ZA793293B - (di)-16-phenoxy and 16-substituted phenoxy-9-keto prostatrienoic acid derivatives and processes for the production thereof - Google Patents

(di)-16-phenoxy and 16-substituted phenoxy-9-keto prostatrienoic acid derivatives and processes for the production thereof

Info

Publication number
ZA793293B
ZA793293B ZA793293A ZA793293A ZA793293B ZA 793293 B ZA793293 B ZA 793293B ZA 793293 A ZA793293 A ZA 793293A ZA 793293 A ZA793293 A ZA 793293A ZA 793293 B ZA793293 B ZA 793293B
Authority
ZA
South Africa
Prior art keywords
phenoxy
keto
processes
production
acid derivatives
Prior art date
Application number
ZA793293A
Other languages
English (en)
Inventor
G Garay
A Van Horn
J Edwards
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Priority to IE1294/79A priority Critical patent/IE48656B1/en
Publication of ZA793293B publication Critical patent/ZA793293B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/582—Recycling of unreacted starting or intermediate materials

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ZA793293A 1978-07-10 1979-07-03 (di)-16-phenoxy and 16-substituted phenoxy-9-keto prostatrienoic acid derivatives and processes for the production thereof ZA793293B (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IE1294/79A IE48656B1 (en) 1978-07-10 1979-08-08 (di)-16-phenoxy-and 16-substituted phenoxy-9-keto prostatrienoic acid derivatives and processes for the production thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/922,957 US4178457A (en) 1978-07-10 1978-07-10 (dl)-16-Phenoxy- and 16-substituted phenoxy-9-keto prostatrienoic acid derivatives and processes for the production thereof

Publications (1)

Publication Number Publication Date
ZA793293B true ZA793293B (en) 1981-02-25

Family

ID=25447871

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA793293A ZA793293B (en) 1978-07-10 1979-07-03 (di)-16-phenoxy and 16-substituted phenoxy-9-keto prostatrienoic acid derivatives and processes for the production thereof

Country Status (26)

Country Link
US (1) US4178457A (en:Method)
EP (1) EP0008003B1 (en:Method)
JP (1) JPS5513282A (en:Method)
KR (1) KR890002773B1 (en:Method)
AT (1) ATE2427T1 (en:Method)
AU (1) AU527516B2 (en:Method)
CA (1) CA1149802A (en:Method)
CS (1) CS209927B2 (en:Method)
DD (1) DD146179A5 (en:Method)
DE (2) DE2964709D1 (en:Method)
DK (1) DK157753C (en:Method)
ES (1) ES482330A1 (en:Method)
FI (1) FI69061C (en:Method)
FR (1) FR2430939A1 (en:Method)
GB (1) GB2025413B (en:Method)
HK (1) HK41384A (en:Method)
HU (1) HU184185B (en:Method)
IT (1) IT1121462B (en:Method)
MY (1) MY8500576A (en:Method)
NO (4) NO150836C (en:Method)
NZ (1) NZ190924A (en:Method)
PL (4) PL120632B1 (en:Method)
SG (1) SG82483G (en:Method)
SU (1) SU1031407A3 (en:Method)
YU (3) YU41870B (en:Method)
ZA (1) ZA793293B (en:Method)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4328245A (en) * 1981-02-13 1982-05-04 Syntex (U.S.A.) Inc. Carbonate diester solutions of PGE-type compounds
US4358603A (en) * 1981-04-16 1982-11-09 Syntex (U.S.A.) Inc. Acetal stabilized prostaglandin compositions
US4409239A (en) * 1982-01-21 1983-10-11 Syntex (U.S.A.) Inc. Propylene glycol diester solutions of PGE-type compounds
US4600785A (en) * 1983-12-22 1986-07-15 Syntex (U.S.A.) Inc. Processes and intermediates for making 16-phenoxy and 16-substituted phenoxy-prostatrienoic acid derivatives
US4804787A (en) * 1983-12-22 1989-02-14 Syntex (U.S.A.) Inc. Processes and intermediates for making 16-phenoxy and 16-substituted phenoxy-prostatrienoic acid derivatives
US4912235A (en) * 1983-12-22 1990-03-27 Syntex (U.S.A.) Inc. Processes and intermediates for making 16-phenoxy- and 16-substituted phenoxy-prostatrienoic acid derivatives and their stereoisomers
DE3414509A1 (de) * 1984-04-13 1985-10-24 Schering AG, 1000 Berlin und 4709 Bergkamen Neue 9-halogen-prostaglandine
US4618696A (en) * 1984-07-31 1986-10-21 Syntex (U.S.A.) Inc. 9-oxo-15α-hydroxy-16-phenoxy and 16-substituted phenoxy 17,18,19,20-tetranorprosta-4,5,13,(E)-trienoates
US5057621A (en) * 1984-07-31 1991-10-15 Syntex (U.S.A.) Inc. 11-substituted-16-phenoxy and 16-substituted phenoxy-prostatrienoic acid derivatives
US4792617A (en) * 1984-07-31 1988-12-20 Syntex (U.S.A.) Inc. 11-substituted-16-phenoxy and 16-substituted phenoxy-prostatrienioc acid derivatives
ES8607921A1 (es) * 1984-07-31 1986-06-16 Syntex Inc Procedimiento para preparar derivados de acidos 11-sustitui-dos-16-fenoxi y 16-fenoxi sustituido-prostatrienoicos
US4778904A (en) * 1985-09-13 1988-10-18 Syntex (U.S.A.) Inc. Intermediates for making 16-phenoxy- and 16-(substituted phenoxy)-prostatrienoic acid derivatives
EP0248999A3 (en) * 1986-04-11 1988-03-16 Syntex (U.S.A.) Inc. Uses of enprostil-type prostaglandins in regulating fat and carbohydrate metabolism
US4755531A (en) * 1986-08-11 1988-07-05 Syntex (U.S.A.) Inc. Thiol esters of 4,5-allenyl prostaglandins and use thereof as antigastric secretion agents
GB8625321D0 (en) * 1986-10-22 1986-11-26 Glaxo Group Ltd Chemical compounds
US4689419A (en) * 1986-11-14 1987-08-25 G. D. Searle & Co. Novel intermediate compounds in a process for producing 16-phenoxy- and 16-substituted phenoxy-9-keto-prostatrienoic acid derivatives
US6103765A (en) * 1997-07-09 2000-08-15 Androsolutions, Inc. Methods for treating male erectile dysfunction
AU742787B2 (en) 1997-07-09 2002-01-10 Androsolutions, Inc. Improved methods and compositions for treating male erectile dysfunction
US20020172693A1 (en) 2000-03-31 2002-11-21 Delong Michell Anthony Compositions and methods for treating hair loss using non-naturally occurring prostaglandins
US20020037914A1 (en) 2000-03-31 2002-03-28 Delong Mitchell Anthony Compositions and methods for treating hair loss using C16-C20 aromatic tetrahydro prostaglandins
US20020013294A1 (en) 2000-03-31 2002-01-31 Delong Mitchell Anthony Cosmetic and pharmaceutical compositions and methods using 2-decarboxy-2-phosphinico derivatives
US8966971B2 (en) * 2008-07-28 2015-03-03 Ford Global Technologies, Llc Vehicle engine with fluid measuring system
US8623918B2 (en) 2008-10-29 2014-01-07 Novaer Holdings, Inc. Amino acid salts of prostaglandins
EP2349242B1 (en) * 2008-10-29 2018-12-05 Novaer Holdings, Inc. Amino acid salts of prostaglandins
US8722739B2 (en) 2008-10-29 2014-05-13 Novaer Holdings, Inc. Amino acid salts of prostaglandins
US20110293549A1 (en) 2009-02-03 2011-12-01 Athena Cosmetics, Inc. Composition, method and kit for enhancing hair

