TW201722413A - 用於治療肥胖及肥胖相關病症之包含卡格列淨（ｃａｎａｇｌｉｆｌｏｚｉｎ）與芬特明（ｐｈｅｎｔｅｒｍｉｎｅ）的協同治療 - Google Patents

用於治療肥胖及肥胖相關病症之包含卡格列淨（ｃａｎａｇｌｉｆｌｏｚｉｎ）與芬特明（ｐｈｅｎｔｅｒｍｉｎｅ）的協同治療 Download PDF

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Publication number
TW201722413A
TW201722413A TW105129698A TW105129698A TW201722413A TW 201722413 A TW201722413 A TW 201722413A TW 105129698 A TW105129698 A TW 105129698A TW 105129698 A TW105129698 A TW 105129698A TW 201722413 A TW201722413 A TW 201722413A
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Taiwan
Prior art keywords
phentermine
administered
amount
obesity
subject
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TW105129698A
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English (en)
Chinese (zh)
Inventor
Norman R Rosenthal
Paul Rothenberg
David C Polidori
Douglas K Ways
peter p Stein
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Janssen Pharmaceutica Nv
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Publication of TW201722413A publication Critical patent/TW201722413A/zh

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Emergency Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
TW105129698A 2015-09-15 2016-09-13 用於治療肥胖及肥胖相關病症之包含卡格列淨（ｃａｎａｇｌｉｆｌｏｚｉｎ）與芬特明（ｐｈｅｎｔｅｒｍｉｎｅ）的協同治療 TW201722413A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562218842P 2015-09-15 2015-09-15
US201662306110P 2016-03-10 2016-03-10
US15/262,038 US20170071970A1 (en) 2015-09-15 2016-09-12 Co-therapy comprising canagliflozin and phentermine for the treatment of obesity and obesity related disorders

Publications (1)

Publication Number Publication Date
TW201722413A true TW201722413A (zh) 2017-07-01

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
TW105129698A TW201722413A (zh) 2015-09-15 2016-09-13 用於治療肥胖及肥胖相關病症之包含卡格列淨（ｃａｎａｇｌｉｆｌｏｚｉｎ）與芬特明（ｐｈｅｎｔｅｒｍｉｎｅ）的協同治療

Country Status (18)

Country Link
US (3) US20170071970A1 (enExample)
EP (1) EP3349740B1 (enExample)
JP (1) JP2018527374A (enExample)
KR (1) KR20180051560A (enExample)
CN (1) CN108024977A (enExample)
AU (1) AU2016322537B2 (enExample)
CA (1) CA2998730A1 (enExample)
CO (1) CO2018002708A2 (enExample)
EA (1) EA201890738A1 (enExample)
ES (1) ES2873117T3 (enExample)
HK (1) HK1248124A1 (enExample)
IL (1) IL257876A (enExample)
MX (1) MX383002B (enExample)
PH (1) PH12018500501A1 (enExample)
TW (1) TW201722413A (enExample)
UA (1) UA122974C2 (enExample)
WO (1) WO2017048670A1 (enExample)
ZA (1) ZA201802448B (enExample)

Families Citing this family (6)

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TWI835735B (zh) * 2017-06-12 2024-03-21 比利時商健生藥品公司 減少或預防第ii型糖尿病患者中心血管事件之方法
CN110038009B (zh) * 2019-05-13 2021-01-08 浙江大学 卡格列净在制备抗肿瘤药物中的应用
MX2022009844A (es) * 2020-02-18 2022-09-05 Novo Nordisk As Composiciones y usos del peptido similar al glucagon-1 (glp-1).
CN112716940A (zh) * 2021-02-18 2021-04-30 苏州大学 卡格列净在制备治疗与stat6蛋白相关疾病的药物中的应用
CN113812378B (zh) * 2021-09-29 2023-02-03 湖北天勤生物技术研究院有限公司 一种食蟹猴肥胖症模型的建立方法及其应用
CN113893349B (zh) * 2021-12-13 2022-07-22 北京大学第三医院（北京大学第三临床医学院） 达格列净及其类似物在制备防治雄性生殖功能障碍的药物中的用途

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