HK1216502A1 - 用於癌症治療的反式-克羅米芬 - Google Patents

用於癌症治療的反式-克羅米芬

Info

Publication number
HK1216502A1
HK1216502A1 HK16104449.1A HK16104449A HK1216502A1 HK 1216502 A1 HK1216502 A1 HK 1216502A1 HK 16104449 A HK16104449 A HK 16104449A HK 1216502 A1 HK1216502 A1 HK 1216502A1
Authority
HK
Hong Kong
Prior art keywords
cancer therapy
trans clomiphene
clomiphene
trans
cancer
Prior art date
Application number
HK16104449.1A
Other languages
English (en)
Inventor
Joseph S Podolski
Ronald D Wiehle
Kuang Hsu
Greg Fontenot
Original Assignee
Repros Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Repros Therapeutics Inc filed Critical Repros Therapeutics Inc
Publication of HK1216502A1 publication Critical patent/HK1216502A1/zh

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
HK16104449.1A 2012-11-02 2016-04-19 用於癌症治療的反式-克羅米芬 HK1216502A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261722013P 2012-11-02 2012-11-02
PCT/US2013/066141 WO2014070523A1 (en) 2012-11-02 2013-10-22 Trans-clomiphene for use in cancer therapy

Publications (1)

Publication Number Publication Date
HK1216502A1 true HK1216502A1 (zh) 2016-11-18

Family

ID=50627954

Family Applications (1)

Application Number Title Priority Date Filing Date
HK16104449.1A HK1216502A1 (zh) 2012-11-02 2016-04-19 用於癌症治療的反式-克羅米芬

Country Status (10)

Country Link
US (1) US9687458B2 (zh)
EP (1) EP2914294A1 (zh)
JP (3) JP2015535283A (zh)
CN (1) CN104994877A (zh)
AU (1) AU2013338311A1 (zh)
CA (1) CA2889770A1 (zh)
HK (1) HK1216502A1 (zh)
IL (1) IL238453A0 (zh)
MX (1) MX2015005160A (zh)
WO (1) WO2014070523A1 (zh)

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WO2016022325A1 (en) * 2014-08-05 2016-02-11 The Penn State Research Foundation Novel triarylethylene compounds and methods using same
CN108348605B (zh) 2015-11-10 2023-06-09 帕拉卡林治疗公司 用pdgf-cc抑制剂和抗雌激素治疗er阴性乳癌
JP2018002619A (ja) * 2016-06-29 2018-01-11 国立大学法人 東京大学 オートファジー阻害剤
EP3515424A4 (en) * 2016-09-26 2020-05-06 Repros Therapeutics Inc. ANTI-ESTROGEN AND / OR AROMATASE INHIBITORS FOR USE IN THE TREATMENT OF ADIPOSITAS AND RELATED SYMPTOMS
CN108420806A (zh) * 2017-02-15 2018-08-21 武汉华杰世纪生物医药有限公司 具有靶向性的抗肿瘤药物
WO2019236209A2 (en) * 2018-04-27 2019-12-12 Jin Byung Ju Methods for high-content drug screening

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Also Published As

Publication number Publication date
US20150283099A1 (en) 2015-10-08
JP2021046448A (ja) 2021-03-25
MX2015005160A (es) 2015-07-17
IL238453A0 (en) 2015-06-30
WO2014070523A1 (en) 2014-05-08
JP2018123168A (ja) 2018-08-09
CN104994877A (zh) 2015-10-21
US9687458B2 (en) 2017-06-27
EP2914294A1 (en) 2015-09-09
CA2889770A1 (en) 2014-05-08
AU2013338311A1 (en) 2015-05-14
JP2015535283A (ja) 2015-12-10

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