AR018634A1 - Derivados de benzo(b)tiepin-1,1,-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos, procedimiento para la preparacion de medicamentos y su empleo para la preparacion de medicamentos. - Google Patents

Derivados de benzo(b)tiepin-1,1,-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos, procedimiento para la preparacion de medicamentos y su empleo para la preparacion de medicamentos.

Info

Publication number
AR018634A1
AR018634A1 ARP990102716A ARP990102716A AR018634A1 AR 018634 A1 AR018634 A1 AR 018634A1 AR P990102716 A ARP990102716 A AR P990102716A AR P990102716 A ARP990102716 A AR P990102716A AR 018634 A1 AR018634 A1 AR 018634A1
Authority
AR
Argentina
Prior art keywords
preparation
acid radical
procedure
medicines
alkyl
Prior art date
Application number
ARP990102716A
Other languages
English (en)
Spanish (es)
Original Assignee
Gompel Marie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gompel Marie filed Critical Gompel Marie
Publication of AR018634A1 publication Critical patent/AR018634A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D337/00—Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02—Seven-membered rings
    • C07D337/06—Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/08—Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/04—Drugs for disorders of the urinary system for urolithiasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06086—Dipeptides with the first amino acid being basic
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08G—MACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
    • C08G65/00—Macromolecular compounds obtained by reactions forming an ether link in the main chain of the macromolecule
    • C08G65/02—Macromolecular compounds obtained by reactions forming an ether link in the main chain of the macromolecule from cyclic ethers by opening of the heterocyclic ring
    • C08G65/32—Polymers modified by chemical after-treatment
    • C08G65/329—Polymers modified by chemical after-treatment with organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Polymers & Plastics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ARP990102716A 1998-06-10 1999-06-08 Derivados de benzo(b)tiepin-1,1,-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos, procedimiento para la preparacion de medicamentos y su empleo para la preparacion de medicamentos. AR018634A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19825804A DE19825804C2 (de) 1998-06-10 1998-06-10 1,4-Benzothiepin-1,1-dioxidderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
AR018634A1 true AR018634A1 (es) 2001-11-28

Family

ID=7870440

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP990102716A AR018634A1 (es) 1998-06-10 1999-06-08 Derivados de benzo(b)tiepin-1,1,-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos, procedimiento para la preparacion de medicamentos y su empleo para la preparacion de medicamentos.
ARP990102715A AR018633A1 (es) 1998-06-10 1999-06-08 Derivados de benzo(b)tiepin-1,1-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos y su empleo

Family Applications After (1)

Application Number Title Priority Date Filing Date
ARP990102715A AR018633A1 (es) 1998-06-10 1999-06-08 Derivados de benzo(b)tiepin-1,1-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos y su empleo

Country Status (25)

Country Link
US (1) US6387944B1 (enExample)
EP (2) EP1086092B1 (enExample)
JP (2) JP4374426B2 (enExample)
KR (2) KR100681721B1 (enExample)
CN (2) CN1127497C (enExample)
AR (2) AR018634A1 (enExample)
AT (2) ATE227715T1 (enExample)
AU (2) AU753275B2 (enExample)
BR (2) BR9912188B1 (enExample)
CA (2) CA2334775C (enExample)
CZ (2) CZ297989B6 (enExample)
DE (3) DE19825804C2 (enExample)
DK (2) DK1086092T3 (enExample)
ES (2) ES2182535T3 (enExample)
HU (2) HU229761B1 (enExample)
ID (2) ID28695A (enExample)
IL (1) IL140078A (enExample)
NO (1) NO327075B1 (enExample)
NZ (1) NZ508681A (enExample)
PL (2) PL196074B1 (enExample)
PT (2) PT1086092E (enExample)
RU (2) RU2215001C2 (enExample)
TR (2) TR200003634T2 (enExample)
WO (2) WO1999064410A1 (enExample)
ZA (2) ZA200007061B (enExample)

