UA81257C2 - Thiazolopyrimidinone compounds, pharmaceutical composition containing them and processes for the preparation thereof - Google Patents
Thiazolopyrimidinone compounds, pharmaceutical composition containing them and processes for the preparation thereof Download PDFInfo
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- UA81257C2 UA81257C2 UAA200501951A UA2005001951A UA81257C2 UA 81257 C2 UA81257 C2 UA 81257C2 UA A200501951 A UAA200501951 A UA A200501951A UA 2005001951 A UA2005001951 A UA 2005001951A UA 81257 C2 UA81257 C2 UA 81257C2
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- Ukraine
- Prior art keywords
- compound
- formula
- pharmaceutically acceptable
- acceptable salt
- solvate
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Landscapes
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Applications Claiming Priority (2)
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GBGB0221828.7A GB0221828D0 (en) | 2002-09-20 | 2002-09-20 | Novel compound |
PCT/GB2003/003998 WO2004026880A1 (en) | 2002-09-20 | 2003-09-16 | Novel compound |
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UAA200501951A UA81257C2 (en) | 2002-09-20 | 2003-09-16 | Thiazolopyrimidinone compounds, pharmaceutical composition containing them and processes for the preparation thereof |
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US (2) | US7585867B2 (ja) |
EP (1) | EP1543013B1 (ja) |
JP (1) | JP4619787B2 (ja) |
KR (1) | KR20050057427A (ja) |
CN (1) | CN1315848C (ja) |
AR (1) | AR041340A1 (ja) |
AT (1) | ATE419254T1 (ja) |
AU (1) | AU2003267571B2 (ja) |
BR (1) | BR0314844A (ja) |
CA (1) | CA2498762A1 (ja) |
DE (1) | DE60325614D1 (ja) |
DK (1) | DK1543013T3 (ja) |
ES (1) | ES2318152T3 (ja) |
GB (1) | GB0221828D0 (ja) |
HK (1) | HK1077060A1 (ja) |
IS (1) | IS7793A (ja) |
MX (1) | MXPA05002935A (ja) |
NO (1) | NO20051892L (ja) |
NZ (1) | NZ538826A (ja) |
PL (1) | PL375952A1 (ja) |
PT (1) | PT1543013E (ja) |
RU (1) | RU2342389C2 (ja) |
SI (1) | SI1543013T1 (ja) |
TW (1) | TW200413395A (ja) |
UA (1) | UA81257C2 (ja) |
WO (1) | WO2004026880A1 (ja) |
ZA (1) | ZA200502272B (ja) |
Families Citing this family (18)
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SE9903544D0 (sv) * | 1999-10-01 | 1999-10-01 | Astra Pharma Prod | Novel compounds |
GB2359551A (en) * | 2000-02-23 | 2001-08-29 | Astrazeneca Uk Ltd | Pharmaceutically active pyrimidine derivatives |
SE0003828D0 (sv) | 2000-10-20 | 2000-10-20 | Astrazeneca Ab | Novel compounds |
SE0102716D0 (sv) * | 2001-08-14 | 2001-08-14 | Astrazeneca Ab | Novel compounds |
GB0221829D0 (en) * | 2002-09-20 | 2002-10-30 | Astrazeneca Ab | Novel compound |
GB0221828D0 (en) | 2002-09-20 | 2002-10-30 | Astrazeneca Ab | Novel compound |
GB0328243D0 (en) * | 2003-12-05 | 2004-01-07 | Astrazeneca Ab | Methods |
UA90707C2 (en) | 2005-04-06 | 2010-05-25 | Астразенека Аб | Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives |
AR053347A1 (es) * | 2005-04-06 | 2007-05-02 | Astrazeneca Ab | Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos |
JP5305905B2 (ja) * | 2005-08-08 | 2013-10-02 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | チアゾロピリミジンキナーゼ阻害剤 |
PE20080145A1 (es) | 2006-03-21 | 2008-02-11 | Janssen Pharmaceutica Nv | Tetrahidro-pirimidoazepinas como moduladores de trpv1 |
TW200820973A (en) | 2006-09-29 | 2008-05-16 | Astrazeneca Ab | Novel compounds 480 |
PE20091102A1 (es) | 2007-12-17 | 2009-07-25 | Janssen Pharmaceutica Nv | Moduladores imidazolo-, oxazolo-, y tiazolopirimidina del trpv1 |
AR071036A1 (es) * | 2008-03-26 | 2010-05-19 | Astrazeneca Ab | Derivados 5, 7-disustituidos de [1, 3]tiazolo[4, 5-d]pirimidin-2 (3h)-ona, una composicion farmaceutica que los comprende y su uso en el tratamiento de enfermedades mediadas por el receptor cx3cr1. |
