TW200519104A - Quinazoline derivatives - Google Patents

Quinazoline derivatives

Info

Publication number
TW200519104A
TW200519104A TW093127785A TW93127785A TW200519104A TW 200519104 A TW200519104 A TW 200519104A TW 093127785 A TW093127785 A TW 093127785A TW 93127785 A TW93127785 A TW 93127785A TW 200519104 A TW200519104 A TW 200519104A
Authority
TW
Taiwan
Prior art keywords
quinazoline derivatives
formula
medicament
diseases
expected
Prior art date
Application number
TW093127785A
Other languages
English (en)
Inventor
Christopher Thomas Halsall
Laurent Francois Andre Hennequin
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34315440&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TW200519104(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB0321620.7A external-priority patent/GB0321620D0/en
Priority claimed from GB0406163A external-priority patent/GB0406163D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of TW200519104A publication Critical patent/TW200519104A/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C04—CEMENTS; CONCRETE; ARTIFICIAL STONE; CERAMICS; REFRACTORIES
    • C04B—LIME, MAGNESIA; SLAG; CEMENTS; COMPOSITIONS THEREOF, e.g. MORTARS, CONCRETE OR LIKE BUILDING MATERIALS; ARTIFICIAL STONE; CERAMICS; REFRACTORIES; TREATMENT OF NATURAL STONE
    • C04B35/00—Shaped ceramic products characterised by their composition; Ceramics compositions; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/622—Forming processes; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/626—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B
    • C04B35/63—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
    • C04B35/632—Organic additives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
TW093127785A 2003-09-16 2004-09-14 Quinazoline derivatives TW200519104A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0321620.7A GB0321620D0 (en) 2003-09-16 2003-09-16 Quinazoline derivatives
GB0406163A GB0406163D0 (en) 2004-03-19 2004-03-19 Quinazoline derivatives

Publications (1)

Publication Number Publication Date
TW200519104A true TW200519104A (en) 2005-06-16

Family

ID=34315440

Family Applications (1)

Application Number Title Priority Date Filing Date
TW093127785A TW200519104A (en) 2003-09-16 2004-09-14 Quinazoline derivatives

Country Status (25)

Country Link
US (2) US7569577B2 (zh)
EP (1) EP1667991B1 (zh)
JP (1) JP4795952B2 (zh)
AR (1) AR045663A1 (zh)
AT (1) ATE395346T1 (zh)
AU (1) AU2004272348B2 (zh)
BR (1) BRPI0414489A8 (zh)
CA (1) CA2538884C (zh)
CO (1) CO5690594A2 (zh)
CY (1) CY1108186T1 (zh)
DE (1) DE602004013806D1 (zh)
DK (1) DK1667991T3 (zh)
ES (1) ES2305844T3 (zh)
HK (1) HK1091480A1 (zh)
HR (1) HRP20080329T3 (zh)
IL (1) IL174261A0 (zh)
MX (1) MXPA06002964A (zh)
NO (1) NO20061322L (zh)
PL (1) PL1667991T3 (zh)
PT (1) PT1667991E (zh)
RU (1) RU2378268C2 (zh)
SI (1) SI1667991T1 (zh)
TW (1) TW200519104A (zh)
UA (1) UA84167C2 (zh)
WO (1) WO2005026150A1 (zh)

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US8017321B2 (en) * 2004-01-23 2011-09-13 The Regents Of The University Of Colorado, A Body Corporate Gefitinib sensitivity-related gene expression and products and methods related thereto
US20080113874A1 (en) * 2004-01-23 2008-05-15 The Regents Of The University Of Colorado Gefitinib sensitivity-related gene expression and products and methods related thereto
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ES2537631T3 (es) * 2004-05-27 2015-06-10 The Regents Of The University Of Colorado Métodos para la predicción del resultado clínico para inhibidores del receptor del factor de crecimiento epidérmico para pacientes de cáncer
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CN102452988B (zh) 2010-10-27 2016-01-27 中国科学院化学研究所 一种喹唑啉衍生物及其制备方法
KR101940340B1 (ko) 2011-03-04 2019-01-18 글락소스미스클라인 인털렉츄얼 프로퍼티 디벨로프먼트 리미티드 키나제 억제제로서의 아미노-퀴놀린
TWI547494B (zh) 2011-08-18 2016-09-01 葛蘭素史克智慧財產發展有限公司 作為激酶抑制劑之胺基喹唑啉類
AR092529A1 (es) * 2012-09-13 2015-04-22 Glaxosmithkline Llc Compuesto de aminoquinazolina, composicion farmaceutica que lo comprende y uso de dicho compuesto para la preparacion de un medicamento
TW201425307A (zh) 2012-09-13 2014-07-01 Glaxosmithkline Llc 作為激酶抑制劑之胺基－喹啉類
KR20150118152A (ko) 2013-02-21 2015-10-21 글락소스미스클라인 인털렉츄얼 프로퍼티 디벨로프먼트 리미티드 키나제 억제제로서의 퀴나졸린
JP7265985B2 (ja) 2016-11-17 2023-04-27 ボード オブ リージェンツ，ザ ユニバーシティ オブ テキサス システム Ｅｇｆｒまたはｈｅｒ２のエクソン２０変異を有するがん細胞に対する抗腫瘍活性を有する化合物

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Also Published As

Publication number Publication date
AU2004272348B2 (en) 2008-09-04
UA84167C2 (ru) 2008-09-25
RU2378268C2 (ru) 2010-01-10
HRP20080329T3 (en) 2008-08-31
CA2538884A1 (en) 2005-03-24
EP1667991B1 (en) 2008-05-14
CY1108186T1 (el) 2014-02-12
HK1091480A1 (en) 2007-01-19
SI1667991T1 (sl) 2008-10-31
RU2006112599A (ru) 2007-11-10
DE602004013806D1 (en) 2008-06-26
PL1667991T3 (pl) 2008-12-31
PT1667991E (pt) 2008-07-14
DK1667991T3 (da) 2008-08-18
ES2305844T3 (es) 2008-11-01
EP1667991A1 (en) 2006-06-14
ATE395346T1 (de) 2008-05-15
BRPI0414489A (pt) 2006-11-14
US7569577B2 (en) 2009-08-04
NO20061322L (no) 2006-06-15
CO5690594A2 (es) 2006-10-31
AU2004272348A1 (en) 2005-03-24
MXPA06002964A (es) 2006-06-14
BRPI0414489A8 (pt) 2019-01-15
WO2005026150A1 (en) 2005-03-24
CA2538884C (en) 2010-09-21
JP2007505872A (ja) 2007-03-15
IL174261A0 (en) 2006-08-01
JP4795952B2 (ja) 2011-10-19
US20090312343A1 (en) 2009-12-17
AR045663A1 (es) 2005-11-02
US20070043009A1 (en) 2007-02-22

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