinációk
CA2728887A1 (en) 2008-07-04 2010-01-07 Basf Se Fungicidal mixtures comprising substituted 1-methylpyrazol-4-ylcarboxanilides
MY150841A (en) 2008-10-27 2014-02-28 Syngenta Participations Ag Process for the preparation of benzonorbornenes
BRPI0923527A2 (pt) 2008-12-24 2016-08-09 Syngenta Ltd métodos de preparo de fungicidas
JP6153864B2 (ja) * 2010-04-20 2017-06-28 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト ピラゾールカルボン酸アミドの調製方法
AR083876A1 (es) 2010-11-15 2013-03-27 Bayer Cropscience Ag 5-halogenopirazolcarboxamidas
RU2493145C1 (ru) * 2012-10-02 2013-09-20 Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Волгоградский государственный технический университет" (ВолгГТУ) Способ получения 2-(аминоалкил)-3-(аминофенил)бицикло[2.2.1]гептанов
EP2975939B1 (en) 2013-03-14 2020-08-05 Dow AgroSciences LLC Broadleaf crop control with 6-arylpicoline carboxylic acids, 2-arylpyrimidine carboxylic acids, or salts or esters thereof
US11560384B2 (en) 2017-05-04 2023-01-24 University Of Utah Research Foundation Benzonorbornadiene derivatives and reactions thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1086978A (en) * 1965-09-21 1967-10-11 Shionogi & Co Improvements in or relating to the preparation of 7-oxobenzonorbornene derivatives
JPH075487B2 (ja) 1985-11-14 1995-01-25 住友化学工業株式会社 １―ブロモ―２―クロロ―４―フルオロベンゼンの製造法
US7223879B2 (en) 1998-07-10 2007-05-29 Massachusetts Institute Of Technology Ligands for metals and improved metal-catalyzed processes based thereon
JPWO2002076922A1 (ja) * 2001-03-16 2004-07-15 出光興産株式会社 芳香族アミノ化合物の製造方法
JP4219622B2 (ja) * 2002-06-11 2009-02-04 独立行政法人科学技術振興機構 ベンザイン化合物の新規製造法
US7531559B2 (en) * 2002-08-22 2009-05-12 Syngenta Crop Protection, Inc. Fungicidal 1,2,3 triazole derivatives
GB0224316D0 (en) * 2002-10-18 2002-11-27 Syngenta Participations Ag Chemical compounds
AU2006326289B2 (en) * 2005-12-12 2011-12-22 Syngenta Participations Ag Process for the preparation of amines

Also Published As

Publication number Publication date
IL191760A0 (en) 2008-12-29
WO2007068417A2 (en) 2007-06-21
IL218350A0 (en) 2012-04-30
TW200800854A (en) 2008-01-01
EA200870038A1 (ru) 2008-10-30
CN101360703A (zh) 2009-02-04
EP1963251A2 (en) 2008-09-03
EP2316813B1 (en) 2013-04-03
US20090221856A1 (en) 2009-09-03
US7781615B2 (en) 2010-08-24
CN101360703B (zh) 2012-07-18
CL2010000015A1 (es) 2010-07-02
IL218351A (en) 2014-05-28
KR20080077011A (ko) 2008-08-20
WO2007068417A3 (en) 2007-10-04
EP2316815A1 (en) 2011-05-04
CN102516086A (zh) 2012-06-27
AU2006326289B2 (en) 2011-12-22
EP2316814A1 (en) 2011-05-04
TWI396676B (zh) 2013-05-21
CN104151132B (zh) 2016-07-06
EP2316809B1 (en) 2014-06-18
CR10052A (es) 2008-09-17
BRPI0619629B1 (pt) 2016-03-01
BRPI0619629A2 (pt) 2011-10-04
EP2316813A1 (en) 2011-05-04
CN104151132A (zh) 2014-11-19
CA2631973A1 (en) 2007-06-21
AU2006326289A1 (en) 2007-06-21
IL191760A (en) 2014-05-28
EA014275B1 (ru) 2010-10-29
PL1963251T3 (pl) 2013-01-31
KR101364220B1 (ko) 2014-02-21
EP2316809A1 (en) 2011-05-04
ECSP088525A (es) 2008-07-30
CL2012000114A1 (es) 2012-08-31
EG25547A (en) 2012-02-15
IN2015DN00818A (es) 2015-07-10
JP2009518346A (ja) 2009-05-07
ES2391904T3 (es) 2012-11-30
DK1963251T3 (da) 2012-11-26
CA2631973C (en) 2015-02-03
JP5144533B2 (ja) 2013-02-13
CN102516086B (zh) 2014-10-22
IL218351A0 (en) 2012-04-30
EP1963251B1 (en) 2012-08-15

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