CA2654449A1 - Composes destines au traitement d'une maladie periodontale - Google Patents

Composes destines au traitement d'une maladie periodontale Download PDF

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Publication number
CA2654449A1
CA2654449A1 CA002654449A CA2654449A CA2654449A1 CA 2654449 A1 CA2654449 A1 CA 2654449A1 CA 002654449 A CA002654449 A CA 002654449A CA 2654449 A CA2654449 A CA 2654449A CA 2654449 A1 CA2654449 A1 CA 2654449A1
Authority
CA
Canada
Prior art keywords
substituted
alkyl
unsubstituted
compound
species
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002654449A
Other languages
English (en)
Inventor
Virginia Sanders
Kirk R. Maples
Jacob J. Plattner
Carolyn Bellinger-Kawahara
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Anacor Pharmaceuticals Inc
Original Assignee
Anacor Pharmaceuticals, Inc.
Virginia Sanders
Kirk R. Maples
Jacob J. Plattner
Carolyn Bellinger-Kawahara
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anacor Pharmaceuticals, Inc., Virginia Sanders, Kirk R. Maples, Jacob J. Plattner, Carolyn Bellinger-Kawahara filed Critical Anacor Pharmaceuticals, Inc.
Publication of CA2654449A1 publication Critical patent/CA2654449A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/58Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing atoms other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur or phosphorus
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q11/00Preparations for care of the teeth, of the oral cavity or of dentures; Dentifrices, e.g. toothpastes; Mouth rinses
CA002654449A 2006-06-12 2007-06-12 Composes destines au traitement d'une maladie periodontale Abandoned CA2654449A1 (fr)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US80450406P 2006-06-12 2006-06-12
US60/804,504 2006-06-12
US82389306P 2006-08-29 2006-08-29
US60/823,893 2006-08-29
PCT/US2007/071049 WO2007146965A2 (fr) 2006-06-12 2007-06-12 Composés destinés au traitement d'une maladie périodontale

Publications (1)

Publication Number Publication Date
CA2654449A1 true CA2654449A1 (fr) 2007-12-21

Family

ID=38832802

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002654449A Abandoned CA2654449A1 (fr) 2006-06-12 2007-06-12 Composes destines au traitement d'une maladie periodontale

Country Status (9)

Country Link
EP (1) EP2044091A4 (fr)
KR (1) KR20090029797A (fr)
AU (1) AU2007257689A1 (fr)
BR (1) BRPI0713010A2 (fr)
CA (1) CA2654449A1 (fr)
IL (1) IL195571A0 (fr)
MX (1) MX2008015918A (fr)
RU (1) RU2008152367A (fr)
WO (1) WO2007146965A2 (fr)

