UA71938C2 - BENZYOXAZOLES AND PHENONES AS a2-ANTAGONISTS - Google Patents
BENZYOXAZOLES AND PHENONES AS a2-ANTAGONISTS Download PDFInfo
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- UA71938C2 UA71938C2 UA2001064352A UA2001064352A UA71938C2 UA 71938 C2 UA71938 C2 UA 71938C2 UA 2001064352 A UA2001064352 A UA 2001064352A UA 2001064352 A UA2001064352 A UA 2001064352A UA 71938 C2 UA71938 C2 UA 71938C2
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
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- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Psychiatry (AREA)
- Emergency Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Ophthalmology & Optometry (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Hospice & Palliative Care (AREA)
- Obesity (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP98204358 | 1998-12-21 | ||
| PCT/EP1999/010054 WO2000037466A1 (en) | 1998-12-21 | 1999-12-14 | BENZISOXAZOLES AND PHENONES AS α2-ANTAGONISTS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA71938C2 true UA71938C2 (en) | 2005-01-17 |
Family
ID=8234508
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UA2001064352A UA71938C2 (en) | 1998-12-21 | 1999-12-14 | BENZYOXAZOLES AND PHENONES AS a2-ANTAGONISTS |
Country Status (30)
| Country | Link |
|---|---|
| US (1) | US6576640B1 (xx) |
| EP (1) | EP1140934B1 (xx) |
| JP (1) | JP4717216B2 (xx) |
| KR (2) | KR20060093139A (xx) |
| CN (1) | CN1154646C (xx) |
| AR (1) | AR021924A1 (xx) |
| AT (1) | ATE251622T1 (xx) |
| AU (1) | AU765751B2 (xx) |
| BG (1) | BG65162B1 (xx) |
| BR (1) | BR9916427A (xx) |
| CA (1) | CA2355716C (xx) |
| CZ (1) | CZ294532B6 (xx) |
| DE (1) | DE69911995T2 (xx) |
| EA (1) | EA003606B1 (xx) |
| EE (1) | EE200100329A (xx) |
| ES (1) | ES2209553T3 (xx) |
| HK (1) | HK1045686B (xx) |
| HR (1) | HRP20010444A2 (xx) |
| HU (1) | HUP0104812A3 (xx) |
| ID (1) | ID28967A (xx) |
| IL (2) | IL143830A0 (xx) |
| NO (1) | NO317892B1 (xx) |
| NZ (1) | NZ511411A (xx) |
| PL (1) | PL196958B1 (xx) |
| SK (1) | SK285560B6 (xx) |
| TR (1) | TR200101813T2 (xx) |
| TW (1) | TWI229673B (xx) |
| UA (1) | UA71938C2 (xx) |
| WO (1) | WO2000037466A1 (xx) |
| ZA (1) | ZA200105067B (xx) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA04000036A (es) | 2001-07-05 | 2004-05-21 | Upjohn Co | Benzofuranos sustituidos con (hetero) arilo como ligandos 5-ht. |
| CA2480266C (en) * | 2002-04-03 | 2011-07-12 | Orion Corporation | Use of an alpha2-adrenoreceptor antagonist for cns-related diseases |
| EP1757605A4 (en) * | 2004-04-12 | 2007-12-19 | Taisho Pharmaceutical Co Ltd | CYCLIC AMINE COMPOUND |
| KR20080034171A (ko) * | 2005-07-28 | 2008-04-18 | 브리스톨-마이어스 스큅 컴퍼니 | 세로토닌 수용체 효능제 및 길항제로서의 치환된테트라히드로-1ｈ-피리도[4,3,ｂ]인돌 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3419568A (en) * | 1966-12-07 | 1968-12-31 | Abbott Lab | Derivatives of 1,2,3,4-tetrahydro-5h-pyrido[4,3b]indoles |
| US3382250A (en) * | 1966-12-07 | 1968-05-07 | Abbott Lab | Aroylalkyl derivatives of 1, 2, 3, 4-tetrahydro-5h-pyrido[4, 3b]indoles |
| US3718657A (en) * | 1970-12-03 | 1973-02-27 | Abbott Lab | Certain-2-substituted-1,2,3,4-tetrahydro-beta or gamma carbolines |
| JPS4729395U (xx) * | 1971-04-26 | 1972-12-04 | ||
| AR206812A1 (es) * | 1974-04-01 | 1976-08-23 | Pfizer | Compuestos intermediarios de azaciclo(3,4-a)indoles 4- y 5-fenil substituidos desprovistos de actividad terapeutica |
| US4001263A (en) * | 1974-04-01 | 1977-01-04 | Pfizer Inc. | 5-Aryl-1,2,3,4-tetrahydro-γ-carbolines |
