UY30761A1 - Derivados de 2.3-dihidroimidazo(1,2-c) quinazolina sustituida utiles para el tratamiento de enfermedades y trastornos hiper-proliferativos asociados con la angiogénesis - Google Patents

Derivados de 2.3-dihidroimidazo(1,2-c) quinazolina sustituida utiles para el tratamiento de enfermedades y trastornos hiper-proliferativos asociados con la angiogénesis

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Publication number
UY30761A1
UY30761A1 UY30761A UY30761A UY30761A1 UY 30761 A1 UY30761 A1 UY 30761A1 UY 30761 A UY30761 A UY 30761A UY 30761 A UY30761 A UY 30761A UY 30761 A1 UY30761 A1 UY 30761A1
Authority
UY
Uruguay
Prior art keywords
treatment
hyper
angiogenesis
diseases associated
kinazoline
Prior art date
Application number
UY30761A
Other languages
English (en)
Inventor
Robert William Scott
Aniko Redman
Ann-Marie Campbell
Dr Martin Michels
Martin F Hentemann
Ann-Marie Bullion
Jill E Wood
R Bruce Rowley
Original Assignee
Bayer Pharmaceuticals Corp
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39492563&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY30761(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Pharmaceuticals Corp filed Critical Bayer Pharmaceuticals Corp
Publication of UY30761A1 publication Critical patent/UY30761A1/es

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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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Abstract

RESUMEN Esta invencion se refiere a nuevos compuestos de 2,3-dihidroimodazo [1,2-c]quinazolina, a composiciones farmacéuticas que contienen dichos compuestos y a la utilizacion de esos compuestos o composiciones para la inhibicion de fosfotidilinositol-3-quinasa (P13K), y para el tratamiento de enfermedades asociadas con la actividad del fosfotidilinositol-3-quinasa (P13K) en particular para el tratamiento de transtornos de angiogénesis y/o hiper-proliferativos, como un agente unico o en combinacion con otros ingredientes activos.
UY30761A 2006-12-05 2007-12-04 Derivados de 2.3-dihidroimidazo(1,2-c) quinazolina sustituida utiles para el tratamiento de enfermedades y trastornos hiper-proliferativos asociados con la angiogénesis UY30761A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US87309006P 2006-12-05 2006-12-05

Publications (1)

Publication Number Publication Date
UY30761A1 true UY30761A1 (es) 2008-07-03

Family

ID=39492563

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30761A UY30761A1 (es) 2006-12-05 2007-12-04 Derivados de 2.3-dihidroimidazo(1,2-c) quinazolina sustituida utiles para el tratamiento de enfermedades y trastornos hiper-proliferativos asociados con la angiogénesis

Country Status (42)

Country Link
US (3) USRE46856E1 (es)
EP (1) EP2096919B1 (es)
JP (1) JP5326092B2 (es)
KR (1) KR101501785B1 (es)
CN (4) CN105254634B (es)
AR (1) AR064106A1 (es)
AU (1) AU2007328008B2 (es)
BR (1) BRPI0720178B8 (es)
CA (1) CA2671614C (es)
CL (1) CL2007003508A1 (es)
CO (1) CO6220908A2 (es)
CR (1) CR10838A (es)
CU (1) CU23796B7 (es)
DK (1) DK2096919T3 (es)
DO (1) DOP2009000135A (es)
EA (1) EA018839B1 (es)
EC (1) ECSP099387A (es)
ES (1) ES2572189T3 (es)
GT (1) GT200900154A (es)
HK (1) HK1217953A1 (es)
HN (1) HN2009001131A (es)
HU (1) HUE028773T2 (es)
IL (1) IL198273A (es)
JO (1) JO3147B1 (es)
MA (1) MA31283B1 (es)
MX (1) MX2009006001A (es)
MY (1) MY157944A (es)
NO (1) NO342348B1 (es)
NZ (1) NZ577342A (es)
PA (1) PA8759601A1 (es)
PE (1) PE20081444A1 (es)
PL (1) PL2096919T3 (es)
RS (1) RS56045B1 (es)
SG (1) SG177170A1 (es)
SI (1) SI2096919T1 (es)
SV (1) SV2009003288A (es)
TN (1) TN2009000137A1 (es)
TW (1) TWI406662B (es)
UA (1) UA96965C2 (es)
UY (1) UY30761A1 (es)
WO (1) WO2008070150A1 (es)
ZA (1) ZA200904691B (es)

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