RU2013152132A - Борсодержащие малые молекулы в качестве противовоспалительных средств - Google Patents
Борсодержащие малые молекулы в качестве противовоспалительных средств Download PDFInfo
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- RU2013152132A RU2013152132A RU2013152132/15A RU2013152132A RU2013152132A RU 2013152132 A RU2013152132 A RU 2013152132A RU 2013152132/15 A RU2013152132/15 A RU 2013152132/15A RU 2013152132 A RU2013152132 A RU 2013152132A RU 2013152132 A RU2013152132 A RU 2013152132A
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- 230000003110 anti-inflammatory effect Effects 0.000 title 1
- 150000003384 small molecules Chemical class 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 claims abstract 10
- 125000004404 heteroalkyl group Chemical group 0.000 claims abstract 10
- 125000003118 aryl group Chemical group 0.000 claims abstract 9
- 125000000753 cycloalkyl group Chemical group 0.000 claims abstract 9
- 125000001072 heteroaryl group Chemical group 0.000 claims abstract 9
- 125000000592 heterocycloalkyl group Chemical group 0.000 claims abstract 9
- 125000004093 cyano group Chemical group *C#N 0.000 claims abstract 8
- 229910052739 hydrogen Inorganic materials 0.000 claims abstract 8
- 208000031295 Animal disease Diseases 0.000 claims abstract 2
- ZOXJGFHDIHLPTG-UHFFFAOYSA-N Boron Chemical group [B] ZOXJGFHDIHLPTG-UHFFFAOYSA-N 0.000 claims abstract 2
- 206010061218 Inflammation Diseases 0.000 claims abstract 2
- 241001465754 Metazoa Species 0.000 claims abstract 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims abstract 2
- 229910052796 boron Inorganic materials 0.000 claims abstract 2
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 claims abstract 2
- 150000001875 compounds Chemical class 0.000 claims abstract 2
- 230000004054 inflammatory process Effects 0.000 claims abstract 2
- 229910052760 oxygen Inorganic materials 0.000 claims abstract 2
- 239000001301 oxygen Substances 0.000 claims abstract 2
- 150000003839 salts Chemical class 0.000 claims abstract 2
- 229910052717 sulfur Inorganic materials 0.000 claims abstract 2
- 239000011593 sulfur Substances 0.000 claims abstract 2
- 125000004429 atom Chemical group 0.000 claims 6
- 229910052736 halogen Inorganic materials 0.000 claims 2
- 150000002367 halogens Chemical class 0.000 claims 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 2
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 1
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Abstract
Способ лечения или профилактики у человека или животного заболевания, связанного с воспалением, при этом указанный способ включает введение человеку или животному терапевтически эффективного количества соединения, имеющего структуру, соответствующую формуле I:,где B представляет собой бор;Rявляется представителем, выбранным из группы, включающей отрицательный заряд, противоион соли, H, циано, замещенный или незамещенный алкил, замещенный или незамещенный гетероалкил, замещенный или незамещенный циклоалкил, замещенный или незамещенный гетероциклоалкил, замещенный или незамещенный арил и замещенный или незамещенный гетероарил;M является представителем, выбранным из кислорода, серы и NR;Rявляется представителем, выбранным из группы, включающей H, замещенный или незамещенный алкил, замещенный или незамещенный гетероалкил, замещенный или незамещенный циклоалкил, замещенный или незамещенный гетероциклоалкил, замещенный или незамещенный арил и замещенный или незамещенный гетероарил;J является представителем, выбранным из (CRR)и CR;R, Rи Rявляются представителями, независимо выбранными из группы, включающей H, циано, замещенный или незамещенный алкил, замещенный или незамещенный гетероалкил, замещенный или незамещенный циклоалкил, замещенный или незамещенный гетероциклоалкил, замещенный или незамещенный арил и замещенный или незамещенный гетероарил;n1 означает целое число, выбранное из 0-2;W является представителем, выбранным из C=O (карбонил), (CRR)и CR;R, Rи Rявляются представителями, независимо выбранными из группы, включающей H, циано, замещенный или незамещенный алкил, замещенный или незамещенный гетероалкил, замещ
