SK286461B6 - [1,5-a]-Pyrazolo-1,3,5-triazíny, ich použitie a farmaceutické kompozície na ich báze - Google Patents
[1,5-a]-Pyrazolo-1,3,5-triazíny, ich použitie a farmaceutické kompozície na ich báze Download PDFInfo
- Publication number
- SK286461B6 SK286461B6 SK97-99A SK9799A SK286461B6 SK 286461 B6 SK286461 B6 SK 286461B6 SK 9799 A SK9799 A SK 9799A SK 286461 B6 SK286461 B6 SK 286461B6
- Authority
- SK
- Slovakia
- Prior art keywords
- formula
- compounds
- ome
- nhch
- alkyl
- Prior art date
Links
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Detergent Compositions (AREA)
- Coloring (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US68604796A | 1996-07-24 | 1996-07-24 | |
US2329096P | 1996-07-24 | 1996-07-24 | |
US08/899,242 US6124289A (en) | 1996-07-24 | 1997-07-23 | Azolo triazines and pyrimidines |
PCT/US1997/013072 WO1998003510A1 (en) | 1996-07-24 | 1997-07-23 | AZOLO TRIAZINES AND PYRIMIDINES |
Publications (2)
Publication Number | Publication Date |
---|---|
SK9799A3 SK9799A3 (sk) | 2005-04-01 |
SK286461B6 true SK286461B6 (sk) | 2008-10-07 |
Family
ID=27362048
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SK97-99A SK286461B6 (sk) | 1996-07-24 | 1997-07-23 | [1,5-a]-Pyrazolo-1,3,5-triazíny, ich použitie a farmaceutické kompozície na ich báze |
Country Status (15)
Country | Link |
---|---|
JP (2) | JP4704521B2 (no) |
CN (3) | CN1104432C (no) |
AR (1) | AR049583A2 (no) |
BR (1) | BR9710544A (no) |
CA (1) | CA2259583C (no) |
CZ (1) | CZ299451B6 (no) |
EA (1) | EA004403B1 (no) |
EE (1) | EE04316B1 (no) |
HR (1) | HRP970413A2 (no) |
IL (4) | IL127871A0 (no) |
NO (1) | NO315610B1 (no) |
NZ (1) | NZ333777A (no) |
PL (1) | PL195762B1 (no) |
SI (1) | SI9720045B (no) |
SK (1) | SK286461B6 (no) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR0208357A (pt) * | 2001-03-13 | 2004-06-29 | Bristol Myers Squibb Pharma Co | Composto, composição farmacêutica, método de antagonização de um receptor de fator de liberação de corticotropina (crf), método de tratamento de disfunção, método de triagem de ligantes, método de detecção de receptores de crf, método de inibição da ligação de crf, artigo industrializado e usos do composto |
WO2004110454A1 (ja) * | 2003-06-13 | 2004-12-23 | Ishihara Sangyo Kaisha, Ltd. | アデノシンA2a受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物 |
US7329662B2 (en) * | 2003-10-03 | 2008-02-12 | Hoffmann-La Roche Inc. | Pyrazolo-pyridine |
GB0519957D0 (en) * | 2005-09-30 | 2005-11-09 | Sb Pharmco Inc | Chemical compound |
UA96458C2 (ru) * | 2006-09-20 | 2011-11-10 | Эли Лилли Энд Компани | Тиазолпиразолопиримидиновые соединения как антагонисты рецептора crf1 |
CN103694242B (zh) * | 2013-12-10 | 2016-01-06 | 昆明翔昊科技有限公司 | 吡唑并嘧啶类化合物及其药物组合物和其在制药中的应用 |
AU2018317398A1 (en) | 2017-08-14 | 2019-11-21 | Spruce Biosciences, Inc. | Corticotropin releasing factor receptor antagonists |
CN112592346B (zh) * | 2019-07-30 | 2022-04-26 | 厦门宝太生物科技股份有限公司 | 一种a2a和/或a2b抑制剂中间体的制备方法 |
MX2023001688A (es) | 2020-08-12 | 2023-02-22 | Spruce Biosciences Inc | Metodos y composiciones para tratar el sindrome de ovario poliquistico. |
US11708372B2 (en) | 2021-11-19 | 2023-07-25 | Spruce Biosciences, Inc. | Crystalline composition of tildacerfont and methods of use and preparation thereof |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3995039A (en) * | 1975-05-27 | 1976-11-30 | Merck & Co., Inc. | Pyrazolo [1,5-a] [1,3,5] triazines |
JPS6157587A (ja) * | 1984-08-29 | 1986-03-24 | Shionogi & Co Ltd | 縮合複素環誘導体および抗潰瘍剤 |
