WO2007095638A3 - Petites molecules contenant du bore en tant qu'agents anti-inflammatoires - Google Patents

Petites molecules contenant du bore en tant qu'agents anti-inflammatoires Download PDF

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Publication number
WO2007095638A3
WO2007095638A3 PCT/US2007/062350 US2007062350W WO2007095638A3 WO 2007095638 A3 WO2007095638 A3 WO 2007095638A3 US 2007062350 W US2007062350 W US 2007062350W WO 2007095638 A3 WO2007095638 A3 WO 2007095638A3
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WO
WIPO (PCT)
Prior art keywords
boron
small molecules
containing small
inflammatory agents
disclosed
Prior art date
Application number
PCT/US2007/062350
Other languages
English (en)
Other versions
WO2007095638A2 (fr
Inventor
Stephen J Baker
Virginia Sanders
Tsutomu Akama
Carolyn Bellinger-Kawahara
Yvonne Freund
Kirk R Maples
Jacob J Plattner
Yong-Kang Zhang
Huchen Zhou
Vincent S Hernandez
Original Assignee
Anacor Pharmaceuticals Inc
Stephen J Baker
Virginia Sanders
Tsutomu Akama
Carolyn Bellinger-Kawahara
Yvonne Freund
Kirk R Maples
Jacob J Plattner
Yong-Kang Zhang
Huchen Zhou
Vincent S Hernandez
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38372267&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=WO2007095638(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority to BRPI0708051-4A priority Critical patent/BRPI0708051A2/pt
Priority to ES07757149.5T priority patent/ES2542342T3/es
Priority to KR1020147013817A priority patent/KR20140082842A/ko
Priority to NZ570257A priority patent/NZ570257A/en
Priority to MX2008010381A priority patent/MX2008010381A/es
Priority to RS20150474A priority patent/RS54108B1/en
Priority to EP07757149.5A priority patent/EP1988779B1/fr
Priority to KR1020177001541A priority patent/KR101819869B1/ko
Priority to EP13179945.4A priority patent/EP2719388B1/fr
Priority to KR1020137025594A priority patent/KR20130120552A/ko
Priority to KR1020147035518A priority patent/KR101622870B1/ko
Priority to AU2007214421A priority patent/AU2007214421B2/en
Priority to PL07757149T priority patent/PL1988779T3/pl
Priority to MX2013015092A priority patent/MX360301B/es
Priority to KR1020157027015A priority patent/KR20150113219A/ko
Application filed by Anacor Pharmaceuticals Inc, Stephen J Baker, Virginia Sanders, Tsutomu Akama, Carolyn Bellinger-Kawahara, Yvonne Freund, Kirk R Maples, Jacob J Plattner, Yong-Kang Zhang, Huchen Zhou, Vincent S Hernandez filed Critical Anacor Pharmaceuticals Inc
Priority to RU2008137086/15A priority patent/RU2508113C2/ru
Priority to KR1020157000589A priority patent/KR20150013941A/ko
Priority to MEP-2015-97A priority patent/ME02188B/me
Priority to CN2007800133393A priority patent/CN101420854B/zh
Priority to JP2008555528A priority patent/JP5419466B2/ja
Priority to SI200731663T priority patent/SI1988779T1/sl
Priority to DK07757149.5T priority patent/DK1988779T5/en
Priority to PL13179945T priority patent/PL2719388T3/pl
Priority to CA2642583A priority patent/CA2642583C/fr
Publication of WO2007095638A2 publication Critical patent/WO2007095638A2/fr
Publication of WO2007095638A3 publication Critical patent/WO2007095638A3/fr
Priority to IL193230A priority patent/IL193230A/en
Priority to ZA2008/06754A priority patent/ZA200806754B/en
Priority to HK09101607.4A priority patent/HK1121344A1/xx
Priority to HRP20150710TT priority patent/HRP20150710T1/hr
Priority to IL241792A priority patent/IL241792B/en
Priority to CY20191100519T priority patent/CY1121899T1/el

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    • A61P7/08Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/02Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
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    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02Boron compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02Boron compounds
    • C07F5/027Organoboranes and organoborohydrides
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23LFOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BY SUBCLASSES A21D OR A23B-A23J; THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OF NUTRITIVE QUALITIES, PHYSICAL TREATMENT; PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
    • A23L33/00Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
    • A23L33/10Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof using additives
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23VINDEXING SCHEME RELATING TO FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES AND LACTIC OR PROPIONIC ACID BACTERIA USED IN FOODSTUFFS OR FOOD PREPARATION
    • A23V2002/00Food compositions, function of food ingredients or processes for food or foodstuffs
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23VINDEXING SCHEME RELATING TO FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES AND LACTIC OR PROPIONIC ACID BACTERIA USED IN FOODSTUFFS OR FOOD PREPARATION
    • A23V2200/00Function of food ingredients
    • A23V2200/30Foods, ingredients or supplements having a functional effect on health
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00Preparations for use in therapy
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

La présente invention concerne des procédés destinés à traiter des états anti-inflammatoires à l'aide de petites molécules contenant du bore.
PCT/US2007/062350 2006-02-16 2007-02-16 Petites molecules contenant du bore en tant qu'agents anti-inflammatoires WO2007095638A2 (fr)

Priority Applications (30)

