SV2010003718A - Inhibidores de bace - Google Patents

Inhibidores de bace

Info

Publication number
SV2010003718A
SV2010003718A SV2010003718A SV2010003718A SV2010003718A SV 2010003718 A SV2010003718 A SV 2010003718A SV 2010003718 A SV2010003718 A SV 2010003718A SV 2010003718 A SV2010003718 A SV 2010003718A SV 2010003718 A SV2010003718 A SV 2010003718A
Authority
SV
El Salvador
Prior art keywords
bace inhibitors
methods
inhibitors
bace
formula
Prior art date
Application number
SV2010003718A
Other languages
English (en)
Spanish (es)
Inventor
James Edmund Audia
Dusin James Mergott
Scott Martin Sheehan
Brian Morgan Watson
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40839645&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SV2010003718(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of SV2010003718A publication Critical patent/SV2010003718A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/04—1,3-Thiazines; Hydrogenated 1,3-thiazines
    • C07D279/06—1,3-Thiazines; Hydrogenated 1,3-thiazines not condensed with other rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SV2010003718A 2008-05-02 2010-10-29 Inhibidores de bace SV2010003718A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US4988108P 2008-05-02 2008-05-02

Publications (1)

Publication Number Publication Date
SV2010003718A true SV2010003718A (es) 2011-02-14

Family

ID=40839645

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2010003718A SV2010003718A (es) 2008-05-02 2010-10-29 Inhibidores de bace

Country Status (32)

Country Link
US (1) US7648983B2 (da)
EP (1) EP2297120B1 (da)
JP (3) JP5658139B2 (da)
KR (1) KR101253835B1 (da)
CN (1) CN102015667B (da)
AR (1) AR071187A1 (da)
AU (1) AU2009241515B2 (da)
CA (1) CA2723207C (da)
CL (1) CL2009000860A1 (da)
CO (1) CO6311079A2 (da)
CR (1) CR11776A (da)
DK (1) DK2297120T3 (da)
DO (1) DOP2010000328A (da)
EA (1) EA016955B1 (da)
EC (1) ECSP10010582A (da)
ES (1) ES2549087T3 (da)
HR (1) HRP20150941T1 (da)
HU (1) HUE025520T2 (da)
IL (1) IL208350A (da)
MA (1) MA32351B1 (da)
MX (1) MX2010011972A (da)
NZ (1) NZ588300A (da)
PE (1) PE20091816A1 (da)
PL (1) PL2297120T3 (da)
PT (1) PT2297120E (da)
RS (1) RS54260B1 (da)
SI (1) SI2297120T1 (da)
SV (1) SV2010003718A (da)
TW (1) TWI431004B (da)
UA (1) UA102251C2 (da)
WO (1) WO2009134617A1 (da)
ZA (1) ZA201006868B (da)

Families Citing this family (86)

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EP2151435A4 (en) 2007-04-24 2011-09-14 Shionogi & Co PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF ALZHEIMER'S DISEASE
ES2548774T3 (es) * 2008-01-18 2015-10-20 Eisai R&D Management Co., Ltd. Derivado de aminodihidrotiazina condensado
EP2283016B1 (en) 2008-04-22 2014-09-24 Merck Sharp & Dohme Corp. Thiophenyl-substituted 2-imino-3-methyl pyrrolo pyrimidinone compounds as bace-1 inhibitors, compositions, and their use
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EP2514747A4 (en) 2009-12-09 2013-05-08 Shionogi & Co SUBSTITUTED AMINOTHIAZINE DERIVATIVE
CN102834384A (zh) 2009-12-11 2012-12-19 盐野义制药株式会社 *嗪衍生物
WO2011077726A1 (ja) 2009-12-24 2011-06-30 塩野義製薬株式会社 ４－アミノ－１，３－チアジンまたはオキサジン誘導体
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JP5853033B2 (ja) 2011-03-01 2016-02-09 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプＪａｎｓｓｅｎ Ｐｈａｒｍａｃｅｕｔｉｃａ Ｎａａｍｌｏｚｅ Ｖｅｎｎｏｏｔｓｃｈａｐ β−セクレターゼ（ＢＡＣＥ）の阻害剤として有用な６，７−ジヒドロ−ピラゾロ［１，５−ａ］ピラジン−４−イルアミン誘導体
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Also Published As

Publication number Publication date
PE20091816A1 (es) 2009-11-25
CO6311079A2 (es) 2011-08-22
CN102015667B (zh) 2013-06-12
EP2297120A1 (en) 2011-03-23
SI2297120T1 (sl) 2015-11-30
EP2297120B1 (en) 2015-08-19
TW200946522A (en) 2009-11-16
CR11776A (es) 2011-01-28
JP5658139B2 (ja) 2015-01-21
PT2297120E (pt) 2015-10-26
HUE025520T2 (en) 2016-02-29
US20090275566A1 (en) 2009-11-05
MA32351B1 (fr) 2011-06-01
DOP2010000328A (es) 2010-11-15
AR071187A1 (es) 2010-06-02
KR20100125475A (ko) 2010-11-30
TWI431004B (zh) 2014-03-21
JP2011519854A (ja) 2011-07-14
NZ588300A (en) 2012-07-27
CA2723207A1 (en) 2009-11-05
JP2015051980A (ja) 2015-03-19
US7648983B2 (en) 2010-01-19
WO2009134617A1 (en) 2009-11-05
AU2009241515A1 (en) 2009-11-05
CA2723207C (en) 2016-07-12
MX2010011972A (es) 2010-11-25
KR101253835B1 (ko) 2013-04-15
IL208350A (en) 2014-05-28
HRP20150941T1 (hr) 2015-10-09
AU2009241515B2 (en) 2012-04-19
CL2009000860A1 (es) 2010-05-07
UA102251C2 (ru) 2013-06-25
EA016955B1 (ru) 2012-08-30
PL2297120T3 (pl) 2016-01-29
IL208350A0 (en) 2010-12-30
RS54260B1 (en) 2016-02-29
DK2297120T3 (da) 2015-10-12
ES2549087T3 (es) 2015-10-22
ZA201006868B (en) 2012-03-28
JP2017048212A (ja) 2017-03-09
ECSP10010582A (es) 2010-11-30
CN102015667A (zh) 2011-04-13
EA201071264A1 (ru) 2011-04-29

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