UA120632C2 - Тверді форми конденсованих гетероароматичних піролідинонів - Google Patents

Тверді форми конденсованих гетероароматичних піролідинонів Download PDF

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Publication number
UA120632C2
UA120632C2 UAA201707489A UAA201707489A UA120632C2 UA 120632 C2 UA120632 C2 UA 120632C2 UA A201707489 A UAA201707489 A UA A201707489A UA A201707489 A UAA201707489 A UA A201707489A UA 120632 C2 UA120632 C2 UA 120632C2
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UA
Ukraine
Prior art keywords
compound
still
cancer
shi
prd
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UAA201707489A
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English (en)
Ukrainian (uk)
Inventor
Жунлян Чень
Томонорі Ітібакасе
Томонори Итибакасе
Чуньжун Ма
Кристофер Меттьюс
Хадзіме Мотойосі
Хадзиме Мотойоси
Колін О'Брайан
Колин О'Брайан
Кентаро Ядзі
Кентаро Ядзи
Наокі Йосікава
Наоки ЙОСИКАВА
Original Assignee
Такеда Фармасьютікал Компані Лімітед
Такеда Фармасьютикал Компани Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=55299676&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA120632(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Такеда Фармасьютікал Компані Лімітед, Такеда Фармасьютикал Компани Лимитед filed Critical Такеда Фармасьютікал Компані Лімітед
Publication of UA120632C2 publication Critical patent/UA120632C2/uk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
UAA201707489A 2014-12-18 2015-12-17 Тверді форми конденсованих гетероароматичних піролідинонів UA120632C2 (uk)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201462093564P 2014-12-18 2014-12-18
US201562115223P 2015-02-12 2015-02-12
US201562180222P 2015-06-16 2015-06-16
PCT/IB2015/002489 WO2016097862A2 (en) 2014-12-18 2015-12-17 Solid state forms of fused heteroaromatic pyrrolidinones

Publications (1)

Publication Number Publication Date
UA120632C2 true UA120632C2 (uk) 2020-01-10

Family

ID=55299676

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201707489A UA120632C2 (uk) 2014-12-18 2015-12-17 Тверді форми конденсованих гетероароматичних піролідинонів

Country Status (29)

Country Link
US (3) US10676473B2 (enExample)
EP (2) EP3677582B1 (enExample)
JP (3) JP6778195B2 (enExample)
KR (1) KR102037502B1 (enExample)
CN (1) CN107108609B (enExample)
AU (1) AU2015365580B2 (enExample)
BR (1) BR112017013149B1 (enExample)
CA (1) CA2970864C (enExample)
CL (1) CL2017001561A1 (enExample)
CO (1) CO2017005910A2 (enExample)
CR (1) CR20170249A (enExample)
DK (1) DK3233857T3 (enExample)
DO (1) DOP2017000130A (enExample)
EA (1) EA032291B1 (enExample)
EC (1) ECSP17038100A (enExample)
ES (1) ES2788454T3 (enExample)
GE (2) GEP20197050B (enExample)
IL (1) IL252941B (enExample)
MX (1) MX373586B (enExample)
MY (1) MY199935A (enExample)
NZ (1) NZ732371A (enExample)
PE (1) PE20171179A1 (enExample)
PH (1) PH12017501123A1 (enExample)
PL (1) PL3233857T3 (enExample)
SG (1) SG11201701911QA (enExample)
TN (1) TN2017000080A1 (enExample)
UA (1) UA120632C2 (enExample)
WO (1) WO2016097862A2 (enExample)
ZA (1) ZA201701800B (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL3233857T3 (pl) * 2014-12-18 2020-07-27 Takeda Pharmaceutical Company Limited Stałe postacie skondensowanych heteroaromatycznych pirolidynonów
JP2019520419A (ja) * 2016-07-13 2019-07-18 武田薬品工業株式会社 脾臓チロシンキナーゼ阻害剤と他の治療薬の併用
AU2018350683A1 (en) 2017-10-19 2020-04-02 Bayer Animal Health Gmbh Use of fused heteroaromatic pyrrolidones for treatment and prevention of diseases in animals
WO2019088039A1 (en) 2017-10-30 2019-05-09 Takeda Pharmaceutical Company Limited Treatment of acute myeloid leukemia
MY208604A (en) 2018-12-14 2025-05-20 Chia Tai Tianqing Pharmaceutical Group Co Ltd Salt of syk inhibitor and crystalline form thereof
MX2021009521A (es) 2019-02-07 2021-09-08 Janssen Biotech Inc Inhibidores de dihidroorotato deshidrogenasa.
TW202104207A (zh) 2019-04-17 2021-02-01 美商健生生物科技公司 二氫乳清酸脫氫酶抑制劑
CN114630822B (zh) 2019-10-10 2024-10-01 詹森生物科技公司 联芳基二氢乳清酸脱氢酶抑制剂
UY38988A (es) 2019-12-19 2021-06-30 Janssen Pharmaceutica Nv Derivados espiráncos sustituidos de cadena lineal
WO2022074534A1 (en) 2020-10-05 2022-04-14 Janssen Biotech, Inc. Combinations of dihydroorotate dehydrogenase inhibitors and hypomethylating agents
CN115698005B (zh) * 2020-12-18 2024-02-06 山东轩竹医药科技有限公司 稠环类AhR抑制剂
AU2022274071A1 (en) 2021-05-11 2024-01-04 Janssen Pharmaceutica Nv Combination therapies
KR20240006638A (ko) 2021-05-11 2024-01-15 얀센 파마슈티카 엔브이 조합 요법
KR102539612B1 (ko) 2021-12-24 2023-06-02 엘에스일렉트릭(주) IP 기반 RAPIEnet을 지원하는 통신 디바이스 및 이를 포함하는 네트워크 시스템
JP2025540759A (ja) 2022-11-30 2025-12-16 ヤンセン ファーマシューティカ エヌ.ベー. メニン-mll阻害剤及び少なくとも1つの他の治療剤を含む組み合わせ
JP2025540762A (ja) 2022-11-30 2025-12-16 ヤンセン ファーマシューティカ エヌ.ベー. メニン-mll阻害剤及びbcl-2阻害剤を含む組み合わせ
AU2024400853A1 (en) 2023-12-15 2026-05-28 Ishihara Sangyo Kaisha, Ltd. N-substituted oxy-2-aminothiazolecarboxamide compound or salt thereof and agricultural and horticultural fungicide