Application Number Priority Date Filing Date Title
CA2642583A CA2642583C (fr) 2006-02-16 2007-02-16 Petites molecules contenant du bore en tant qu'agents anti-inflammatoires
KR1020157000589A KR20150013941A (ko) 2006-02-16 2007-02-16 항염증제로서 보론함유 소분자
KR1020147013817A KR20140082842A (ko) 2006-02-16 2007-02-16 항염증제로서 보론함유 소분자
RU2008137086/15A RU2508113C2 (ru) 2006-02-16 2007-02-16 Борсодержащие малые молекулы в качестве противовоспалительных средств
MX2008010381A MX2008010381A (es) 2006-02-16 2007-02-16 Moleculas pequeñas que contienen boro como agentes antiinflamatorios.
RS20150474A RS54108B1 (en) 2006-02-16 2007-02-16 SMALL MOLECULES CONTAINING BORON AS AGENTS FOR INFLAMMATION
EP07757149.5A EP1988779B1 (fr) 2006-02-16 2007-02-16 Petites molecules contenant du bore en tant qu'agents anti-inflammatoires
ES07757149.5T ES2542342T3 (es) 2006-02-16 2007-02-16 Pequeñas moléculas que contienen boro como agentes antiinflamatorios
EP13179945.4A EP2719388B1 (fr) 2006-02-16 2007-02-16 Petites molécules contenant du bore en tant qu'agents anti-inflammatoires
KR1020137025594A KR20130120552A (ko) 2006-02-16 2007-02-16 항염증제로서 보론함유 소분자
KR1020147035518A KR101622870B1 (ko) 2006-02-16 2007-02-16 항염증제로서 보론함유 소분자
AU2007214421A AU2007214421B2 (en) 2006-02-16 2007-02-16 Boron-containing small molecules as anti-inflammatory agents
PL07757149T PL1988779T3 (pl) 2006-02-16 2007-02-16 Małe cząsteczki zawierające bor jako środki przeciwzapalne
MEP-2015-97A ME02188B (me) 2006-02-16 2007-02-16 Mali molekuli koji sadrže boron kao antiinflamatorni agensi
KR1020157027015A KR20150113219A (ko) 2006-02-16 2007-02-16 항염증제로서 보론함유 소분자
BRPI0708051-4A BRPI0708051A2 (pt) 2006-02-16 2007-02-16 moléculas pequenas contendo boro como agentes antiflamatórios
NZ570257A NZ570257A (en) 2006-02-16 2007-02-16 Boron-containing small molecules as anti-inflammatory agents
KR1020177001541A KR101819869B1 (ko) 2006-02-16 2007-02-16 항염증제로서 보론함유 소분자
MX2013015092A MX360301B (es) 2006-02-16 2007-02-16 Moleculas pequeñas que contienen boro como agentes antiinflamatorios.
CN2007800133393A CN101420854B (zh) 2006-02-16 2007-02-16 作为抗炎药的含硼的小分子
JP2008555528A JP5419466B2 (ja) 2006-02-16 2007-02-16 抗炎症剤としてのホウ素含有小分子
SI200731663T SI1988779T1 (sl) 2006-02-16 2007-02-16 Bor-vsebujoče majhne molekule kot protivnetna sredstva
DK07757149.5T DK1988779T5 (en) 2006-02-16 2007-02-16 SMALL boron MOLECULES AS ANTI-INFLAMMATORY AGENTS
PL13179945T PL2719388T3 (pl) 2006-02-16 2007-02-16 Małe cząsteczki zawierające bor jako środki przeciwzapalne
ZA2008/06754A ZA200806754B (en) 2006-02-16 2008-08-04 Boron-containing small molecules as anti-inflammatory agents
IL193230A IL193230A (en) 2006-02-16 2008-08-04 Use of benzoxoborol derivatives in the preparation of drugs for the treatment of inflammatory diseases
HK09101607.4A HK1121344A1 (en) 2006-02-16 2009-02-19 Boron-containing small molecules as anti-inflammatory agents
HRP20150710TT HRP20150710T1 (hr) 2006-02-16 2015-07-01 Male molekule koje sadrže bor kao protu-upalni agensi
IL241792A IL241792B (en) 2006-02-16 2015-09-21 Boron-containing molecules with anti-inflammatory ingredients
CY20191100519T CY1121899T1 (el) 2006-02-16 2019-05-14 Βοριουχα μικρομορια ως αντιφλεγμονωδεις παραγοντες

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US77453206P 2006-02-16 2006-02-16
US60/774,532 2006-02-16
US82388806P 2006-08-29 2006-08-29
US60/823,888 2006-08-29

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WO2007095638A2 WO2007095638A2 (fr) 2007-08-23
WO2007095638A3 true WO2007095638A3 (fr) 2008-07-31

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US (11) US8168614B2 (fr)
EP (2) EP2719388B1 (fr)
JP (4) JP5419466B2 (fr)
KR (7) KR101622870B1 (fr)
CN (2) CN101420854B (fr)
AU (1) AU2007214421B2 (fr)
BR (1) BRPI0708051A2 (fr)
CA (2) CA2642583C (fr)
CY (1) CY1121899T1 (fr)
DK (2) DK1988779T5 (fr)
ES (2) ES2542342T3 (fr)
HK (1) HK1121344A1 (fr)
HR (1) HRP20150710T1 (fr)
HU (2) HUE044941T2 (fr)
IL (2) IL193230A (fr)
ME (1) ME02188B (fr)
MX (2) MX360301B (fr)
NZ (1) NZ570257A (fr)
PL (2) PL1988779T3 (fr)
PT (2) PT2719388T (fr)
RS (1) RS54108B1 (fr)
RU (2) RU2642628C2 (fr)
SI (2) SI2719388T1 (fr)
WO (1) WO2007095638A2 (fr)
ZA (1) ZA200806754B (fr)

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