CO5590934A2 - Procedimiento de preparacion de derivados de equinocandina - Google Patents
Procedimiento de preparacion de derivados de equinocandinaInfo
- Publication number
- CO5590934A2 CO5590934A2 CO04055277A CO04055277A CO5590934A2 CO 5590934 A2 CO5590934 A2 CO 5590934A2 CO 04055277 A CO04055277 A CO 04055277A CO 04055277 A CO04055277 A CO 04055277A CO 5590934 A2 CO5590934 A2 CO 5590934A2
- Authority
- CO
- Colombia
- Prior art keywords
- equinocandina
- preparation procedure
- derivatives preparation
- derivatives
- dihydrochloride
- Prior art date
Links
- 239000003814 drug Substances 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
1.- La invención se refiere a un procedimiento de preparación de compuestos de fórmula (I): en la que R es tal como se ha definido en la memoria descriptiva así como sus sales, intermedios, la aplicación del dihidrocloruro como fármaco y las composiciones farmacéuticas que los contienen.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0116230A FR2833596B1 (fr) | 2001-12-14 | 2001-12-14 | Procede de preparation de derives d'echinocandine |
Publications (1)
Publication Number | Publication Date |
---|---|
CO5590934A2 true CO5590934A2 (es) | 2005-12-30 |
Family
ID=8870520
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CO04055277A CO5590934A2 (es) | 2001-12-14 | 2004-06-11 | Procedimiento de preparacion de derivados de equinocandina |
Country Status (29)
Country | Link |
---|---|
US (3) | US20070105760A1 (es) |
EP (1) | EP1456229B1 (es) |
JP (1) | JP4510461B2 (es) |
KR (1) | KR20040066167A (es) |
CN (2) | CN100584859C (es) |
AR (1) | AR037827A1 (es) |
AT (1) | ATE441662T1 (es) |
AU (1) | AU2002364991B9 (es) |
BR (1) | BR0214937A (es) |
CA (1) | CA2469918A1 (es) |
CO (1) | CO5590934A2 (es) |
CY (1) | CY1110694T1 (es) |
DE (1) | DE60233589D1 (es) |
DK (1) | DK1456229T3 (es) |
EA (1) | EA007964B1 (es) |
ES (1) | ES2333784T3 (es) |
FR (1) | FR2833596B1 (es) |
HK (2) | HK1071900A1 (es) |
HU (1) | HUP0402602A3 (es) |
IL (1) | IL162385A0 (es) |
MX (1) | MXPA04005484A (es) |
NO (1) | NO20042640L (es) |
NZ (1) | NZ533864A (es) |
PL (1) | PL371763A1 (es) |
PT (1) | PT1456229E (es) |
SI (1) | SI1456229T1 (es) |
TW (1) | TWI322820B (es) |
WO (1) | WO2003054001A2 (es) |
ZA (1) | ZA200404631B (es) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2833596B1 (fr) * | 2001-12-14 | 2005-02-18 | Aventis Pharma Sa | Procede de preparation de derives d'echinocandine |
TW200826957A (en) * | 2006-10-16 | 2008-07-01 | Teva Gyogyszergyar Zartkoruen Mukodo Reszvenytarsasag | Purification processes for echinocandin-type compounds |
FR2921060B1 (fr) * | 2007-09-14 | 2012-06-15 | Novexel | Nouveau procede de preparation d'une piperidine disubsituee et nouveaux intermediaires |
FR2936798B1 (fr) * | 2008-10-03 | 2012-09-28 | Novexel | Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens. |
FR2937034B1 (fr) * | 2008-10-10 | 2012-11-23 | Novexel | Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens |
FR2936951B1 (fr) * | 2008-10-10 | 2010-12-03 | Novexel | Nouvelles combinaisons de composes heterocycliques azotes antibacteriens avec d'autres composes antibacteriens et leur utilisation comme medicaments |
CN101928670B (zh) | 2009-09-24 | 2012-02-22 | 上海天伟生物制药有限公司 | 一种抗生素的高产菌株及其制备方法和用途 |
CN102659930B (zh) * | 2012-03-30 | 2014-04-23 | 上海天伟生物制药有限公司 | 一种高纯度环肽类物质的晶体及其制备方法和用途 |
CN102627689B (zh) * | 2012-03-30 | 2014-08-06 | 上海天伟生物制药有限公司 | 一种环肽类化合物的水合物及其制备方法和用途 |
CN102627688B (zh) * | 2012-03-30 | 2014-12-31 | 上海天伟生物制药有限公司 | 一种高纯度环肽化合物及其制备方法和用途 |
EP3464319A4 (en) * | 2014-10-07 | 2020-02-26 | Alaparthi, Lakshmi Prasad | INTERMEDIATES AND PROCESSES FOR THE PREPARATION OF ANIDULAFUNGIN |
CN112646854B (zh) * | 2020-12-11 | 2022-10-11 | 浙江工业大学 | 一种棘白菌素b合成培养基及应用 |
CN115785226A (zh) * | 2021-09-09 | 2023-03-14 | 上海天伟生物制药有限公司 | 一种棘白菌素药物杂质及其制备、纯化方法和应用 |
Family Cites Families (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4293484A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | Derivatives of A-30912H nucleus |
US5207710A (en) * | 1988-09-29 | 1993-05-04 | Collagen Corporation | Method for improving implant fixation |
US5539122A (en) * | 1989-05-23 | 1996-07-23 | Abbott Laboratories | Retroviral protease inhibiting compounds |
US5386009A (en) * | 1990-03-19 | 1995-01-31 | Merck & Co. Inc. | Lipopeptide derivatives |
