ZA934388B - Polymer-bound paclitaxel derivatives - Google Patents

Polymer-bound paclitaxel derivatives

Info

Publication number
ZA934388B
ZA934388B ZA934388A ZA934388A ZA934388B ZA 934388 B ZA934388 B ZA 934388B ZA 934388 A ZA934388 A ZA 934388A ZA 934388 A ZA934388 A ZA 934388A ZA 934388 B ZA934388 B ZA 934388B
Authority
ZA
South Africa
Prior art keywords
phe
gly
leu
ala
beta
Prior art date
Application number
ZA934388A
Other languages
English (en)
Inventor
Nicola Mongelli
Francesco Angelucci
Enrico Pesenti
Antoninio Suarato
Giovanni Biasoli
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of ZA934388B publication Critical patent/ZA934388B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/58—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. poly[meth]acrylate, polyacrylamide, polystyrene, polyvinylpyrrolidone, polyvinylalcohol or polystyrene sulfonic acid resin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Epoxy Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Analysing Materials By The Use Of Radiation (AREA)
ZA934388A 1992-06-19 1993-06-18 Polymer-bound paclitaxel derivatives ZA934388B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929213077A GB9213077D0 (en) 1992-06-19 1992-06-19 Polymerbound taxol derivatives

Publications (1)

Publication Number Publication Date
ZA934388B true ZA934388B (en) 1994-08-29

Family

ID=10717411

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA934388A ZA934388B (en) 1992-06-19 1993-06-18 Polymer-bound paclitaxel derivatives

Country Status (25)

Country Link
US (4) US5362831A (fi)
EP (1) EP0600062B1 (fi)
JP (1) JP3693340B2 (fi)
KR (1) KR100281606B1 (fi)
CN (1) CN1041281C (fi)
AT (1) ATE205725T1 (fi)
AU (2) AU659750B2 (fi)
CA (1) CA2112482A1 (fi)
CZ (1) CZ62094A3 (fi)
DE (1) DE69330776T2 (fi)
ES (1) ES2164663T3 (fi)
FI (1) FI940733A (fi)
GB (1) GB9213077D0 (fi)
HU (2) HUT67914A (fi)
IL (1) IL106023A (fi)
MX (1) MX9303598A (fi)
MY (1) MY109213A (fi)
NZ (1) NZ253116A (fi)
PL (1) PL173898B1 (fi)
RU (1) RU2130462C1 (fi)
SG (1) SG49248A1 (fi)
TW (1) TW266201B (fi)
UA (1) UA39926C2 (fi)
WO (1) WO1994000156A1 (fi)
ZA (1) ZA934388B (fi)

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