| US4224329A (en) * | 1979-01-23 | 1980-09-23 | Pfizer Inc. | 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles |
| FR2570701B1 (fr) * | 1984-09-27 | 1987-05-22 | Synthelabo | Derives de furo(3,2-c)pyridines, leur preparation et leur application en therapeutique |
| DE3522959A1 (de) * | 1985-06-27 | 1987-01-08 | Merck Patent Gmbh | Indolderivate |
| EP0339959A3 (en) * | 1988-04-27 | 1991-03-20 | Glaxo Group Limited | Lactam derivatives |
| WO1994008040A1 (en) * | 1992-09-25 | 1994-04-14 | Synaptic Pharmaceutical Corporation | Dna encoding human alpha 1 adrenergic receptors and uses thereof |
| US5403847A (en) | 1992-11-13 | 1995-04-04 | Synaptic Pharmaceutical Corporation | Use of α1C specific compounds to treat benign prostatic hyperlasia |
| US5508306A (en) * | 1992-11-13 | 1996-04-16 | Synaptic Pharmaceutical Corporation | Aromatic amine derivatives |
| UA52681C2 (uk) * | 1997-04-08 | 2003-01-15 | Янссен Фармацевтика Н.В. | Похідні 1,2,3,4-тетрагідро-бензофуро[3,2,-c]піридину, спосіб їх одержання та фармацевтична композиція на їх основі |
-
1999
- 1999-12-14 US US09/868,756 patent/US6576640B1/en not_active Expired - Lifetime
- 1999-12-14 AU AU24327/00A patent/AU765751B2/en not_active Ceased
- 1999-12-14 CN CNB998147095A patent/CN1154646C/zh not_active Expired - Fee Related
- 1999-12-14 EP EP99967955A patent/EP1140934B1/en not_active Expired - Lifetime
- 1999-12-14 UA UA2001064352A patent/UA71938C2/uk unknown
- 1999-12-14 ID IDW00200101335A patent/ID28967A/id unknown
- 1999-12-14 ES ES99967955T patent/ES2209553T3/es not_active Expired - Lifetime
- 1999-12-14 KR KR1020067015507A patent/KR20060093139A/ko not_active Application Discontinuation
- 1999-12-14 HU HU0104812A patent/HUP0104812A3/hu unknown
- 1999-12-14 DE DE69911995T patent/DE69911995T2/de not_active Expired - Lifetime
- 1999-12-14 IL IL14383099A patent/IL143830A0/xx active IP Right Grant
- 1999-12-14 AT AT99967955T patent/ATE251622T1/de not_active IP Right Cessation
- 1999-12-14 CA CA2355716A patent/CA2355716C/en not_active Expired - Fee Related
- 1999-12-14 EE EEP200100329A patent/EE200100329A/xx unknown
- 1999-12-14 BR BR9916427-2A patent/BR9916427A/pt not_active Application Discontinuation
- 1999-12-14 WO PCT/EP1999/010054 patent/WO2000037466A1/en not_active Application Discontinuation
- 1999-12-14 SK SK858-2001A patent/SK285560B6/sk unknown
- 1999-12-14 JP JP2000589537A patent/JP4717216B2/ja not_active Expired - Fee Related
- 1999-12-14 KR KR1020017004946A patent/KR100657540B1/ko not_active IP Right Cessation
- 1999-12-14 PL PL348421A patent/PL196958B1/pl unknown
- 1999-12-14 NZ NZ511411A patent/NZ511411A/xx unknown
- 1999-12-14 TR TR2001/01813T patent/TR200101813T2/xx unknown
- 1999-12-14 EA EA200100709A patent/EA003606B1/ru not_active IP Right Cessation
- 1999-12-14 CZ CZ20012120A patent/CZ294532B6/cs not_active IP Right Cessation
- 1999-12-16 TW TW088122067A patent/TWI229673B/zh not_active IP Right Cessation
- 1999-12-20 AR ARP990106577A patent/AR021924A1/es active IP Right Grant
-
2001
- 2001-05-18 BG BG105521A patent/BG65162B1/bg unknown
- 2001-06-06 NO NO20012783A patent/NO317892B1/no unknown
- 2001-06-14 HR HR20010444A patent/HRP20010444A2/hr not_active Application Discontinuation
- 2001-06-19 IL IL143830A patent/IL143830A/en not_active IP Right Cessation
- 2001-06-20 ZA ZA200105067A patent/ZA200105067B/en unknown
-
2002
- 2002-07-09 HK HK02105098.8A patent/HK1045686B/zh not_active IP Right Cessation
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