UA113291C2 - Метаболіти транскломіфену і їх застосування - Google Patents
Метаболіти транскломіфену і їх застосування Download PDFInfo
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- UA113291C2 UA113291C2 UAA201402168A UAA201402168A UA113291C2 UA 113291 C2 UA113291 C2 UA 113291C2 UA A201402168 A UAA201402168 A UA A201402168A UA A201402168 A UAA201402168 A UA A201402168A UA 113291 C2 UA113291 C2 UA 113291C2
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- clomiphene
- trans
- metabolite
- pharmaceutical composition
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Classifications
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- C07C217/04—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C217/06—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted
- C07C217/14—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring
- C07C217/18—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring the six-membered aromatic ring or condensed ring system containing that ring being further substituted
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- A—HUMAN NECESSITIES
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161515278P | 2011-08-04 | 2011-08-04 | |
| PCT/US2012/049451 WO2013020017A1 (en) | 2011-08-04 | 2012-08-03 | Trans-clomiphene metabolites and uses thereof |
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| Publication Number | Publication Date |
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| UA113291C2 true UA113291C2 (xx) | 2017-01-10 |
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| Application Number | Title | Priority Date | Filing Date |
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| UAA201402168A UA113291C2 (xx) | 2011-08-04 | 2012-03-08 | Метаболіти транскломіфену і їх застосування |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US9981906B2 (https=) |
| EP (2) | EP3351527A1 (https=) |
| JP (2) | JP6433785B2 (https=) |
| KR (1) | KR20140054110A (https=) |
| CN (1) | CN103702975B (https=) |
| AU (2) | AU2012289964B2 (https=) |
| BR (1) | BR112014000908A2 (https=) |
| CA (1) | CA2841572C (https=) |
| CL (1) | CL2014000268A1 (https=) |
| CO (1) | CO6862154A2 (https=) |
| CR (1) | CR20140124A (https=) |
| EA (1) | EA201490416A1 (https=) |
| IL (1) | IL230287B (https=) |
| MX (1) | MX355316B (https=) |
| MY (2) | MY191802A (https=) |
| NI (1) | NI201400008A (https=) |
| PH (1) | PH12014500144A1 (https=) |
| SG (1) | SG10201606425WA (https=) |
| UA (1) | UA113291C2 (https=) |
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Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20120284764A1 (en) * | 2011-05-05 | 2012-11-08 | Keith Ball | Method and system for requesting services by a media device |
| UA113291C2 (xx) | 2011-08-04 | 2017-01-10 | Метаболіти транскломіфену і їх застосування | |
| SG11201407397WA (en) | 2012-05-31 | 2014-12-30 | Repros Therapeutics Inc | Formulations and methods for vaginal delivery of antiprogestins |
| ES2688821T3 (es) | 2012-11-02 | 2018-11-07 | Repros Therapeutics Inc. | Métodos y composiciones para tratar afecciones dependientes de la progesterona |
| WO2014070523A1 (en) * | 2012-11-02 | 2014-05-08 | Repros Therapeutics Inc. | Trans-clomiphene for use in cancer therapy |
| WO2017123577A1 (en) * | 2016-01-12 | 2017-07-20 | Repros Therapeutics Inc. | Trans-clomiphene and progesterone receptor antagonist combination therapy for treating hormone-dependent conditions |
