UY32124A - Terapia combinada para tratar infección por hcv - Google Patents

Terapia combinada para tratar infección por hcv

Info

Publication number
UY32124A
UY32124A UY0001032124A UY32124A UY32124A UY 32124 A UY32124 A UY 32124A UY 0001032124 A UY0001032124 A UY 0001032124A UY 32124 A UY32124 A UY 32124A UY 32124 A UY32124 A UY 32124A
Authority
UY
Uruguay
Prior art keywords
hcv infection
combined therapy
treat hcv
compounds
relates
Prior art date
Application number
UY0001032124A
Other languages
English (en)
Inventor
Huang David
Gerhard G Steinmann
Jerry O Stern
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41571875&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY32124(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of UY32124A publication Critical patent/UY32124A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/7056Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing five-membered rings with nitrogen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/06Tripeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/19Cytokines; Lymphokines; Interferons
    • A61K38/21Interferons [IFN]
    • A61K38/212IFN-alpha
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

La presente invención se refiere a combinaciones terapéuticas que comprenden (a) Compuetos (1), o una sal farmacéuticamente aceptable del mismo, tal como se describe en el presente documento, (b) un interferón alfa y (c) ribavirina. El Compuetos (1) es un inhibidor selectivo y potente de la proteasa de serina NS3 de HCV. La presente invención se refiere también a métodos para emplear tales combinaciones terapéuticas para el tratamiento de infección por HCV o para aliviar uno o más síntomas de la misma en un paciente.
UY0001032124A 2008-09-17 2009-09-16 Terapia combinada para tratar infección por hcv UY32124A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US9775308P 2008-09-17 2008-09-17
US10903308P 2008-10-28 2008-10-28
US17193509P 2009-04-23 2009-04-23

Publications (1)

Publication Number Publication Date
UY32124A true UY32124A (es) 2010-04-30

Family

ID=41571875

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032124A UY32124A (es) 2008-09-17 2009-09-16 Terapia combinada para tratar infección por hcv

Country Status (25)

Country Link
US (1) US8399484B2 (es)
EP (1) EP2337583A1 (es)
JP (1) JP5539363B2 (es)
KR (1) KR20110054003A (es)
CN (1) CN102159245B (es)
AR (1) AR073516A1 (es)
AU (1) AU2009293493B2 (es)
BR (1) BRPI0918653A2 (es)
CA (1) CA2737376A1 (es)
CL (1) CL2011000571A1 (es)
CO (1) CO6351753A2 (es)
EA (1) EA019965B1 (es)
EC (1) ECSP11010877A (es)
HK (1) HK1156865A1 (es)
IL (1) IL210152A0 (es)
MA (1) MA32634B1 (es)
MX (1) MX2011002602A (es)
MY (1) MY152824A (es)
NZ (1) NZ591030A (es)
PE (1) PE20110343A1 (es)
TW (1) TWI454263B (es)
UA (1) UA103496C2 (es)
UY (1) UY32124A (es)
WO (1) WO2010033443A1 (es)
ZA (1) ZA201009151B (es)

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Also Published As

Publication number Publication date
CL2011000571A1 (es) 2011-07-29
TWI454263B (zh) 2014-10-01
JP2012502999A (ja) 2012-02-02
CN102159245B (zh) 2013-07-24
NZ591030A (en) 2012-10-26
CN102159245A (zh) 2011-08-17
UA103496C2 (uk) 2013-10-25
BRPI0918653A2 (pt) 2015-12-01
ZA201009151B (en) 2011-09-28
US8399484B2 (en) 2013-03-19
AR073516A1 (es) 2010-11-10
PE20110343A1 (es) 2011-06-25
TW201016218A (en) 2010-05-01
AU2009293493A1 (en) 2010-03-25
EP2337583A1 (en) 2011-06-29
AU2009293493B2 (en) 2014-09-18
WO2010033443A1 (en) 2010-03-25
CO6351753A2 (es) 2011-12-20
EA201100506A1 (ru) 2011-10-31
CA2737376A1 (en) 2010-03-25
ECSP11010877A (es) 2011-04-29
MX2011002602A (es) 2011-04-07
EA019965B1 (ru) 2014-07-30
MY152824A (en) 2014-11-28
US20100068182A1 (en) 2010-03-18
JP5539363B2 (ja) 2014-07-02
HK1156865A1 (en) 2012-06-22
IL210152A0 (en) 2011-03-31
MA32634B1 (fr) 2011-09-01
KR20110054003A (ko) 2011-05-24

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Effective date: 20181114