US4824834A (en) * | 1986-10-31 | 1989-04-25 | Otsuka Pharmaceutical Company, Limited | Pyrazolotriazine compounds |
JP2691317B2 (ja) * | 1989-08-25 | 1997-12-17 | 株式会社大塚製薬工場 | 4―ヒドロキシ―8―(3―低級アルコキシ―4―フェニルスルフィニルフェニル)ピラゾロ〔1,5―a〕―1,3,5―トリアジン光学活性体の塩類及びその製造方法 |
WO1992006096A1 (en) * | 1990-10-09 | 1992-04-16 | Otsuka Pharmaceutical Co., Ltd. | Pyrimidine derivative, production thereof, and androgen inhibitor |
ES2126573T3 (es) * | 1991-04-22 | 1999-04-01 | Otsuka Pharma Co Ltd | Derivado de pirazol (1,5-a)pirimidina y agente antiinflamatorio que contiene este derivado. |
US5356897A (en) * | 1991-09-09 | 1994-10-18 | Fujisawa Pharmaceutical Co., Ltd. | 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines |
-
1997
- 1997-07-23 CA CA002259583A patent/CA2259583C/en not_active Expired - Lifetime
- 1997-07-23 EA EA199900158A patent/EA004403B1/ru not_active IP Right Cessation
- 1997-07-23 SK SK97-99A patent/SK286461B6/sk not_active IP Right Cessation
- 1997-07-23 NZ NZ333777A patent/NZ333777A/en not_active IP Right Cessation
- 1997-07-23 CN CN97196525A patent/CN1104432C/zh not_active Expired - Lifetime
- 1997-07-23 IL IL12787197A patent/IL127871A0/xx unknown
- 1997-07-23 SI SI9720045A patent/SI9720045B/sl active Search and Examination
- 1997-07-23 EE EEP199900019A patent/EE04316B1/xx unknown
- 1997-07-23 BR BR9710544A patent/BR9710544A/pt not_active IP Right Cessation
- 1997-07-23 JP JP50723398A patent/JP4704521B2/ja not_active Expired - Fee Related
- 1997-07-23 PL PL97331523A patent/PL195762B1/pl unknown
- 1997-07-23 CZ CZ0018499A patent/CZ299451B6/cs not_active IP Right Cessation
- 1997-07-24 HR HRP970413 patent/HRP970413A2/hr not_active Application Discontinuation
-
1998
- 1998-12-30 IL IL127871A patent/IL127871A/en not_active IP Right Cessation
-
1999
- 1999-01-21 NO NO19990264A patent/NO315610B1/no not_active IP Right Cessation
-
2001
- 2001-05-30 CN CN 01120849 patent/CN1250223C/zh not_active Expired - Lifetime
-
2002
- 2002-04-25 CN CN 02118589 patent/CN1388126A/zh active Pending
- 2002-06-11 IL IL150163A patent/IL150163A/en not_active IP Right Cessation
-
2004
- 2004-07-23 JP JP2004216483A patent/JP4194539B2/ja not_active Expired - Fee Related
- 2004-10-12 IL IL164513A patent/IL164513A/en not_active IP Right Cessation
-
2005
- 2005-07-11 AR ARP050102868A patent/AR049583A2/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
SI9720045B (sl) | 2008-02-29 |
EA199900158A1 (ru) | 1999-10-28 |
PL331523A1 (en) | 1999-07-19 |
JP2005097257A (ja) | 2005-04-14 |
IL127871A0 (en) | 1999-10-28 |
JP4194539B2 (ja) | 2008-12-10 |
IL127871A (en) | 2010-04-29 |
SI9720045A (sl) | 1999-10-31 |
PL195762B1 (pl) | 2007-10-31 |
NO990264L (no) | 1999-03-10 |
CN1104432C (zh) | 2003-04-02 |
EE9900019A (et) | 1999-08-16 |
NZ333777A (en) | 2000-07-28 |
AR049583A2 (es) | 2006-08-16 |
IL164513A0 (en) | 2005-12-18 |
CN1250223C (zh) | 2006-04-12 |
NO990264D0 (no) | 1999-01-21 |
CN1388126A (zh) | 2003-01-01 |
CN1225637A (zh) | 1999-08-11 |
JP2002513382A (ja) | 2002-05-08 |
CZ299451B6 (cs) | 2008-07-30 |
CA2259583C (en) | 2009-11-17 |
HRP970413A2 (en) | 1998-10-31 |
SK9799A3 (sk) | 2005-04-01 |
JP4704521B2 (ja) | 2011-06-15 |
CZ18499A3 (cs) | 1999-11-17 |
CA2259583A1 (en) | 1998-01-29 |
NO315610B3 (no) | 2003-09-29 |
NO315610B1 (no) | 2003-09-29 |
IL150163A (en) | 2010-12-30 |
EE04316B1 (et) | 2004-06-15 |
IL164513A (en) | 2010-04-29 |
EA004403B1 (ru) | 2004-04-29 |
BR9710544A (pt) | 1999-08-17 |
CN1327793A (zh) | 2001-12-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MK4A | Expiry of patent |
Expiry date: 20170723 |