| CN108883083A (zh) * | 2016-02-25 | 2018-11-23 | 艾森潘帕克制药股份有限公司 | 两种氯米芬异构体的口服剂型及使用其治疗继发性腺功能减退症的方法 |
| WO2017182097A1 (en) | 2016-04-22 | 2017-10-26 | F.I.S. - Fabbrica Italiana Sintetici S.P.A. | Process for the preparation of enclomiphene citrate having needle shaped crystal habit. |
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2012
- 2012-03-08 UA UAA201402168A patent/UA113291C2/uk unknown
- 2012-08-03 JP JP2014524097A patent/JP6433785B2/ja not_active Expired - Fee Related
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- 2012-08-03 MY MYPI2017001676A patent/MY191802A/en unknown
- 2012-08-03 KR KR1020147004588A patent/KR20140054110A/ko not_active Ceased
- 2012-08-03 WO PCT/US2012/049451 patent/WO2013020017A1/en not_active Ceased
- 2012-08-03 PH PH1/2014/500144A patent/PH12014500144A1/en unknown
- 2012-08-03 BR BR112014000908A patent/BR112014000908A2/pt active Search and Examination
- 2012-08-03 EA EA201490416A patent/EA201490416A1/ru unknown
- 2012-08-03 EP EP18161551.9A patent/EP3351527A1/en not_active Withdrawn
- 2012-08-03 SG SG10201606425WA patent/SG10201606425WA/en unknown
- 2012-08-03 CN CN201280038230.6A patent/CN103702975B/zh not_active Expired - Fee Related
- 2012-08-03 EP EP12750508.9A patent/EP2744777A1/en not_active Withdrawn
- 2012-08-03 MY MYPI2014000022A patent/MY170718A/en unknown
- 2012-08-03 US US14/236,868 patent/US9981906B2/en not_active Expired - Fee Related
- 2012-08-03 MX MX2014000825A patent/MX355316B/es active IP Right Grant
- 2012-08-03 CA CA2841572A patent/CA2841572C/en not_active Expired - Fee Related
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2014
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- 2014-01-17 ZA ZA2014/00406A patent/ZA201400406B/en unknown
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- 2014-01-30 NI NI201400008A patent/NI201400008A/es unknown
- 2014-02-03 CL CL2014000268A patent/CL2014000268A1/es unknown
- 2014-03-13 CR CR20140124A patent/CR20140124A/es unknown
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2017
- 2017-06-20 AU AU2017204171A patent/AU2017204171A1/en not_active Abandoned
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2018
- 2018-10-01 JP JP2018186696A patent/JP2019023210A/ja active Pending
Also Published As
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|---|---|
| US20140163114A1 (en) | 2014-06-12 |
| EP2744777A1 (en) | 2014-06-25 |
| CN103702975A (zh) | 2014-04-02 |
| NI201400008A (es) | 2015-12-10 |
| US9981906B2 (en) | 2018-05-29 |
| EA201490416A1 (ru) | 2014-11-28 |
| AU2012289964A1 (en) | 2014-01-30 |
| KR20140054110A (ko) | 2014-05-08 |
| PH12014500144A1 (en) | 2014-02-24 |
| CL2014000268A1 (es) | 2014-11-14 |
| HK1196349A1 (zh) | 2014-12-12 |
| JP2014529584A (ja) | 2014-11-13 |
| SG10201606425WA (en) | 2016-09-29 |
| JP2019023210A (ja) | 2019-02-14 |
| IL230287B (en) | 2019-07-31 |
| NZ621892A (en) | 2016-03-31 |
| EP3351527A1 (en) | 2018-07-25 |
| BR112014000908A2 (pt) | 2017-02-21 |
| CO6862154A2 (es) | 2014-02-10 |
| CA2841572A1 (en) | 2013-02-07 |
| AU2012289964B2 (en) | 2017-03-23 |
| MX355316B (es) | 2018-04-16 |
| CN103702975B (zh) | 2016-03-16 |
| WO2013020017A1 (en) | 2013-02-07 |
| JP6433785B2 (ja) | 2018-12-05 |
| CA2841572C (en) | 2020-10-13 |
| MY191802A (en) | 2022-07-15 |
| ZA201400406B (en) | 2014-11-26 |
| MX2014000825A (es) | 2014-02-27 |
| AU2017204171A1 (en) | 2017-07-13 |
| IL230287A0 (en) | 2014-03-06 |
| CR20140124A (es) | 2014-05-13 |
| MY170718A (en) | 2019-08-27 |
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