Families Citing this family (41)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUE040060T2 (hu) 2005-02-16 2019-02-28 Anacor Pharmaceuticals Inc Halogén-szubsztituált boronftalidok fertõzések kezelésére
CN106008583A (zh) 2005-12-30 2016-10-12 安纳考尔医药公司 含硼的小分子
US8168614B2 (en) 2006-02-16 2012-05-01 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-inflammatory agents
JO3598B1 (ar) 2006-10-10 2020-07-05 Infinity Discovery Inc الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني
JO3396B1 (ar) 2007-06-20 2019-10-20 Anacor Pharmaceuticals Inc جزيئات صغيرة تحتوي على البورون
RU2547441C2 (ru) 2008-03-06 2015-04-10 Анакор Фармасьютикалз, Инк. Борсодержащие малые молекулы в качестве противовоспалительных агентов
PE20091838A1 (es) 2008-04-09 2009-12-18 Infinity Pharmaceuticals Inc Inhibidores de amida hidrolasa de acido graso
WO2010018837A2 (fr) * 2008-08-11 2010-02-18 独立行政法人科学技術振興機構 Inhibiteur de la réticulation de protéines
WO2010028005A1 (fr) 2008-09-04 2010-03-11 Anacor Pharmaceuticals, Inc. Petites molécules contenant du bore
EP2348863A4 (fr) 2008-09-04 2012-03-07 Anacor Pharmaceuticals Inc Petites molécules contenant du bore
US9493489B2 (en) 2008-10-15 2016-11-15 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agents
US8461364B2 (en) 2008-12-17 2013-06-11 Glaxosmithkline Llc Polymorphs of (S)-3-aminomethyl-7-(3-hydroxy-propoxy)-3H-benzo[C][1,2]oxaborol-1-OL
CA2757622A1 (fr) 2009-04-07 2010-10-14 Infinity Pharmaceuticals, Inc. Inhibiteurs d'hydrolase d'amide d'acide gras
EP2416660B1 (fr) 2009-04-07 2014-07-02 Infinity Pharmaceuticals, Inc. Inhibiteurs d'amide d'hydrolase d'acide gras
TW201109022A (en) * 2009-06-03 2011-03-16 Colgate Palmolive Co Borinic compositions
WO2011017125A1 (fr) 2009-07-28 2011-02-10 Anacor Pharmaceuticals, Inc. Molécules contenant du bore trisubstitué
WO2011019618A1 (fr) 2009-08-14 2011-02-17 Anacor Pharmaceuticals, Inc. Petites molécules contenant du bore et utilisables en tant qu'agents antiprotozoaires
WO2011049971A1 (fr) 2009-10-20 2011-04-28 Anacor Pharmaceuticals, Inc. Petites molécules contenant du bore comme agents antiprotozoaires
US20110212918A1 (en) 2009-11-11 2011-09-01 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2011063293A1 (fr) * 2009-11-20 2011-05-26 Anacor Pharmaceuticals, Inc. Petites molécules contenant du bore en tant qu'agents antihelminthes
RU2414210C1 (ru) * 2009-12-28 2011-03-20 Общество С Ограниченной Ответственностью "Сплат-Косметика" (Ооо "Сплат-Косметика") Средство для удаления табачных смол и композиции на его основе
US8716478B2 (en) 2010-01-27 2014-05-06 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
RU2569061C2 (ru) 2010-02-03 2015-11-20 Инфинити Фармасьютикалз, Инк. Ингибиторы амид-гидролазы жирных кислот
AP2012006482A0 (en) 2010-03-19 2012-10-31 Anacor Pharmacueticals Inc Boron-containing small molecules as anti-protozoalagent
ES2635333T3 (es) 2010-09-07 2017-10-03 Anacor Pharmaceuticals, Inc. Derivados de benzoxaborol para tratar infecciones bacterianas
AR088668A1 (es) * 2011-11-21 2014-06-25 Lilly Co Eli Moleculas pequeñas que contienen boro
US9585396B2 (en) 2013-01-30 2017-03-07 Agrofresh Inc. Volatile applications against pathogens
CA2899317A1 (fr) 2013-01-30 2014-08-07 Dow Agrosciences Llc Utilisation des benzoxaboroles a titre d'agents antimicrobiens volatils sur les viandes, les plantes, ou des parties de plantes
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
US8669207B1 (en) 2013-01-30 2014-03-11 Dow Agrosciences, Llc. Compounds and compositions
WO2016001834A1 (fr) 2014-07-01 2016-01-07 Daiichi Sankyo Company, Limited Benzoxaboroles tricycliques en tant qu'agents antibactériens
CA3015662A1 (fr) 2016-03-07 2017-09-14 Agrofresh Inc. Procedes synergiques d'utilisation de composes de benzoxaborole et de gaz de conservation en tant qu'agent antimicrobien pour les plantes cultivees
US11447506B2 (en) 2016-05-09 2022-09-20 Anacor Pharmaceuticals, Inc. Crystal forms of crisaborole in free form and preparation method and use thereof
AU2017262235C1 (en) * 2016-05-09 2020-08-20 Anacor Pharmaceuticals, Llc Crystal forms of crisaborole in free form and preparation method and use thereof
CN107759625B (zh) * 2016-08-22 2020-12-29 药源药物化学(上海)有限公司 4-(1-羟基-1,3-二氢苯并[c][1,2]氧杂硼杂环戊二烯-5-基氧基)苯氰的制备方法
US10961261B2 (en) 2017-03-01 2021-03-30 Anacor Pharmaceuticals, Inc. Oxaborole analogs and uses thereof
EP3576747A4 (fr) * 2017-03-09 2020-12-16 The Penn State Research Foundation Petites molécules contenant du bore pour inhiber l'activité d'une protéine tyrosine phosphatase de type récepteur
CN110183477B (zh) * 2019-07-03 2022-03-04 石家庄诚志永华显示材料有限公司 有机电致发光化合物及其应用
WO2022043936A1 (fr) 2020-08-31 2022-03-03 Pfizer Inc. Procédés de protection de l'arn
KR102638321B1 (ko) * 2022-01-27 2024-02-19 마이크로바이오헬스케어 주식회사 바이오필름 형성 억제 활성을 갖는 신규 화합물 및 이의 용도

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4716035A (en) * 1985-05-24 1987-12-29 The Procter & Gamble Company Oral compositions and methods for treating gingivitis
WO2000044387A1 (fr) * 1999-01-29 2000-08-03 Nitto Kasei Co., Ltd. Composes organobores presentant une activite de coccidiostats
US7390806B2 (en) * 2002-12-18 2008-06-24 Anacor Pharmaceuticals, Inc. Antibiotics containing borinic acid complexes and methods of use
US20040224923A1 (en) * 2002-12-18 2004-11-11 Ving Lee Antibiotics containing borinic acid complexes and methods of use
ATE417052T1 (de) * 2003-09-02 2008-12-15 Yissum Res Dev Co Oxazaborolidine als bakterielle effektoren
AR049916A1 (es) * 2004-06-14 2006-09-13 Anacor Pharmaceuticals Inc Usos anti-parasitarios de complejos de acido borinico
AR049915A1 (es) * 2004-06-14 2006-09-13 Anacor Pharmaceuticals Inc Compuestos con contenido de boro y metodos de uso de los mismos

Also Published As

Publication number Publication date
EP2044091A4 (fr) 2010-08-04
IL195571A0 (en) 2009-09-01
KR20090029797A (ko) 2009-03-23
MX2008015918A (es) 2009-01-14
EP2044091A2 (fr) 2009-04-08
RU2008152367A (ru) 2010-07-20
BRPI0713010A2 (pt) 2012-10-09
WO2007146965A3 (fr) 2008-12-04
AU2007257689A1 (en) 2007-12-21
WO2007146965A2 (fr) 2007-12-21

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Legal Events

Date Code Title Description
FZDE Discontinued