WO2009151910A2 (en) * | 2008-05-25 | 2009-12-17 | Wyeth | Combination product of receptor tyrosine kinase inhibitor and fatty acid synthase inhibitor for treating cancer |
JP5731538B2 (ja) | 2009-12-23 | 2015-06-10 | アイアンウッド ファーマシューティカルズ インコーポレイテッド | Crth2モジュレーター |
US20130216552A1 (en) | 2010-07-12 | 2013-08-22 | Ironwood Pharmaceuticals, Inc. | Crth2 modulators |
WO2012009134A1 (en) | 2010-07-12 | 2012-01-19 | Ironwood Pharmaceuticals, Inc. | Crth2 modulators |
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-
2002
- 2002-09-20 GB GBGB0221828.7A patent/GB0221828D0/en not_active Ceased
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2003
- 2003-09-16 MX MXPA05002935A patent/MXPA05002935A/es unknown
- 2003-09-16 DE DE60325614T patent/DE60325614D1/de not_active Expired - Lifetime
- 2003-09-16 RU RU2005106356/04A patent/RU2342389C2/ru not_active IP Right Cessation
- 2003-09-16 PL PL03375952A patent/PL375952A1/xx not_active Application Discontinuation
- 2003-09-16 NZ NZ538826A patent/NZ538826A/en unknown
- 2003-09-16 ES ES03748263T patent/ES2318152T3/es not_active Expired - Lifetime
- 2003-09-16 CA CA002498762A patent/CA2498762A1/en not_active Abandoned
- 2003-09-16 AU AU2003267571A patent/AU2003267571B2/en not_active Ceased
- 2003-09-16 KR KR1020057004643A patent/KR20050057427A/ko active IP Right Grant
- 2003-09-16 WO PCT/GB2003/003998 patent/WO2004026880A1/en active Application Filing
- 2003-09-16 UA UAA200501951A patent/UA81257C2/uk unknown
- 2003-09-16 SI SI200331519T patent/SI1543013T1/sl unknown
- 2003-09-16 EP EP03748263A patent/EP1543013B1/en not_active Expired - Lifetime
- 2003-09-16 JP JP2004537276A patent/JP4619787B2/ja not_active Expired - Fee Related
- 2003-09-16 BR BR0314844-0A patent/BR0314844A/pt not_active IP Right Cessation
- 2003-09-16 US US10/528,316 patent/US7585867B2/en not_active Expired - Fee Related
- 2003-09-16 AT AT03748263T patent/ATE419254T1/de not_active IP Right Cessation
- 2003-09-16 PT PT03748263T patent/PT1543013E/pt unknown
- 2003-09-16 DK DK03748263T patent/DK1543013T3/da active
- 2003-09-16 CN CNB03822335XA patent/CN1315848C/zh not_active Expired - Fee Related
- 2003-09-19 AR ARP030103432A patent/AR041340A1/es unknown
- 2003-09-19 TW TW092125983A patent/TW200413395A/zh unknown
-
2005
- 2005-03-17 ZA ZA200502272A patent/ZA200502272B/en unknown
- 2005-04-11 IS IS7793A patent/IS7793A/is unknown
- 2005-04-19 NO NO20051892A patent/NO20051892L/no not_active Application Discontinuation
- 2005-10-13 HK HK05109051.2A patent/HK1077060A1/xx not_active IP Right Cessation
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2007
- 2007-12-27 US US11/965,486 patent/US20080306262A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
BR0314844A (pt) | 2005-08-09 |
KR20050057427A (ko) | 2005-06-16 |
US7585867B2 (en) | 2009-09-08 |
EP1543013B1 (en) | 2008-12-31 |
CN1681826A (zh) | 2005-10-12 |
JP2006503835A (ja) | 2006-02-02 |
DE60325614D1 (de) | 2009-02-12 |
US20080306262A1 (en) | 2008-12-11 |
IS7793A (is) | 2005-04-11 |
ZA200502272B (en) | 2005-09-19 |
RU2342389C2 (ru) | 2008-12-27 |
NZ538826A (en) | 2006-12-22 |
TW200413395A (en) | 2004-08-01 |
SI1543013T1 (sl) | 2009-04-30 |
AR041340A1 (es) | 2005-05-11 |
AU2003267571A1 (en) | 2004-04-08 |
CN1315848C (zh) | 2007-05-16 |
NO20051892L (no) | 2005-06-17 |
EP1543013A1 (en) | 2005-06-22 |
DK1543013T3 (da) | 2009-03-09 |
PL375952A1 (en) | 2005-12-12 |
ATE419254T1 (de) | 2009-01-15 |
CA2498762A1 (en) | 2004-04-01 |
RU2005106356A (ru) | 2005-11-20 |
MXPA05002935A (es) | 2005-05-27 |
HK1077060A1 (en) | 2006-02-03 |
GB0221828D0 (en) | 2002-10-30 |
JP4619787B2 (ja) | 2011-01-26 |
PT1543013E (pt) | 2009-02-27 |
AU2003267571B2 (en) | 2007-08-16 |
WO2004026880A1 (en) | 2004-04-01 |
US20060100221A1 (en) | 2006-05-11 |
ES2318152T3 (es) | 2009-05-01 |
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