ES436157A1 - Un procedimiento para la preparacion de compuestos de indo- lina. - Google Patents

Un procedimiento para la preparacion de compuestos de indo- lina.

Info

Publication number
ES436157A1
ES436157A1 ES436157A ES436157A ES436157A1 ES 436157 A1 ES436157 A1 ES 436157A1 ES 436157 A ES436157 A ES 436157A ES 436157 A ES436157 A ES 436157A ES 436157 A1 ES436157 A1 ES 436157A1
Authority
ES
Spain
Prior art keywords
hydrogen
formula
chlorine
fluorine
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES436157A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US456641A external-priority patent/US3925409A/en
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES436157A1 publication Critical patent/ES436157A1/es
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Anesthesiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
ES436157A 1974-04-01 1975-03-31 Un procedimiento para la preparacion de compuestos de indo- lina. Expired ES436157A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US45664074A 1974-04-01 1974-04-01
US456641A US3925409A (en) 1974-04-01 1974-04-01 4-Aryl-1,2,3,4-tetrahydropyrrolo{8 3,4-b{9 indoles

Publications (1)

Publication Number Publication Date
ES436157A1 true ES436157A1 (es) 1977-04-16

Family

ID=27038317

Family Applications (3)

Application Number Title Priority Date Filing Date
ES436157A Expired ES436157A1 (es) 1974-04-01 1975-03-31 Un procedimiento para la preparacion de compuestos de indo- lina.
ES453788A Expired ES453788A1 (es) 1974-04-01 1976-11-30 Un procedimiento para la preparacion de compuestos de nido- lina.
ES453787A Expired ES453787A1 (es) 1974-04-01 1976-11-30 Un procedimiento para la preparacion de compuestos de nido- lina.

Family Applications After (2)

Application Number Title Priority Date Filing Date
ES453788A Expired ES453788A1 (es) 1974-04-01 1976-11-30 Un procedimiento para la preparacion de compuestos de nido- lina.
ES453787A Expired ES453787A1 (es) 1974-04-01 1976-11-30 Un procedimiento para la preparacion de compuestos de nido- lina.

Country Status (15)

Country Link
JP (1) JPS587635B2 (es)
AR (2) AR207799A1 (es)
AU (1) AU7955975A (es)
DD (1) DD118879A5 (es)
DE (1) DE2514084A1 (es)
DK (2) DK130575A (es)
ES (3) ES436157A1 (es)
FI (1) FI750940A (es)
FR (1) FR2265368A1 (es)
IL (1) IL46925A0 (es)
LU (1) LU72182A1 (es)
NL (1) NL7503700A (es)
NO (1) NO751055L (es)
RO (1) RO72884A (es)
SE (2) SE423630B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4224329A (en) * 1979-01-23 1980-09-23 Pfizer Inc. 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4451655A (en) * 1982-05-17 1984-05-29 Pfizer Inc. Process for preparing carboline derivatives and compounds used in their preparation
HUP0104812A3 (en) * 1998-12-21 2003-12-29 Janssen Pharmaceutica Nv Benzisoxazoles and phenones as alpha2-antagonists, process for their preparation and medicaments containing them
RU2320662C1 (ru) * 2006-08-24 2008-03-27 Андрей Александрович Иващенко ЗАМЕЩЕННЫЕ ПИРРОЛО[4,3-b]ИНДОЛЫ, КОМБИНАТОРНАЯ И ФОКУСИРОВАННАЯ БИБЛИОТЕКИ, ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ, СПОСОБЫ ИХ ПОЛУЧЕНИЯ И ПРИМЕНЕНИЯ
ES2602503T3 (es) * 2010-04-22 2017-02-21 Intra-Cellular Therapies, Inc. Compuestos orgánicos

Also Published As

Publication number Publication date
ES453788A1 (es) 1978-01-01
JPS587635B2 (ja) 1983-02-10
JPS50140494A (es) 1975-11-11
NO751055L (es) 1975-10-02
FI750940A (es) 1975-10-02
SE423630B (sv) 1982-05-17
SE7502927L (es) 1975-10-02
NL7503700A (nl) 1975-10-03
DK130575A (es) 1975-10-02
AR207799A1 (es) 1976-10-29
DD118879A5 (es) 1976-03-20
IL46925A0 (en) 1975-05-22
FR2265368A1 (en) 1975-10-24
SE8200047L (sv) 1982-01-07
RO72884B (ro) 1983-07-30
FR2265368B1 (es) 1978-07-28
RO72884A (ro) 1983-08-03
ES453787A1 (es) 1978-01-01
LU72182A1 (es) 1976-03-02
AU7955975A (en) 1976-09-30
DK187878A (da) 1978-05-01
AR206812A1 (es) 1976-08-23
DE2514084A1 (de) 1975-11-20

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