CA2091663C (en) * | 1992-03-19 | 2007-10-30 | Frederick Joseph Burkhardt | Cyclic peptide antifungal agents and process for preparation thereof |
DE69435105D1 (de) * | 1993-08-09 | 2008-08-07 | Sod Conseils Rech Applic | Derivate therapeutischer Peptide |
JP3107691B2 (ja) * | 1993-12-03 | 2000-11-13 | 株式会社東芝 | 半導体記憶装置及びその製造方法 |
ATE223226T1 (de) * | 1994-09-16 | 2002-09-15 | Merck & Co Inc | Azazyklohexapeptid-verbindungen |
US5646111A (en) * | 1995-04-07 | 1997-07-08 | Eli Lilly And Company | Cyclic peptide antifungal Agents |
US5652213A (en) * | 1995-05-26 | 1997-07-29 | Eli Lilly And Company | Cyclic peptide antifungal agents |
US5852213A (en) * | 1996-07-10 | 1998-12-22 | American Cyanamid Company | Mercaptoketones and mercaptoalcohols and a process for their preparation |
US6207710B1 (en) * | 1996-11-22 | 2001-03-27 | Elan Pharmaceuticals, Inc. | Compounds for inhibiting β-amyloid peptide release and/or its synthesis |
UA72200C2 (uk) * | 1997-12-10 | 2005-02-15 | Авентіс Фарма С.А. | Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція |
FR2794746B1 (fr) * | 1999-06-09 | 2002-12-06 | Hoechst Marion Roussel Inc | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques |
FR2794747B1 (fr) * | 1999-06-09 | 2004-04-16 | Hoechst Marion Roussel Inc | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques |
US7166572B1 (en) * | 1999-07-27 | 2007-01-23 | Aventis Pharma Deutschland Gmbh | Cyclohexapeptide compounds, processes for their production and their use as a pharmaceutical |
FR2833596B1 (fr) * | 2001-12-14 | 2005-02-18 | Aventis Pharma Sa | Procede de preparation de derives d'echinocandine |
-
2001
- 2001-12-14 FR FR0116230A patent/FR2833596B1/fr not_active Expired - Fee Related
-
2002
- 2002-12-12 AU AU2002364991A patent/AU2002364991B9/en not_active Ceased
- 2002-12-12 BR BR0214937-0A patent/BR0214937A/pt not_active Application Discontinuation
- 2002-12-12 NZ NZ533864A patent/NZ533864A/xx not_active IP Right Cessation
- 2002-12-12 PL PL02371763A patent/PL371763A1/xx not_active Application Discontinuation
- 2002-12-12 SI SI200230861T patent/SI1456229T1/sl unknown
- 2002-12-12 DE DE60233589T patent/DE60233589D1/de not_active Expired - Lifetime
- 2002-12-12 PT PT02805374T patent/PT1456229E/pt unknown
- 2002-12-12 HU HU0402602A patent/HUP0402602A3/hu unknown
- 2002-12-12 CA CA002469918A patent/CA2469918A1/fr not_active Abandoned
- 2002-12-12 CN CN02824928A patent/CN100584859C/zh not_active Expired - Fee Related
- 2002-12-12 WO PCT/FR2002/004308 patent/WO2003054001A2/fr active Application Filing
- 2002-12-12 US US11/591,898 patent/US20070105760A1/en not_active Abandoned
- 2002-12-12 MX MXPA04005484A patent/MXPA04005484A/es active IP Right Grant
- 2002-12-12 AT AT02805374T patent/ATE441662T1/de active
- 2002-12-12 EP EP02805374A patent/EP1456229B1/fr not_active Expired - Lifetime
- 2002-12-12 DK DK02805374T patent/DK1456229T3/da active
- 2002-12-12 JP JP2003554717A patent/JP4510461B2/ja not_active Expired - Fee Related
- 2002-12-12 KR KR10-2004-7009121A patent/KR20040066167A/ko active IP Right Grant
- 2002-12-12 EA EA200400806A patent/EA007964B1/ru not_active IP Right Cessation
- 2002-12-12 ES ES02805374T patent/ES2333784T3/es not_active Expired - Lifetime
- 2002-12-12 CN CNB2005101156130A patent/CN1326872C/zh not_active Expired - Fee Related
- 2002-12-13 AR ARP020104846A patent/AR037827A1/es active IP Right Grant
- 2002-12-13 TW TW091136168A patent/TWI322820B/zh not_active IP Right Cessation
- 2002-12-24 IL IL16238502A patent/IL162385A0/xx unknown
-
2004
- 2004-06-10 ZA ZA200404631A patent/ZA200404631B/en unknown
- 2004-06-11 CO CO04055277A patent/CO5590934A2/es not_active Application Discontinuation
- 2004-06-14 US US10/867,070 patent/US7148322B2/en not_active Expired - Fee Related
- 2004-06-23 NO NO20042640A patent/NO20042640L/no not_active Application Discontinuation
-
2005
- 2005-06-08 HK HK05104783.8A patent/HK1071900A1/xx not_active IP Right Cessation
-
2006
- 2006-07-13 HK HK06107828A patent/HK1087720A1/xx not_active IP Right Cessation
-
2009
- 2009-12-01 CY CY20091101267T patent/CY1110694T1/el unknown
-
2010
- 2010-07-06 US US12/830,941 patent/US20100273977A1/en not_active Abandoned
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Application granted | ||
FD | Application lapsed |