AR012181A1 - Un derivado de pirimidina, procedimientos para prepararlo, una composicion farmaceutica que lo comprende, y un compuesto util como intermediario parapreparar dicho derivado de pirimidina. - Google Patents

Un derivado de pirimidina, procedimientos para prepararlo, una composicion farmaceutica que lo comprende, y un compuesto util como intermediario parapreparar dicho derivado de pirimidina.

Info

Publication number
AR012181A1
AR012181A1 ARP980101380A ARP980101380A AR012181A1 AR 012181 A1 AR012181 A1 AR 012181A1 AR P980101380 A ARP980101380 A AR P980101380A AR P980101380 A ARP980101380 A AR P980101380A AR 012181 A1 AR012181 A1 AR 012181A1
Authority
AR
Argentina
Prior art keywords
methyl
hydrogen
substituted
formula
pirimidine
Prior art date
Application number
ARP980101380A
Other languages
English (en)
Spanish (es)
Original Assignee
Yuhan Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yuhan Corp filed Critical Yuhan Corp
Publication of AR012181A1 publication Critical patent/AR012181A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ARP980101380A 1997-03-27 1998-03-26 Un derivado de pirimidina, procedimientos para prepararlo, una composicion farmaceutica que lo comprende, y un compuesto util como intermediario parapreparar dicho derivado de pirimidina. AR012181A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR19970010862 1997-03-27
KR19970010863 1997-03-27

Publications (1)

Publication Number Publication Date
AR012181A1 true AR012181A1 (es) 2000-09-27

Family

ID=26632616

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP980101380A AR012181A1 (es) 1997-03-27 1998-03-26 Un derivado de pirimidina, procedimientos para prepararlo, una composicion farmaceutica que lo comprende, y un compuesto util como intermediario parapreparar dicho derivado de pirimidina.

Country Status (21)

Country Link
US (1) US6352993B1 (instruction)
EP (1) EP1015444B1 (instruction)
JP (1) JP3176379B2 (instruction)
KR (1) KR100278857B1 (instruction)
CN (1) CN1118464C (instruction)
AR (1) AR012181A1 (instruction)
AT (1) ATE241613T1 (instruction)
AU (1) AU720385B2 (instruction)
BR (1) BR9808070A (instruction)
CA (1) CA2284795C (instruction)
DE (1) DE69815126T2 (instruction)
DK (1) DK1015444T3 (instruction)
ES (1) ES2200324T3 (instruction)
HU (1) HUP0000851A3 (instruction)
IN (1) IN188411B (instruction)
PT (1) PT1015444E (instruction)
RU (1) RU2203894C2 (instruction)
TR (1) TR199902383T2 (instruction)
TW (1) TW542831B (instruction)
UY (1) UY24938A1 (instruction)
WO (1) WO1998043968A1 (instruction)

