SU895291A3 - Способ получени производных 4-амино-2-пиперидинохиназолина или их солей с фармацевтически приемлимыми кислотами - Google Patents

Способ получени производных 4-амино-2-пиперидинохиназолина или их солей с фармацевтически приемлимыми кислотами Download PDF

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Publication number
SU895291A3
SU895291A3 SU802877159A SU2877159A SU895291A3 SU 895291 A3 SU895291 A3 SU 895291A3 SU 802877159 A SU802877159 A SU 802877159A SU 2877159 A SU2877159 A SU 2877159A SU 895291 A3 SU895291 A3 SU 895291A3
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SU
USSR - Soviet Union
Prior art keywords
vacuo
piperidine
chloroform
solvent
solution
Prior art date
Application number
SU802877159A
Other languages
English (en)
Russian (ru)
Inventor
Фрейзер Кэмпбелл Саймон
Кристофер Данилевич Джон
Вильямс Гринграсс Колин
Original Assignee
Пфайзер Корпорейшн (Фирма)
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Application filed by Пфайзер Корпорейшн (Фирма) filed Critical Пфайзер Корпорейшн (Фирма)
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Publication of SU895291A3 publication Critical patent/SU895291A3/ru

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/46Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SU802877159A 1979-01-31 1980-01-30 Способ получени производных 4-амино-2-пиперидинохиназолина или их солей с фармацевтически приемлимыми кислотами SU895291A3 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7903398 1979-01-31

Publications (1)

Publication Number Publication Date
SU895291A3 true SU895291A3 (ru) 1981-12-30

Family

ID=10502852

Family Applications (1)

Application Number Title Priority Date Filing Date
SU802877159A SU895291A3 (ru) 1979-01-31 1980-01-30 Способ получени производных 4-амино-2-пиперидинохиназолина или их солей с фармацевтически приемлимыми кислотами

Country Status (28)

Country Link
JP (1) JPS55104278A (fi)
AR (1) AR222208A1 (fi)
AT (1) AT373595B (fi)
BE (1) BE881448A (fi)
CA (1) CA1131636A (fi)
CS (1) CS231970B2 (fi)
DD (1) DD148720A5 (fi)
DE (1) DE3003323A1 (fi)
DK (1) DK540879A (fi)
ES (1) ES488129A0 (fi)
FI (1) FI63936C (fi)
FR (1) FR2447919A1 (fi)
GR (1) GR73626B (fi)
HU (1) HU184233B (fi)
IE (1) IE800178L (fi)
IL (1) IL59252A (fi)
IT (1) IT1149902B (fi)
LU (1) LU82115A1 (fi)
NL (1) NL8000571A (fi)
NO (1) NO800230L (fi)
NZ (1) NZ192744A (fi)
PH (1) PH15436A (fi)
PL (1) PL121890B1 (fi)
PT (1) PT70749A (fi)
SE (1) SE8000699L (fi)
SU (1) SU895291A3 (fi)
YU (1) YU22980A (fi)
ZA (1) ZA80557B (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2483920A1 (fr) * 1980-06-09 1981-12-11 Synthelabo Nouveaux derives de quinazoline, leur procede de preparation et leur application en therapeutique
ES515338A0 (es) * 1981-09-09 1983-11-01 Orion Yhtymae Oy "metodo para la preparacion de piperidinilquinazolidinas substituidas".
US5280032A (en) * 1989-02-14 1994-01-18 Toyama Chemical Co., Ltd. 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
WO2013070852A2 (en) * 2011-11-08 2013-05-16 Emory University Compounds and compositions used to epigenetically transform cells and methods related thereto

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1088068A (en) * 1977-11-16 1980-10-21 Simon F. Campbell Piperidino-quinazolines
GB2021108B (en) * 1978-05-18 1982-07-21 Pfizer Ltd 6,7 - di - 4 - amino - 2 - quinazolines

Also Published As

Publication number Publication date
NL8000571A (nl) 1980-08-04
GR73626B (fi) 1984-03-26
FI63936C (fi) 1983-09-12
AT373595B (de) 1984-02-10
SE8000699L (sv) 1980-08-01
PT70749A (en) 1980-02-01
JPS5728711B2 (fi) 1982-06-18
YU22980A (en) 1983-02-28
IT1149902B (it) 1986-12-10
CS60780A2 (en) 1984-01-16
PL121890B1 (en) 1982-06-30
IE800178L (en) 1980-07-31
AR222208A1 (es) 1981-04-30
FI63936B (fi) 1983-05-31
CA1131636A (en) 1982-09-14
PL221683A1 (fi) 1980-12-01
NZ192744A (en) 1984-03-30
DE3003323A1 (de) 1980-08-14
PH15436A (en) 1983-01-18
AU5502480A (en) 1980-08-07
ES8101583A1 (es) 1980-12-16
HU184233B (en) 1984-07-30
DK540879A (da) 1980-08-01
IT8019537A0 (it) 1980-01-29
FR2447919A1 (fr) 1980-08-29
IL59252A (en) 1983-11-30
LU82115A1 (fr) 1980-04-23
JPS55104278A (en) 1980-08-09
FR2447919B1 (fi) 1983-02-11
CS231970B2 (en) 1985-01-16
ZA80557B (en) 1981-08-26
IL59252A0 (en) 1980-05-30
FI800252A (fi) 1980-08-01
ATA46980A (de) 1983-06-15
ES488129A0 (es) 1980-12-16
NO800230L (no) 1980-08-01
BE881448A (fr) 1980-07-30
DD148720A5 (de) 1981-06-10

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