ZA200609237B - CXCR1 and CXCR2 chemokine antagonists - Google Patents
CXCR1 and CXCR2 chemokine antagonistsInfo
- Publication number
- ZA200609237B ZA200609237B ZA200609237A ZA200609237A ZA200609237B ZA 200609237 B ZA200609237 B ZA 200609237B ZA 200609237 A ZA200609237 A ZA 200609237A ZA 200609237 A ZA200609237 A ZA 200609237A ZA 200609237 B ZA200609237 B ZA 200609237B
- Authority
- ZA
- South Africa
- Prior art keywords
- cxcr1
- chemokine antagonists
- cxcr2 chemokine
- cxcr2
- antagonists
- Prior art date
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- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/36—Nitrogen atoms
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EP (1) | EP1745032B1 (xx) |
JP (2) | JP2007537272A (xx) |
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AU (1) | AU2005245399A1 (xx) |
CA (1) | CA2565519A1 (xx) |
IL (1) | IL179162A0 (xx) |
MX (1) | MXPA06013118A (xx) |
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PL2076502T3 (pl) | 2006-06-08 | 2011-09-30 | Lilly Co Eli | Podstawione karboksyamidy jako antagoniści receptorów metabotropowych grupy I |
CA2664359A1 (en) * | 2006-09-26 | 2008-04-03 | Case Western Reserve University | Cytokine signaling |
JP2010510291A (ja) * | 2006-11-23 | 2010-04-02 | ノバルティス アーゲー | CXCR2アンタゴニストとしての5−スルファニルメチル−ピラゾロ[1,5−a]ピリミジン−7−オール |
MX2009005174A (es) * | 2006-11-23 | 2009-05-25 | Novartis Ag | Derivados de 5-sulfanilmetil-[1,2,4]triazol[1,5-a]pirimidin-7-ol como antagonistas de cxcr2. |
EP2116530B1 (en) * | 2007-02-26 | 2012-11-14 | Santen Pharmaceutical Co., Ltd | Novel pyrrole derivative having ureide group and aminocarbonyl group as substituents |
WO2009026248A2 (en) * | 2007-08-17 | 2009-02-26 | The Government Of The United States, As Represented By The Secretary Of Health And Human Services, National Institutes Of Health, Office Of Technology Transfer | Hydrazide, amide, phthalimide and phthalhydrazide analogs as inhibitors of retroviral integrase |
KR101039235B1 (ko) * | 2007-08-29 | 2011-06-07 | 메디포스트(주) | 제대혈 유래 간엽줄기세포를 포함하는 인터루킨-8 또는지알오-알파 발현 세포가 관련된 질병의 진단, 예방 또는치료용 조성물 |
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SG176464A1 (en) | 2008-05-09 | 2011-12-29 | Agency Science Tech & Res | Diagnosis and treatment of kawasaki disease |
KR101588547B1 (ko) | 2008-11-11 | 2016-01-28 | 더 리젠츠 오브 더 유니버시티 오브 미시간 | 항-cxcr1 조성물 및 방법 |
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CN108025189B (zh) * | 2015-09-04 | 2021-07-02 | 美国陶氏益农公司 | 具有杀虫效用的分子,以及与其相关的中间体、组合物和方法 |
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WO2018071687A1 (en) * | 2016-10-13 | 2018-04-19 | The Regents Of The University Of California | Methods of treating pruritis |
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-
2005
- 2005-05-11 CA CA002565519A patent/CA2565519A1/en not_active Abandoned
- 2005-05-11 AU AU2005245399A patent/AU2005245399A1/en not_active Abandoned
- 2005-05-11 MX MXPA06013118A patent/MXPA06013118A/es active IP Right Grant
- 2005-05-11 CN CN2005800232328A patent/CN1984899B/zh not_active Expired - Fee Related
- 2005-05-11 EP EP05779979.3A patent/EP1745032B1/en active Active
- 2005-05-11 JP JP2007513317A patent/JP2007537272A/ja not_active Ceased
- 2005-05-11 KR KR1020067023571A patent/KR20070011475A/ko not_active Application Discontinuation
- 2005-05-11 WO PCT/US2005/016507 patent/WO2005113534A2/en active Application Filing
- 2005-05-11 US US11/126,977 patent/US7326729B2/en not_active Expired - Fee Related
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2006
- 2006-11-06 ZA ZA200609237A patent/ZA200609237B/xx unknown
- 2006-11-09 IL IL179162A patent/IL179162A0/en unknown
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2007
- 2007-07-10 US US11/775,567 patent/US20070248594A1/en not_active Abandoned
-
2011
- 2011-10-11 JP JP2011224353A patent/JP2012006982A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
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JP2007537272A (ja) | 2007-12-20 |
US20060014794A1 (en) | 2006-01-19 |
IL179162A0 (en) | 2007-03-08 |
EP1745032A2 (en) | 2007-01-24 |
EP1745032B1 (en) | 2013-07-31 |
WO2005113534A2 (en) | 2005-12-01 |
JP2012006982A (ja) | 2012-01-12 |
CN1984899A (zh) | 2007-06-20 |
WO2005113534A3 (en) | 2006-10-26 |
MXPA06013118A (es) | 2007-02-28 |
US20070248594A1 (en) | 2007-10-25 |
CN1984899B (zh) | 2011-07-27 |
US7326729B2 (en) | 2008-02-05 |
KR20070011475A (ko) | 2007-01-24 |
CA2565519A1 (en) | 2005-12-01 |
AU2005245399A1 (en) | 2005-12-01 |
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