Claims (1)
- Способ лечения или профилактики у человека или животного заболевания, связанного с воспалением, при этом указанный способ включает введение человеку или животному терапевтически эффективного количества соединения, имеющего структуру, соответствующую формуле I:где B представляет собой бор;R1a является представителем, выбранным из группы, включающей отрицательный заряд, противоион соли, H, циано, замещенный или незамещенный алкил, замещенный или незамещенный гетероалкил, замещенный или незамещенный циклоалкил, замещенный или незамещенный гетероциклоалкил, замещенный или незамещенный арил и замещенный или незамещенный гетероарил;M является представителем, выбранным из кислорода, серы и NR2a;R2a является представителем, выбранным из группы, включающей H, замещенный или незамещенный алкил, замещенный или незамещенный гетероалкил, замещенный или незамещенный циклоалкил, замещенный или незамещенный гетероциклоалкил, замещенный или незамещенный арил и замещенный или незамещенный гетероарил;J является представителем, выбранным из (CR3aR4a)n1 и CR5a;R3a, R4a и R5a являются представителями, независимо выбранными из группы, включающей H, циано, замещенный или незамещенный алкил, замещенный или незамещенный гетероалкил, замещенный или незамещенный циклоалкил, замещенный или незамещенный гетероциклоалкил, замещенный или незамещенный арил и замещенный или незамещенный гетероарил;n1 означает целое число, выбранное из 0-2;W является представителем, выбранным из C=O (карбонил), (CR6aR7a)m1 и CR8a;R6a, R7a и R8a являются представителями, независимо выбранными из группы, включающей H, циано, замещенный или незамещенный алкил, замещенный или незамещенный гетероалкил, замещенный или незамещенный циклоалкил, замещенный или незамещенный гетероциклоалкил, замещенный или незамещенный арил и замещенный или незамещенный гетероарил;m1 означает целое число, выбранное из 0 и 1;A является представителем, выбранным из CR9a и N;D является представителем, выбранным из CR10a и N;E является представителем, выбранным из CR11a и N;G является представителем, выбранным из CR12a и N;R9a, R10a, R11a и R12a являются представителями, независимо выбранными из группы, включающей H, OR*, NR*R**, SR*, -S(O)2R*, -S(O)2NR*R**, -C(O)R*, -C(O)OR*, -C(О)NR*R**, нитро, галоген, циано, замещенный или незамещенный алкил, замещенный или незамещенный гетероалкил, замещенный или незамещенный циклоалкил, замещенный или незамещенный гетероциклоалкил, замещенный или незамещенный арил и замещенный или незамещенный гетероарил;где каждый R* и R** являются представителями, независимо выбранными из группы, включающей H, нитро, галоген, циано, замещенный или незамещенный алкил, замещенный или незамещенный гетероалкил, замещенный или незамещенный циклоалкил, замещенный или незамещенный гетероциклоалкил, замещенный или незамещенный арил и замещенный или незамещенный гетероарил;сочетание атомов азота (A + D + E + G) означает целое число, выбранное из 0-3;представитель, выбранный из R3a, R4a и R5a, и представитель, выбранный из R6a, R7a и R8a, вместе с атомами, с которыми они связаны, необязательно объединяются с образованием 4-7-членного кольца;R3a и R4a вместе с атомами, с которыми они связаны, необязательно объединяются с образованием 4-7-членного кольца;R6a и R7a вместе с атомами, с которыми они связаны, необязательно объединяются с образованием 4-7-членного кольца;R9a и R10a вместе с атомами, с которыми они связаны, необязательно объединяются с образованием 4-7-членного кольца;R10a и R11a вместе с атомами, с которыми они связаны, необязательно объединяются с образованием 4-7-членного кольца;R11a и R12a вместе с атомами, с которыми они связаны, необязательно объединяются с образованием 4-7-членного кольца.
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