AR206812A1 - Compuestos intermediarios de azaciclo(3,4-a)indoles 4- y 5-fenil substituidos desprovistos de actividad terapeutica - Google Patents

Compuestos intermediarios de azaciclo(3,4-a)indoles 4- y 5-fenil substituidos desprovistos de actividad terapeutica

Info

Publication number
AR206812A1
AR206812A1 AR258188A AR25818875A AR206812A1 AR 206812 A1 AR206812 A1 AR 206812A1 AR 258188 A AR258188 A AR 258188A AR 25818875 A AR25818875 A AR 25818875A AR 206812 A1 AR206812 A1 AR 206812A1
Authority
AR
Argentina
Prior art keywords
azaciclo
unproved
indoles
phenyl substituted
therapeutic activity
Prior art date
Application number
AR258188A
Other languages
English (en)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US456641A external-priority patent/US3925409A/en
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of AR206812A1 publication Critical patent/AR206812A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Anesthesiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
AR258188A 1974-04-01 1975-01-01 Compuestos intermediarios de azaciclo(3,4-a)indoles 4- y 5-fenil substituidos desprovistos de actividad terapeutica AR206812A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US45664074A 1974-04-01 1974-04-01
US456641A US3925409A (en) 1974-04-01 1974-04-01 4-Aryl-1,2,3,4-tetrahydropyrrolo{8 3,4-b{9 indoles

Publications (1)

Publication Number Publication Date
AR206812A1 true AR206812A1 (es) 1976-08-23

Family

ID=27038317

Family Applications (2)

Application Number Title Priority Date Filing Date
AR258188A AR206812A1 (es) 1974-04-01 1975-01-01 Compuestos intermediarios de azaciclo(3,4-a)indoles 4- y 5-fenil substituidos desprovistos de actividad terapeutica
AR261449A AR207799A1 (es) 1974-04-01 1975-01-01 Procedimiento para preparar azaciclo(3,4-a)-n-fenilindoles-2-substituidos

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR261449A AR207799A1 (es) 1974-04-01 1975-01-01 Procedimiento para preparar azaciclo(3,4-a)-n-fenilindoles-2-substituidos

Country Status (15)

Country Link
JP (1) JPS587635B2 (es)
AR (2) AR206812A1 (es)
AU (1) AU7955975A (es)
DD (1) DD118879A5 (es)
DE (1) DE2514084A1 (es)
DK (2) DK130575A (es)
ES (3) ES436157A1 (es)
FI (1) FI750940A (es)
FR (1) FR2265368A1 (es)
IL (1) IL46925A0 (es)
LU (1) LU72182A1 (es)
NL (1) NL7503700A (es)
NO (1) NO751055L (es)
RO (1) RO72884A (es)
SE (2) SE423630B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4224329A (en) * 1979-01-23 1980-09-23 Pfizer Inc. 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4451655A (en) * 1982-05-17 1984-05-29 Pfizer Inc. Process for preparing carboline derivatives and compounds used in their preparation
SK285560B6 (sk) * 1998-12-21 2007-03-01 Janssen Pharmaceutica N. V. Benzisoxazoly a fenoly ako alfa2-antagonisty, spôsob ich prípravy a farmaceutický prostriedok
RU2320662C1 (ru) * 2006-08-24 2008-03-27 Андрей Александрович Иващенко ЗАМЕЩЕННЫЕ ПИРРОЛО[4,3-b]ИНДОЛЫ, КОМБИНАТОРНАЯ И ФОКУСИРОВАННАЯ БИБЛИОТЕКИ, ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ, СПОСОБЫ ИХ ПОЛУЧЕНИЯ И ПРИМЕНЕНИЯ
JP5894574B2 (ja) * 2010-04-22 2016-03-30 イントラ−セルラー・セラピーズ・インコーポレイテッドIntra−Cellular Therapies, Inc. 有機化合物

Also Published As

Publication number Publication date
SE8200047L (sv) 1982-01-07
DK187878A (da) 1978-05-01
AR207799A1 (es) 1976-10-29
FI750940A (es) 1975-10-02
LU72182A1 (es) 1976-03-02
SE7502927L (es) 1975-10-02
SE423630B (sv) 1982-05-17
NL7503700A (nl) 1975-10-03
JPS50140494A (es) 1975-11-11
FR2265368B1 (es) 1978-07-28
DD118879A5 (es) 1976-03-20
DK130575A (es) 1975-10-02
RO72884A (ro) 1983-08-03
NO751055L (es) 1975-10-02
IL46925A0 (en) 1975-05-22
FR2265368A1 (en) 1975-10-24
AU7955975A (en) 1976-09-30
JPS587635B2 (ja) 1983-02-10
DE2514084A1 (de) 1975-11-20
ES453787A1 (es) 1978-01-01
RO72884B (ro) 1983-07-30
ES453788A1 (es) 1978-01-01
ES436157A1 (es) 1977-04-16

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