UY36950A - Compuestos útiles como inhibidores de la interacción proteína-proteína pd-1/pd-l1 y cd80/pd-l1 y composiciones que los contienen - Google Patents

Compuestos útiles como inhibidores de la interacción proteína-proteína pd-1/pd-l1 y cd80/pd-l1 y composiciones que los contienen

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Publication number
UY36950A
UY36950A UY0001036950A UY36950A UY36950A UY 36950 A UY36950 A UY 36950A UY 0001036950 A UY0001036950 A UY 0001036950A UY 36950 A UY36950 A UY 36950A UY 36950 A UY36950 A UY 36950A
Authority
UY
Uruguay
Prior art keywords
protein
inhibitors
compositions containing
useful compounds
compounds
Prior art date
Application number
UY0001036950A
Other languages
English (en)
Spanish (es)
Inventor
Kap-Sun Yeung
Timothy P Connolly
David B Frennesson
Katharine A Grant-Young
David R Langley
Zhaoxing Meng
Eric Mull
Kyle E Parcella
Mark George Saulnier
Li-Qiang SUN;
Juliang Zhu
Paul Michael Scola
Piyasena Hewawasam
Alan Xiangdong Wang
Ningning Xu
Original Assignee
Bristol-Myers Squibb Company Una Corporación Del Estado De Delaware
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Company Una Corporación Del Estado De Delaware filed Critical Bristol-Myers Squibb Company Una Corporación Del Estado De Delaware
Publication of UY36950A publication Critical patent/UY36950A/es

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    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
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    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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