ZA949664B - Imidazopyridines - Google Patents

Imidazopyridines

Info

Publication number
ZA949664B
ZA949664B ZA949664A ZA949664A ZA949664B ZA 949664 B ZA949664 B ZA 949664B ZA 949664 A ZA949664 A ZA 949664A ZA 949664 A ZA949664 A ZA 949664A ZA 949664 B ZA949664 B ZA 949664B
Authority
ZA
South Africa
Prior art keywords
imidazopyridines
Prior art date
Application number
ZA949664A
Other languages
English (en)
Inventor
Werner Mederski
Dieter Dorsch
Matthias Osswald
Norbert Beier
Pierre Schelling
Klaus-Otto Minck
Ingeborg Lues
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of ZA949664B publication Critical patent/ZA949664B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA949664A 1993-12-06 1994-12-05 Imidazopyridines ZA949664B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4341453A DE4341453A1 (de) 1993-12-06 1993-12-06 Imidazopyridine

Publications (1)

Publication Number Publication Date
ZA949664B true ZA949664B (en) 1995-08-15

Family

ID=6504241

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA949664A ZA949664B (en) 1993-12-06 1994-12-05 Imidazopyridines

Country Status (16)

Country Link
US (1) US5532276A (hu)
EP (1) EP0657452A1 (hu)
JP (1) JPH07196656A (hu)
KR (1) KR950018006A (hu)
CN (1) CN1109056A (hu)
AU (1) AU7919094A (hu)
CA (1) CA2137213A1 (hu)
CZ (1) CZ304694A3 (hu)
DE (1) DE4341453A1 (hu)
HU (1) HUT72595A (hu)
NO (1) NO944689L (hu)
PL (1) PL306127A1 (hu)
RU (1) RU94042907A (hu)
SK (1) SK149294A3 (hu)
TW (1) TW294665B (hu)
ZA (1) ZA949664B (hu)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5798364A (en) * 1992-03-26 1998-08-25 Merck Patent Gesellschaft Mit Beschrankter Haftung Imidazopyridines
US6348380B1 (en) * 2000-08-25 2002-02-19 Micron Technology, Inc. Use of dilute steam ambient for improvement of flash devices
ES2334990T3 (es) * 2002-02-14 2010-03-18 Pharmacia Corporation Piridinonas sustituidas como moduladores de p38 map quinasa.
DE60307483T2 (de) * 2002-08-07 2007-07-05 Novartis Ag Organische verbindungen als mittel zur behandlung von aldosteronbedingten zuständen
EP1608317B1 (en) 2003-03-25 2012-09-26 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
US7579357B2 (en) 2003-08-13 2009-08-25 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
US7678909B1 (en) 2003-08-13 2010-03-16 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
US7169926B1 (en) 2003-08-13 2007-01-30 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
JP2007505121A (ja) 2003-09-08 2007-03-08 武田薬品工業株式会社 ジペプチジルぺプチダーゼ阻害剤
US7732446B1 (en) 2004-03-11 2010-06-08 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
CN102127057A (zh) 2004-03-15 2011-07-20 武田药品工业株式会社 二肽基肽酶抑制剂
EP1753730A1 (en) 2004-06-04 2007-02-21 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
WO2006019965A2 (en) 2004-07-16 2006-02-23 Takeda San Diego, Inc. Dipeptidyl peptidase inhibitors
KR20070055563A (ko) 2004-08-23 2007-05-30 와이어쓰 혈전증 및 심혈관 질병의 치료에 유용한 플라스미노겐활성화제 억제제 타입-1(pai-1)의 조절제로서의옥사졸로-나프틸 산
WO2006023864A1 (en) * 2004-08-23 2006-03-02 Wyeth Pyrrolo-naphthyl acids as pai-1 inhibitors
RU2007106869A (ru) * 2004-08-23 2008-09-27 Вайет (Us) Тиазол-нафтиловые кислоты как ингибиторы ингибитора активации плазминогена-1
JP2008524331A (ja) 2004-12-21 2008-07-10 武田薬品工業株式会社 ジペプチジルペプチダーゼ阻害剤
ZA200802857B (en) 2005-09-14 2009-09-30 Takeda Pharmaceutical Dipeptidyl peptidase inhibitors for treating diabetes
KR101368988B1 (ko) 2005-09-16 2014-02-28 다케다 야쿠힌 고교 가부시키가이샤 디펩티딜 펩티다제 억제제
WO2007112347A1 (en) 2006-03-28 2007-10-04 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
US8324383B2 (en) 2006-09-13 2012-12-04 Takeda Pharmaceutical Company Limited Methods of making polymorphs of benzoate salt of 2-[[6-[(3R)-3-amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]-benzonitrile
TW200838536A (en) 2006-11-29 2008-10-01 Takeda Pharmaceutical Polymorphs of succinate salt of 2-[6-(3-amino-piperidin-1-yl)-3-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethy]-4-fluor-benzonitrile and methods of use therefor
US8093236B2 (en) 2007-03-13 2012-01-10 Takeda Pharmaceuticals Company Limited Weekly administration of dipeptidyl peptidase inhibitors
JP5627453B2 (ja) * 2008-03-31 2014-11-19 株式会社レナサイエンス プラスミノーゲンアクチベーターインヒビター−1阻害剤
ES2874063T3 (es) * 2009-03-31 2021-11-04 Renascience Inc Inhibidor del inhibidor-1 del activador del plasminógeno
US10092537B2 (en) 2013-04-15 2018-10-09 Renascience Co., Ltd. Use for PAI-1 inhibitor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL94390A (en) * 1989-05-30 1996-03-31 Merck & Co Inc The 6-membered trans-nitrogen-containing heterocycles are compressed with imidazo and pharmaceutical preparations containing them
DE4110019C2 (de) * 1991-03-27 2000-04-13 Merck Patent Gmbh Imidazopyridine, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zubereitungen
US5332750A (en) * 1991-09-04 1994-07-26 Merck Patent Gesellschaft Mit Beschrankter Haftung 1,2-dihydro-2-oxopyridines
DE4141788A1 (de) * 1991-12-18 1993-06-24 Merck Patent Gmbh Imidazopyridine
DE4208304A1 (de) * 1992-03-16 1993-09-23 Merck Patent Gmbh 2-oxochinolinderivate
DE4211474A1 (de) * 1992-04-06 1993-10-07 Merck Patent Gmbh Imidazopyridine
DE4305602A1 (de) * 1992-06-17 1993-12-23 Merck Patent Gmbh Imidazopyridine
DE4225835A1 (de) * 1992-08-05 1994-02-10 Merck Patent Gmbh Verfahren zur Herstellung von Imidazopyridinen
DE4242459A1 (de) * 1992-12-16 1994-06-23 Merck Patent Gmbh Imidazopyridine