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES449162A1 (es) * 1975-06-23 1977-12-16 Syntex Inc Un procedimiento para la preparacion de un compuesto racemi-co u 8r-antimerico.

Also Published As

Publication number Publication date
NO152212B (no) 1985-05-13
YU168579A (en) 1983-02-28
IT7968428A0 (it) 1979-07-09
MY8500576A (en) 1985-12-31
DE2927715C2 (en:Method) 1987-08-27
NO792283L (no) 1980-01-11
JPS5513282A (en) 1980-01-30
PL121778B1 (en) 1982-05-31
AU4864179A (en) 1980-02-07
GB2025413B (en) 1982-07-28
FI792149A7 (fi) 1980-01-11
YU44553B (en) 1990-08-31
HU184185B (en) 1984-07-30
EP0008003B1 (en) 1983-02-09
YU44554B (en) 1990-08-31
SG82483G (en) 1984-08-03
YU73686A (en) 1986-12-31
NO840258L (no) 1980-01-11
PL120633B1 (en) 1982-03-31
GB2025413A (en) 1980-01-23
DE2964709D1 (en) 1983-03-17
FR2430939A1 (fr) 1980-02-08
YU73586A (en) 1986-12-31
CA1149802A (en) 1983-07-12
AU527516B2 (en) 1983-03-10
NO152211B (no) 1985-05-13
DE2927715A1 (de) 1980-01-24
EP0008003A1 (en) 1980-02-20
ATE2427T1 (de) 1983-03-15
FI69061B (fi) 1985-08-30
DK157753C (da) 1990-07-09
NO152211C (no) 1985-08-21
NO152296C (no) 1985-09-04
NO840256L (no) 1980-01-11
NO150836C (no) 1985-01-09
FR2430939B1 (en:Method) 1981-08-14
NO150836B (no) 1984-09-17
NO152296B (no) 1985-05-28
NO840257L (no) 1980-01-11
NZ190924A (en) 1980-11-28
US4178457A (en) 1979-12-11
FI69061C (fi) 1985-12-10
CS209927B2 (en) 1981-12-31
PL217001A1 (en:Method) 1980-03-24
PL120632B1 (en) 1982-03-31
NO152212C (no) 1985-08-21
HK41384A (en) 1984-05-18
DK288879A (da) 1980-01-11
KR890002773B1 (ko) 1989-07-28
DK157753B (da) 1990-02-12
IT1121462B (it) 1986-04-02
SU1031407A3 (ru) 1983-07-23
PL120604B1 (en) 1982-03-31
JPS6210227B2 (en:Method) 1987-03-05
YU41870B (en) 1988-02-29
ES482330A1 (es) 1980-08-16
DD146179A5 (de) 1981-01-28

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