BR0206968A - Ciclobuteno-1,2-dionas 3,4-dissubstituìdas como antagonistas receptores de quimiocina cxc - Google Patents

Ciclobuteno-1,2-dionas 3,4-dissubstituìdas como antagonistas receptores de quimiocina cxc

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Publication number
BR0206968A
BR0206968A BR0206968-7A BR0206968A BR0206968A BR 0206968 A BR0206968 A BR 0206968A BR 0206968 A BR0206968 A BR 0206968A BR 0206968 A BR0206968 A BR 0206968A
Authority
BR
Brazil
Prior art keywords
diones
receptor antagonists
chemokine receptor
cxc chemokine
cyclobutene
Prior art date
Application number
BR0206968-7A
Other languages
English (en)
Inventor
Arthur G Taveras
Cynthia J Aki
Richard W Bond
Jianping Chao
Michael Dwyer
Johan A Ferreira
Jonathan Pachter
John J Baldwin
Bernd Kaiser
Ge Li
J Robert Merritt
Laura L Rokosz
Kingsley H Nelson Jr
Original Assignee
Schering Corp
Pharmacopeia Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp, Pharmacopeia Inc filed Critical Schering Corp
Publication of BR0206968A publication Critical patent/BR0206968A/pt

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Abstract

"CICLOBUTENO-1,2-DIONAS 3,4-DISSUBSTITUìDAS COMO ANTAGONISTAS RECEPTORES DE QUIMIOCINA CXC". A invenção refere-se a compostos da fórmula (1) onde as variáveis A e B são um grupo de heteroarila ou arila como definido nas reivindicações, ou uma pró-droga desta, ou um solvato, isómero ou sal farmaceuticamente aceitável do referido composto ou da referida pró-droga, que são úteis para o tratamento de doenças mediadas por quimiocina tal como distúrbios inflamatórios crónicos e agudos e câncer.
BR0206968-7A 2001-02-02 2002-02-01 Ciclobuteno-1,2-dionas 3,4-dissubstituìdas como antagonistas receptores de quimiocina cxc BR0206968A (pt)

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PCT/US2002/002888 WO2002076926A1 (en) 2001-02-02 2002-02-01 3,4-di-substituted cyclobutene-1, 2-diones as cxc chemokine receptor antagonists

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TW550672B (en) * 2001-02-21 2003-09-01 Semiconductor Energy Lab Method and apparatus for film deposition
SG118118A1 (en) * 2001-02-22 2006-01-27 Semiconductor Energy Lab Organic light emitting device and display using the same

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RU2003126913A (ru) 2005-03-10
AU2002303084B2 (en) 2006-05-25
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US20030097004A1 (en) 2003-05-22
CN1575273A (zh) 2005-02-02
EP1355875A1 (en) 2003-10-29
NO20033424L (no) 2003-09-30
WO2002076926A1 (en) 2002-10-03
SK9782003A3 (en) 2004-01-08
PL367534A1 (en) 2005-02-21
NO20033424D0 (no) 2003-07-31
CZ20032098A3 (cs) 2004-01-14
ZA200305881B (en) 2005-01-26
MXPA03006950A (es) 2003-11-18
IL156793A0 (en) 2004-02-08
CA2436351A1 (en) 2002-10-03
ECSP034712A (es) 2003-09-24
JP2004529911A (ja) 2004-09-30
KR20030090629A (ko) 2003-11-28

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