Also Published As

Publication number Publication date
EP0657452A1 (de) 1995-06-14
JPH07196656A (ja) 1995-08-01
CA2137213A1 (en) 1995-06-07
HU9403451D0 (en) 1995-02-28
HUT72595A (en) 1996-05-28
RU94042907A (ru) 1996-10-20
AU7919094A (en) 1995-06-15
CN1109056A (zh) 1995-09-27
TW294665B (hu) 1997-01-01
US5532276A (en) 1996-07-02
NO944689L (no) 1995-06-07
SK149294A3 (en) 1995-07-11
KR950018006A (ko) 1995-07-22
NO944689D0 (no) 1994-12-05
PL306127A1 (en) 1995-06-12
CZ304694A3 (en) 1995-08-16
DE4341453A1 (de) 1995-06-08

Similar Documents

Publication Publication Date Title
HU9403364D0 (en) Imidazopyridine
ZA939433B (en) Imidazopyridines
DE69400639D1 (en) Rehydratationsgetraenk
DE69401926D1 (en) Hydroxamsäurederivate
ZA949664B (en) Imidazopyridines
DE69405713D1 (en) Carbonylierungsverfahren
HU9401692D0 (en) Imidazopyridines
ZA942543B (en) Tetrohydro beta-carbolines
DE59409705D1 (en) 3-methoxy-2-phenyl-acrylsäuremethylester
ZA932459B (en) Imidazopyridines
DE59408644D1 (en) Jacquardmaschine
EP0730584A4 (en) 3-ACYLAMINOBENZODIAZEPINE
DE59408733D1 (en) Metallhalogenidentladungslampe
ZA937875B (en) Imidazopyridines
HUT69872A (en) Reaper-thresher
DE59410065D1 (en) 3-methoxy-2-phenyl-acrylsäuremethylester
DE69425743D1 (en) Faserreaktive anthrachinon-farbstoffe
GB9406735D0 (en) Drill-mate
DE59407310D1 (en) Phenylazotriazolopyridinfarbstoffe
AU122479S (en) Label-printer
GB9318883D0 (en) Godiver
ZA931368B (en) Sulphonylbenzyl-substituted imidazopyridines
DE69327259D1 (en) Signalmetrikabschätzer
ZA94990B (en) New imidazopyridines
IL119547A0 (en) Imidazopyridine compounds