ZA200209520B - Sustained release pharmaceutical compositions for parenteral administration of hydrophilic compounds. - Google Patents
Sustained release pharmaceutical compositions for parenteral administration of hydrophilic compounds. Download PDFInfo
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- ZA200209520B ZA200209520B ZA200209520A ZA200209520A ZA200209520B ZA 200209520 B ZA200209520 B ZA 200209520B ZA 200209520 A ZA200209520 A ZA 200209520A ZA 200209520 A ZA200209520 A ZA 200209520A ZA 200209520 B ZA200209520 B ZA 200209520B
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- South Africa
- Prior art keywords
- microemulsion
- surfactant
- biologically active
- preparation
- days
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- 238000013268 sustained release Methods 0.000 title claims description 19
- 239000012730 sustained-release form Substances 0.000 title claims description 19
- 238000007911 parenteral administration Methods 0.000 title claims description 9
- 150000002433 hydrophilic molecules Chemical class 0.000 title claims description 3
- 239000008194 pharmaceutical composition Substances 0.000 title description 5
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Classifications
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
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- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Dispersion Chemistry (AREA)
- Epidemiology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT2000MI001173A IT1318539B1 (it) | 2000-05-26 | 2000-05-26 | Composizioni farmaceutiche a rilascio prolungato per lasomministrazione parenterale di sostanze idrofile biologicamente |
Publications (1)
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| ZA200209520B true ZA200209520B (en) | 2003-11-24 |
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| ZA200209520A ZA200209520B (en) | 2000-05-26 | 2002-11-22 | Sustained release pharmaceutical compositions for parenteral administration of hydrophilic compounds. |
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| EP (1) | EP1283700B1 (da) |
| JP (1) | JP4954423B2 (da) |
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| IL (1) | IL153011A0 (da) |
| IT (1) | IT1318539B1 (da) |
| MX (1) | MXPA02011539A (da) |
| NO (1) | NO334880B1 (da) |
| PL (1) | PL203354B1 (da) |
| PT (1) | PT1283700E (da) |
| RU (1) | RU2272615C2 (da) |
| SI (1) | SI1283700T1 (da) |
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| WO (1) | WO2001089479A2 (da) |
| YU (1) | YU88202A (da) |
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| US8119159B2 (en) | 1999-02-22 | 2012-02-21 | Merrion Research Iii Limited | Solid oral dosage form containing an enhancer |
| US7658938B2 (en) | 1999-02-22 | 2010-02-09 | Merrion Reasearch III Limited | Solid oral dosage form containing an enhancer |
| SI1787658T1 (sl) | 2005-11-10 | 2012-07-31 | Chemi Spa | Formulacije z trajnim sproščanjem somatostatin analognih inhibitorjev rastnega hormona |
| AU2007235251B2 (en) | 2006-04-07 | 2013-02-07 | Merrion Research Iii Limited | Solid oral dosage form containing an enhancer |
| KR100816065B1 (ko) * | 2006-11-27 | 2008-03-24 | 동국제약 주식회사 | 초기 방출억제 특성이 우수한 서방출성 마이크로캡슐의제조방법 및 이에 의해 제조되는 마이크로캡슐 |
| RU2362544C2 (ru) * | 2007-04-09 | 2009-07-27 | Закрытое акционерное общество "Санкт-Петербургский институт фармации" | Наноэмульсия с биологически активными веществами |
| WO2009046386A1 (en) * | 2007-10-04 | 2009-04-09 | Py Daniel C | Apparatus and method for formulating and aseptically filling liquid products |
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| WO1994008610A1 (en) | 1992-10-16 | 1994-04-28 | Smithkline Beecham Corporation | Pharmaceutical emulsion compositions |
| SE512663C2 (sv) * | 1997-10-23 | 2000-04-17 | Biogram Ab | Inkapslingsförfarande för aktiv substans i en bionedbrytbar polymer |
| EP1023045A2 (en) * | 1997-10-24 | 2000-08-02 | Neorx Corporation | Delivery vehicles for bioactive agents and uses thereof |
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2000
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- 2001-05-23 SI SI200130529T patent/SI1283700T1/sl unknown
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- 2001-05-23 CN CNB018099254A patent/CN100479856C/zh not_active Expired - Lifetime
- 2001-05-23 PT PT01960242T patent/PT1283700E/pt unknown
- 2001-05-23 AU AU8178601A patent/AU8178601A/xx active Pending
- 2001-05-23 KR KR1020027015828A patent/KR100802625B1/ko active IP Right Grant
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