YU45403A - Novi 1,2-difenil-azetidinoni, postupak za njihovu proizvodnju, lekovi koji sadrže ova jedinjenja i njihova primena za lečenje poremećaja u metabolizmu lipida - Google Patents
Novi 1,2-difenil-azetidinoni, postupak za njihovu proizvodnju, lekovi koji sadrže ova jedinjenja i njihova primena za lečenje poremećaja u metabolizmu lipidaInfo
- Publication number
- YU45403A YU45403A YU45403A YUP45403A YU45403A YU 45403 A YU45403 A YU 45403A YU 45403 A YU45403 A YU 45403A YU P45403 A YUP45403 A YU P45403A YU 45403 A YU45403 A YU 45403A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- compounds
- novel
- producing
- lipid metabolism
- treating disorders
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
- A61P39/06—Free radical scavengers or antioxidants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
Abstract
Pronalazak se odnosi na jedinjenja formule I, u kojima R1, R2, R3, R4, R5 i R6 imaju navedena značenja, kao i na njihove farmaceutski prihvatljive soli. Jedinjenja definisana ovim pronalaskom su pogodna da se primene, na primer, kao hipolipidemijska sredstva.[The invention relates to the compounds of the formula (I), wherein R1, R2, R3, R4, R5, and R6 have the cited meanings, and to their physiologically acceptable salts. The inventive compounds are suitable, for example, as hypolipidemics.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10064398A DE10064398A1 (de) | 2000-12-21 | 2000-12-21 | Neue Diphenylazetidinone, Verfahren zu deren Herstellung, diese Verbindungen enthaltende Arzneimittel und deren Verwendung |
DE2001152981 DE10152981A1 (de) | 2001-10-26 | 2001-10-26 | Neue Diphenylazetidinone, Verfahren zu deren Herstellung, diese Verbindungen enthaltende Arzneimittel und deren Verwendung |
Publications (2)
Publication Number | Publication Date |
---|---|
YU45403A true YU45403A (sh) | 2006-05-25 |
RS50864B RS50864B (sr) | 2010-08-31 |
Family
ID=26008042
Country Status (29)
Country | Link |
---|---|
US (5) | US6992067B2 (sh) |
EP (1) | EP1345895B1 (sh) |
JP (1) | JP4605990B2 (sh) |
KR (1) | KR100833089B1 (sh) |
CN (1) | CN1217927C (sh) |
AR (1) | AR034010A1 (sh) |
AT (1) | ATE349425T1 (sh) |
AU (2) | AU1609702A (sh) |
BR (1) | BR0116325A (sh) |
CA (1) | CA2431983C (sh) |
CY (1) | CY1106383T1 (sh) |
CZ (1) | CZ20031732A3 (sh) |
DE (1) | DE50111751D1 (sh) |
DK (1) | DK1345895T3 (sh) |
EE (1) | EE200300236A (sh) |
ES (1) | ES2277890T3 (sh) |
HK (1) | HK1060120A1 (sh) |
HR (1) | HRP20030498A2 (sh) |
HU (1) | HUP0401081A3 (sh) |
IL (2) | IL156550A0 (sh) |
MX (1) | MXPA03005155A (sh) |
NO (1) | NO325496B1 (sh) |
NZ (1) | NZ526593A (sh) |
PL (1) | PL362379A1 (sh) |
PT (1) | PT1345895E (sh) |
RS (1) | RS50864B (sh) |
SK (1) | SK7822003A3 (sh) |
TW (1) | TWI293626B (sh) |
WO (1) | WO2002050027A1 (sh) |
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- 2001-12-11 AU AU1609702A patent/AU1609702A/xx active Pending
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- 2001-12-11 WO PCT/EP2001/014531 patent/WO2002050027A1/de active IP Right Grant
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