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CA2431983C (en) * 2000-12-21 2010-06-08 Aventis Pharma Deutschland Gmbh Novel 1,2-diphenylazetidinones, processes for their preparation, medicaments comprising these compounds and their use for treating impaired lipid metabolism
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TWI871392B (zh) 2019-12-04 2025-02-01 瑞典商艾爾比瑞歐公司 苯并噻(二)氮呯(benzothia(di)azepine)化合物及其作為膽酸調節劑之用途
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JP2023549226A (ja) 2020-11-12 2023-11-22 アルビレオ エービー 進行性家族性肝内胆汁うっ滞症（ｐｆｉｃ）を処置するためのオデビキシバット
KR20230117393A (ko) 2020-12-04 2023-08-08 알비레오 에이비 벤조티아(디)아제핀 화합물 및 담즙산 조절제로서의용도
TW202313579A (zh) 2021-06-03 2023-04-01 瑞典商艾爾比瑞歐公司 苯并噻(二)氮呯(benzothia(di)azepine)化合物及其作為膽酸調節劑之用途
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JP2025521736A (ja) 2022-07-05 2025-07-10 アルビレオ・アクチボラグ ベンゾチア（ジ）アゼピン化合物及び胆汁酸モジュレータとしてのそれらの使用
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BR9508916A (pt) * 1994-09-13 1997-12-30 Monsanto Co "Novas benzotiepinas tendo atividade como inibidores de transporte do ácido biliar ileal e absorção de taurocolato"
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US6096780A (en) * 1998-08-20 2000-08-01 Takeda Chemical Industries, Ltd. Quaternary ammonium salts and their use

Also Published As

Publication number Publication date
NO20006251L (no) 2001-02-07
WO1999064409A2 (de) 1999-12-16
CA2334773C (en) 2009-05-26
DE59903411D1 (de) 2002-12-19
PL196057B1 (pl) 2007-11-30
JP2002517490A (ja) 2002-06-18
AU753275B2 (en) 2002-10-10
JP4374426B2 (ja) 2009-12-02
EP1086092B1 (de) 2002-11-13
HK1039490A1 (en) 2002-04-26
CN1305469A (zh) 2001-07-25
WO1999064410A1 (de) 1999-12-16
CZ20004592A3 (cs) 2001-04-11
ID28695A (id) 2001-06-28
ATE227715T1 (de) 2002-11-15
PT1086113E (pt) 2004-06-30
ZA200007060B (en) 2001-07-18
US6387944B1 (en) 2002-05-14
ES2182535T3 (es) 2003-03-01
EP1086092A1 (de) 2001-03-28
PT1086092E (pt) 2003-03-31
HUP0102554A3 (en) 2002-12-28
DK1086113T3 (da) 2004-05-24
EP1086113B1 (de) 2004-02-11
HUP0102554A1 (hu) 2001-10-28
NZ508681A (en) 2002-06-28
HU228570B1 (en) 2013-04-29
IL140078A0 (en) 2002-02-10
JP2002517491A (ja) 2002-06-18
DE59908522D1 (de) 2004-03-18
BR9911123B1 (pt) 2010-12-14
DE19825804A1 (de) 1999-12-16
ATE259372T1 (de) 2004-02-15
HUP0102256A1 (hu) 2001-12-28
AR018633A1 (es) 2001-11-28
CA2334773A1 (en) 1999-12-16
BR9912188A (pt) 2001-04-10
CN1152039C (zh) 2004-06-02
IL140078A (en) 2004-08-31
JP3374129B2 (ja) 2003-02-04
AU752633B2 (en) 2002-09-26
CN1127497C (zh) 2003-11-12
RU2220141C2 (ru) 2003-12-27
KR100681721B1 (ko) 2007-02-15
CA2334775C (en) 2009-10-13
KR20010052682A (ko) 2001-06-25
TR200003634T2 (tr) 2001-06-21
PL196074B1 (pl) 2007-12-31
ES2215387T3 (es) 2004-10-01
HUP0102256A3 (en) 2002-04-29
CZ20004591A3 (cs) 2001-04-11
BR9912188B1 (pt) 2010-12-14
WO1999064409A3 (de) 2000-03-02
AU4501999A (en) 1999-12-30
TR200003632T2 (tr) 2001-04-20
ID26876A (id) 2001-02-15
BR9911123A (pt) 2006-01-03
HU229761B1 (hu) 2014-06-30
CN1305487A (zh) 2001-07-25
CZ297925B6 (cs) 2007-05-02
DE19825804C2 (de) 2000-08-24
NO327075B1 (no) 2009-04-20
CZ297989B6 (cs) 2007-05-16
HK1036799A1 (en) 2002-01-18
ZA200007061B (en) 2001-07-18
NO20006251D0 (no) 2000-12-08
KR100562184B1 (ko) 2006-03-20
PL345901A1 (en) 2002-01-14
EP1086113A2 (de) 2001-03-28
RU2215001C2 (ru) 2003-10-27
KR20010052701A (ko) 2001-06-25
DK1086092T3 (da) 2003-03-10
PL344827A1 (en) 2001-11-19
CA2334775A1 (en) 1999-12-16
AU4503199A (en) 1999-12-30

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