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US7211590B2 (en) 2002-08-01 2007-05-01 Nitromed, Inc. Nitrosated proton pump inhibitors, compositions and methods of use
WO2005009980A1 (en) * 2003-07-22 2005-02-03 Neurogen Corporation Substituted pyridin-2-ylamine analogues
AU2004283751B2 (en) * 2003-10-24 2011-05-19 Exelixis, Inc. p70S6 kinase modulators and method of use
KR20060099524A (ko) 2003-11-03 2006-09-19 아스트라제네카 아베 무증상 위식도 역류의 치료를 위한 이미다조[1,2-a]피리딘유도체
KR101122376B1 (ko) * 2005-03-09 2012-03-26 주식회사유한양행 신규의 5,6-다이메틸피리미딘 유도체 및 그의 제조방법
JP2009511548A (ja) * 2005-10-14 2009-03-19 ノイロサーチ アクティーゼルスカブ 新規ピリミジン−2,4−ジアミン誘導体及び小コンダクタンスのカルシウム依存性カリウムチャネルのモジュレーターとしてのこれらの使用
JP4946482B2 (ja) 2007-02-08 2012-06-06 船井電機株式会社 緩衝用梱包材及びtv受像機の緩衝用梱包材
US8367684B2 (en) * 2007-06-13 2013-02-05 Valeant Pharmaceuticals International Derivatives of 4-(N-azacycloalkyl) anilides as potassium channel modulators
WO2010016490A1 (ja) 2008-08-05 2010-02-11 第一三共株式会社 イミダゾピリジン-2-オン誘導体
GB0908394D0 (en) 2009-05-15 2009-06-24 Univ Leuven Kath Novel viral replication inhibitors
GB0913636D0 (en) 2009-08-05 2009-09-16 Univ Leuven Kath Novel viral replication inhibitors
MX2013005478A (es) 2010-11-15 2013-08-29 Univ Leuven Kath Compuestos heterociclicos condensados antivirales.
MX337477B (es) 2011-02-25 2016-03-07 Yuhan Corp Derivados de diaminopiridina y procesos para su preparacion.
CA2864825C (en) * 2012-02-17 2021-01-26 Abbvie Inc. Diaminopyrimidines useful as inhibitors of the human respiratory syncytial virus (rsv)
US9309271B2 (en) 2012-05-29 2016-04-12 Momentive Performance Materials Gmbh Preparation of isocyanato silanes
MA38208B1 (fr) 2012-11-21 2021-12-31 Ptc Therapeutics Inc Inhibiteurs de bmi-1 pyrimidines inversés substitués
US10035801B2 (en) 2013-03-13 2018-07-31 Genentech, Inc. Pyrazolo compounds and uses thereof
TWI692477B (zh) * 2013-08-30 2020-05-01 美商Ptc治療公司 經取代嘧啶bmi-1抑制劑
JP6507157B2 (ja) * 2013-10-07 2019-04-24 カドモン コーポレイション,リミティド ライアビリティ カンパニー Rhoキナーゼ阻害剤
WO2015076800A1 (en) 2013-11-21 2015-05-28 Ptc Therapeutics, Inc. Substituted pyridine and pyrazine bmi-1 inhibitors
US10370360B2 (en) 2014-10-22 2019-08-06 The Board Of Regents Of The University Of Texas System Small-molecule inhibitors targeting discoidin domain receptor 1 and uses thereof
CN105669642B (zh) * 2014-11-19 2020-06-09 江苏天士力帝益药业有限公司 一种盐酸洛氟普啶的制备方法
PL3397622T3 (pl) * 2016-01-04 2022-07-04 ObsEva S.A. Jednoczesne podawanie alfa-aminoestrowej pochodnej hydroksypropylotiazolidynokarboksyamidu i środka tokolitycznego
EP3606915A1 (de) * 2017-04-05 2020-02-12 Bayer CropScience Aktiengesellschaft 2-amino-5-oxyalkyl-pyrimidinderivate und deren verwendung zur bekämpfung unerwünschten pflanzenwachstums
EP3836932A2 (en) 2018-08-17 2021-06-23 PTC Therapeutics, Inc. Method for treating pancreatic cancer
CN114685369B (zh) * 2022-05-17 2024-02-02 河南省科学院高新技术研究中心 一种利用离子液体制备1-甲基-1,2,3,4-四氢异喹啉的方法

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KR0144833B1 (ko) 1992-12-28 1998-07-15 김태훈 신규의 퀴나졸린 유도체 및 그의 제조방법
WO1995005363A1 (en) * 1993-08-12 1995-02-23 Astra Aktiebolag Amidine derivatives with nitric oxide synthetase activities
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ES2165052T3 (es) 1996-05-04 2002-03-01 Yuhan Corp Procedimiento para la preparacion de derivados de pirimidina.

Also Published As

Publication number Publication date
ES2200324T3 (es) 2004-03-01
EP1015444A1 (en) 2000-07-05
JP3176379B2 (ja) 2001-06-18
CN1251586A (zh) 2000-04-26
TW542831B (en) 2003-07-21
AU720385B2 (en) 2000-06-01
IN188411B (instruction) 2002-09-21
HUP0000851A1 (hu) 2001-04-28
DE69815126T2 (de) 2004-04-08
TR199902383T2 (xx) 2000-06-21
ATE241613T1 (de) 2003-06-15
UY24938A1 (es) 2001-01-31
CN1118464C (zh) 2003-08-20
HK1026418A1 (en) 2000-12-15
KR19980080789A (ko) 1998-11-25
KR100278857B1 (ko) 2001-01-15
JP2000513014A (ja) 2000-10-03
HUP0000851A3 (en) 2002-04-29
EP1015444B1 (en) 2003-05-28
CA2284795C (en) 2004-01-20
AU6523998A (en) 1998-10-22
BR9808070A (pt) 2000-03-08
DK1015444T3 (da) 2003-08-18
WO1998043968A1 (en) 1998-10-08
PT1015444E (pt) 2003-10-31
US6352993B1 (en) 2002-03-05
DE69815126D1 (de) 2003-07-03
RU2203894C2 (ru) 2003-05-10
CA2284795A1 (en) 1998-10-08

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