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1960372B1 (en) * 2005-12-15 2015-12-09 Rigel Pharmaceuticals, Inc. Kinase inhibitors and their uses
EP2516434B1 (en) 2009-12-23 2015-05-27 Takeda Pharmaceutical Company Limited Fused heteroaromatic pyrrolidinones as syk inhibitors
WO2012177714A1 (en) 2011-06-22 2012-12-27 Takeda Pharmaceutical Company Limited Substituted 6-aza-isoindolin-1-one derivatives
WO2016048982A2 (en) * 2014-09-24 2016-03-31 Millennium Pharmaceuticals, Inc. COMBINATION TREATMENT WITH PI3Kα INHIBITORS AND TAXANES
PL3233857T3 (pl) * 2014-12-18 2020-07-27 Takeda Pharmaceutical Company Limited Stałe postacie skondensowanych heteroaromatycznych pirolidynonów

Also Published As

Publication number Publication date
US10676473B2 (en) 2020-06-09
ES2788454T3 (es) 2020-10-21
CA2970864A1 (en) 2016-06-23
CA2970864C (en) 2020-04-14
EA032291B1 (ru) 2019-05-31
WO2016097862A2 (en) 2016-06-23
CN107108609A (zh) 2017-08-29
JP2020143081A (ja) 2020-09-10
MX2017007162A (es) 2017-08-28
CR20170249A (es) 2017-09-25
BR112017013149A2 (pt) 2018-04-10
EA201791369A1 (ru) 2017-10-31
GEP20197050B (en) 2019-12-10
KR102037502B1 (ko) 2019-10-28
EP3233857A2 (en) 2017-10-25
DK3233857T3 (da) 2020-04-27
EP3233857B1 (en) 2020-03-11
ECSP17038100A (es) 2017-12-01
GEAP201914545A (en) 2019-08-12
BR112017013149B1 (pt) 2022-10-11
IL252941A0 (en) 2017-08-31
KR20170095374A (ko) 2017-08-22
JP6974534B2 (ja) 2021-12-01
EP3677582B1 (en) 2023-01-25
DOP2017000130A (es) 2017-07-15
JP6778195B2 (ja) 2020-10-28
CN107108609B (zh) 2020-02-18
US20230348461A1 (en) 2023-11-02
TN2017000080A1 (en) 2018-07-04
ZA201701800B (en) 2020-05-27
PL3233857T3 (pl) 2020-07-27
CO2017005910A2 (es) 2017-10-20
AU2015365580A1 (en) 2017-07-06
PE20171179A1 (es) 2017-08-22
US20200339573A1 (en) 2020-10-29
PH12017501123A1 (en) 2017-11-27
NZ732371A (en) 2023-04-28
US11352355B2 (en) 2022-06-07
SG11201701911QA (en) 2017-04-27
IL252941B (en) 2020-11-30
MY199935A (en) 2023-11-29
CL2017001561A1 (es) 2018-01-12
HK1243406A1 (zh) 2018-07-13
WO2016097862A3 (en) 2016-08-11
AU2015365580B2 (en) 2020-04-02
EP3677582A1 (en) 2020-07-08
MX373586B (es) 2020-05-05
JP2022017477A (ja) 2022-01-25
US20160176869A1 (en) 2016-06-23
JP2017537969A (ja) 2017-12-21

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