TW200720249A - Pyrrolidine compound - Google Patents

Pyrrolidine compound

Info

Publication number
TW200720249A
TW200720249A TW095116220A TW95116220A TW200720249A TW 200720249 A TW200720249 A TW 200720249A TW 095116220 A TW095116220 A TW 095116220A TW 95116220 A TW95116220 A TW 95116220A TW 200720249 A TW200720249 A TW 200720249A
Authority
TW
Taiwan
Prior art keywords
pyrrolidine compound
salt
halogen atoms
present
phenyl group
Prior art date
Application number
TW095116220A
Other languages
English (en)
Other versions
TWI410406B (zh
Inventor
Muneaki Kurimura
Shinichi Taira
Takahiro Tomoyasu
Nobuaki Ito
Kuninori Tai
Noriaki Takemura
Takayuki Matsuzaki
Yasuhiro Menjo
Shin Miyamura
Yohji Sakurai
Akihito Watanabe
Yasuyo Sakata
Takumi Masumoto
Kohei Akazawa
Haruhiko Sugino
Naoki Amada
Satoshi Ohashi
Tomoichi Shinohara
Hirofumi Sasaki
Chisako Morita
Junko Yamashita
Satoko Nakajima
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36693623&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TW200720249(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of TW200720249A publication Critical patent/TW200720249A/zh
Application granted granted Critical
Publication of TWI410406B publication Critical patent/TWI410406B/zh

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    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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  • Organic Chemistry (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
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  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Cardiology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Psychology (AREA)
  • Physical Education & Sports Medicine (AREA)
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  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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TW095116220A 2005-05-13 2006-05-08 吡咯烷化合物 TWI410406B (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2005141230 2005-05-13

Publications (2)

Publication Number Publication Date
TW200720249A true TW200720249A (en) 2007-06-01
TWI410406B TWI410406B (zh) 2013-10-01

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TW102143870A TWI449692B (zh) 2005-05-13 2006-05-08 吡咯烷化合物（三）
TW102101997A TWI439452B (zh) 2005-05-13 2006-05-08 吡咯烷化合物（二）
TW095116220A TWI410406B (zh) 2005-05-13 2006-05-08 吡咯烷化合物

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TW102143870A TWI449692B (zh) 2005-05-13 2006-05-08 吡咯烷化合物（三）
TW102101997A TWI439452B (zh) 2005-05-13 2006-05-08 吡咯烷化合物（二）

Country Status (24)

Country Link
US (6) US8084442B2 (zh)
EP (2) EP1881975B8 (zh)
JP (1) JP4776631B2 (zh)
KR (2) KR20100038453A (zh)
CN (3) CN101175748A (zh)
AR (1) AR054191A1 (zh)
AU (2) AU2006244851B2 (zh)
BR (1) BRPI0610279A2 (zh)
CA (1) CA2608184C (zh)
CY (1) CY1114767T1 (zh)
DK (1) DK2407451T3 (zh)
ES (2) ES2451523T3 (zh)
IL (1) IL187311A (zh)
IN (1) IN2012DN00758A (zh)
MX (1) MX2007014252A (zh)
MY (1) MY148653A (zh)
PL (1) PL2407451T3 (zh)
PT (1) PT2407451E (zh)
RU (1) RU2414454C2 (zh)
SG (1) SG162722A1 (zh)
SI (1) SI2407451T1 (zh)
TW (3) TWI449692B (zh)
WO (1) WO2006121218A1 (zh)
ZA (1) ZA200709691B (zh)

Families Citing this family (21)

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Publication number Priority date Publication date Assignee Title
SG173922A1 (en) 2002-11-27 2011-09-29 Incyte Corp 3-aminopyrrolidine derivatives as modulators of chemokine receptors
TWI449692B (zh) * 2005-05-13 2014-08-21 Otsuka Pharma Co Ltd 吡咯烷化合物（三）
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