AR051596A1 - Compuestos heterociclicos condensados nitrogenados como inhibidores de la actividad del receptor canabinoide 1; composiciones farmaceuticas que los contienen y su empleo en la preparacion de medicamentos para el tratamiento de trastornos alimentarios - Google Patents

Compuestos heterociclicos condensados nitrogenados como inhibidores de la actividad del receptor canabinoide 1; composiciones farmaceuticas que los contienen y su empleo en la preparacion de medicamentos para el tratamiento de trastornos alimentarios

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Publication number
AR051596A1
AR051596A1 ARP050104440A ARP050104440A AR051596A1 AR 051596 A1 AR051596 A1 AR 051596A1 AR P050104440 A ARP050104440 A AR P050104440A AR P050104440 A ARP050104440 A AR P050104440A AR 051596 A1 AR051596 A1 AR 051596A1
Authority
AR
Argentina
Prior art keywords
alkyl
halogen
substituted
alkoxy
hydroxyl
Prior art date
Application number
ARP050104440A
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English (en)
Spanish (es)
Original Assignee
Irm Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Irm Llc filed Critical Irm Llc
Publication of AR051596A1 publication Critical patent/AR051596A1/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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ARP050104440A 2004-10-26 2005-10-24 Compuestos heterociclicos condensados nitrogenados como inhibidores de la actividad del receptor canabinoide 1; composiciones farmaceuticas que los contienen y su empleo en la preparacion de medicamentos para el tratamiento de trastornos alimentarios AR051596A1 (es)

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US62250804P 2004-10-26 2004-10-26
US67267005P 2005-04-18 2005-04-18

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AR051596A1 true AR051596A1 (es) 2007-01-24

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ARP050104440A AR051596A1 (es) 2004-10-26 2005-10-24 Compuestos heterociclicos condensados nitrogenados como inhibidores de la actividad del receptor canabinoide 1; composiciones farmaceuticas que los contienen y su empleo en la preparacion de medicamentos para el tratamiento de trastornos alimentarios

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US (2) US8158634B2 (https=)
EP (1) EP1807429A4 (https=)
JP (2) JP2008518016A (https=)
KR (1) KR100919524B1 (https=)
CN (2) CN102241680A (https=)
AR (1) AR051596A1 (https=)
AU (2) AU2005299421B2 (https=)
BR (1) BRPI0517015A (https=)
CA (2) CA2581225C (https=)
EC (1) ECSP077421A (https=)
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IN (1) IN2007DN02514A (https=)
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MX (1) MX2007004936A (https=)
NO (1) NO20072352L (https=)
PE (1) PE20060599A1 (https=)
RU (1) RU2431635C2 (https=)
TN (1) TNSN07161A1 (https=)
TW (1) TW200630096A (https=)
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