ZA200408548B - Benzothiadiazepine derivatives, processes for their preparation and pharmaceutical compositions containing them. - Google Patents
Benzothiadiazepine derivatives, processes for their preparation and pharmaceutical compositions containing them. Download PDFInfo
- Publication number
- ZA200408548B ZA200408548B ZA200408548A ZA200408548A ZA200408548B ZA 200408548 B ZA200408548 B ZA 200408548B ZA 200408548 A ZA200408548 A ZA 200408548A ZA 200408548 A ZA200408548 A ZA 200408548A ZA 200408548 B ZA200408548 B ZA 200408548B
- Authority
- ZA
- South Africa
- Prior art keywords
- solvate
- formula
- salt
- carbamoyl
- pharmaceutically acceptable
- Prior art date
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- 238000002360 preparation method Methods 0.000 title claims description 3
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- 229910052757 nitrogen Inorganic materials 0.000 claims description 62
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Classifications
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/36—Seven-membered rings
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- A61P1/12—Antidiarrhoeals
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A—HUMAN NECESSITIES
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Landscapes
- Health & Medical Sciences (AREA)
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- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0209467.0A GB0209467D0 (en) | 2002-04-25 | 2002-04-25 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200408548B true ZA200408548B (en) | 2005-11-14 |
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| ZA200408548A ZA200408548B (en) | 2002-04-25 | 2004-10-21 | Benzothiadiazepine derivatives, processes for their preparation and pharmaceutical compositions containing them. |
Country Status (23)
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| EP (1) | EP1501813B1 (zh) |
| JP (1) | JP4475960B2 (zh) |
| KR (1) | KR20050007329A (zh) |
| CN (1) | CN100408567C (zh) |
| AR (1) | AR040408A1 (zh) |
| AU (1) | AU2003226565A1 (zh) |
| BR (1) | BR0309493A (zh) |
| CA (1) | CA2483155A1 (zh) |
| ES (1) | ES2434098T3 (zh) |
| GB (1) | GB0209467D0 (zh) |
| IL (1) | IL164798A0 (zh) |
| IS (1) | IS7543A (zh) |
| MX (1) | MXPA04010597A (zh) |
| NO (1) | NO20044597L (zh) |
| NZ (1) | NZ536105A (zh) |
| PL (1) | PL372998A1 (zh) |
| RU (1) | RU2333205C2 (zh) |
| TW (1) | TW200306844A (zh) |
| UA (1) | UA77797C2 (zh) |
| UY (1) | UY27779A1 (zh) |
| WO (1) | WO2003091232A2 (zh) |
| ZA (1) | ZA200408548B (zh) |
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| EG26979A (en) | 2000-12-21 | 2015-03-01 | Astrazeneca Ab | Chemical compounds |
| GB0121337D0 (en) | 2001-09-04 | 2001-10-24 | Astrazeneca Ab | Chemical compounds |
| GB0121622D0 (en) | 2001-09-07 | 2001-10-31 | Astrazeneca Ab | Chemical compounds |
| GB0121621D0 (en) | 2001-09-07 | 2001-10-31 | Astrazeneca Ab | Chemical compounds |
| RU2305681C2 (ru) | 2001-09-08 | 2007-09-10 | Астразенека Аб | Производные бензотиадиазепина, способ их получения (варианты) |
| SE0104333D0 (sv) | 2001-12-19 | 2001-12-19 | Astrazeneca Ab | Therapeutic agents |
| GB0213669D0 (en) | 2002-06-14 | 2002-07-24 | Astrazeneca Ab | Chemical compounds |
| DK1517883T3 (da) * | 2002-06-20 | 2008-05-26 | Astrazeneca Ab | Ortho-substituerede benzoesyrederivater til behandling af insulinresistens |
| GB0304194D0 (en) | 2003-02-25 | 2003-03-26 | Astrazeneca Ab | Chemical compounds |
| GB0307918D0 (en) | 2003-04-05 | 2003-05-14 | Astrazeneca Ab | Therapeutic use |
| AR057828A1 (es) * | 2005-09-29 | 2007-12-19 | Astrazeneca Ab | Compuestos derivados de azetidina, su preparacion y composicion farmaceuutica |
| CN101790512A (zh) * | 2007-03-08 | 2010-07-28 | 阿尔比里奥公司 | 2-取代-3-苯基丙酸衍生物及其在炎性肠病治疗中的用途 |
| US8858916B2 (en) | 2008-09-30 | 2014-10-14 | Mallinckrodt Llc | Metal chelate linked to a hexose carrier for use as a metallopharmaceutical diagnostic or therapeutic agent |
| EP2367554A4 (en) * | 2008-11-26 | 2020-03-25 | Satiogen Pharmaceuticals, Inc. | BILIARY ACID RECYCLING INHIBITORS FOR THE TREATMENT OF OBESITY AND DIABETES |
| BRPI1008749B8 (pt) | 2009-02-05 | 2021-05-25 | Immunogen Inc | compostos derivados de benzodiazepina, seus conjugados, composição farmacêutica, seu uso e seus processos de preparação |
| FR2943342B1 (fr) * | 2009-03-20 | 2011-03-04 | Servier Lab | Nouveaux derives de benzothiadiazepines,leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| KR101313106B1 (ko) | 2009-12-17 | 2013-09-30 | 한국전자통신연구원 | 손가락 착용형 매개 장치 및 상기 장치를 이용한 손가락 동작 인식 방법 |
| WO2011150286A2 (en) | 2010-05-26 | 2011-12-01 | Satiogen Pharmaceuticals,Inc. | Bile acid recycling inhibitors and satiogens for treatment of diabetes, obesity, and inflammatory gastrointestinal conditions |
| BR112013010157B1 (pt) | 2010-11-08 | 2020-02-04 | Albireo Ab | iinibidores do ibat, seus usos, e composição e combinações farmacêuticas |
| AU2011326872C1 (en) | 2010-11-08 | 2015-02-19 | Albireo Ab | A pharmaceutical combination comprising an IBAT inhibitor and a bile acid binder |
| EP3666289A1 (en) | 2011-02-15 | 2020-06-17 | ImmunoGen, Inc. | Cytotoxic benzodiazepine derivatives |
| KR102051030B1 (ko) | 2011-10-28 | 2019-12-02 | 루메나 파마수티컬즈, 인코포레이티드 | 소아 담즙울체성 간 질환 치료용 담즙산 재순환 억제제 |
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