SK286461B6 - [1,5-a]-Pyrazolo-1,3,5-triazíny, ich použitie a farmaceutické kompozície na ich báze - Google Patents

[1,5-a]-Pyrazolo-1,3,5-triazíny, ich použitie a farmaceutické kompozície na ich báze Download PDF

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Publication number
SK286461B6
SK286461B6 SK97-99A SK9799A SK286461B6 SK 286461 B6 SK286461 B6 SK 286461B6 SK 9799 A SK9799 A SK 9799A SK 286461 B6 SK286461 B6 SK 286461B6
Authority
SK
Slovakia
Prior art keywords
formula
compounds
ome
nhch
alkyl
Prior art date
Application number
SK97-99A
Other languages
English (en)
Slovak (sk)
Other versions
SK9799A3 (sk
Inventor
Argyrios Georgious Arvanitis
Robert John Chorvat
Ligi He
Paul Joseph Gilligan
Original Assignee
Bristol-Myers Squibb Pharma Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Pharma Company filed Critical Bristol-Myers Squibb Pharma Company
Priority claimed from US08/899,242 external-priority patent/US6124289A/en
Priority claimed from PCT/US1997/013072 external-priority patent/WO1998003510A1/en
Publication of SK9799A3 publication Critical patent/SK9799A3/sk
Publication of SK286461B6 publication Critical patent/SK286461B6/sk

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Detergent Compositions (AREA)
  • Coloring (AREA)
SK97-99A 1996-07-24 1997-07-23 [1,5-a]-Pyrazolo-1,3,5-triazíny, ich použitie a farmaceutické kompozície na ich báze SK286461B6 (sk)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US68604796A 1996-07-24 1996-07-24
US2329096P 1996-07-24 1996-07-24
US08/899,242 US6124289A (en) 1996-07-24 1997-07-23 Azolo triazines and pyrimidines
PCT/US1997/013072 WO1998003510A1 (en) 1996-07-24 1997-07-23 AZOLO TRIAZINES AND PYRIMIDINES

Publications (2)

Publication Number Publication Date
SK9799A3 SK9799A3 (sk) 2005-04-01
SK286461B6 true SK286461B6 (sk) 2008-10-07

Family

ID=27362048

Family Applications (1)

Application Number Title Priority Date Filing Date
SK97-99A SK286461B6 (sk) 1996-07-24 1997-07-23 [1,5-a]-Pyrazolo-1,3,5-triazíny, ich použitie a farmaceutické kompozície na ich báze

Country Status (15)

Country Link
JP (2) JP4704521B2 (no)
CN (3) CN1104432C (no)
AR (1) AR049583A2 (no)
BR (1) BR9710544A (no)
CA (1) CA2259583C (no)
CZ (1) CZ299451B6 (no)
EA (1) EA004403B1 (no)
EE (1) EE04316B1 (no)
HR (1) HRP970413A2 (no)
IL (4) IL127871A0 (no)
NO (1) NO315610B1 (no)
NZ (1) NZ333777A (no)
PL (1) PL195762B1 (no)
SI (1) SI9720045B (no)
SK (1) SK286461B6 (no)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0208357A (pt) * 2001-03-13 2004-06-29 Bristol Myers Squibb Pharma Co Composto, composição farmacêutica, método de antagonização de um receptor de fator de liberação de corticotropina (crf), método de tratamento de disfunção, método de triagem de ligantes, método de detecção de receptores de crf, método de inibição da ligação de crf, artigo industrializado e usos do composto
WO2004110454A1 (ja) * 2003-06-13 2004-12-23 Ishihara Sangyo Kaisha, Ltd. アデノシンA2a受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物
US7329662B2 (en) * 2003-10-03 2008-02-12 Hoffmann-La Roche Inc. Pyrazolo-pyridine
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
UA96458C2 (ru) * 2006-09-20 2011-11-10 Эли Лилли Энд Компани Тиазолпиразолопиримидиновые соединения как антагонисты рецептора crf1
CN103694242B (zh) * 2013-12-10 2016-01-06 昆明翔昊科技有限公司 吡唑并嘧啶类化合物及其药物组合物和其在制药中的应用
AU2018317398A1 (en) 2017-08-14 2019-11-21 Spruce Biosciences, Inc. Corticotropin releasing factor receptor antagonists
CN112592346B (zh) * 2019-07-30 2022-04-26 厦门宝太生物科技股份有限公司 一种a2a和/或a2b抑制剂中间体的制备方法
MX2023001688A (es) 2020-08-12 2023-02-22 Spruce Biosciences Inc Metodos y composiciones para tratar el sindrome de ovario poliquistico.
US11708372B2 (en) 2021-11-19 2023-07-25 Spruce Biosciences, Inc. Crystalline composition of tildacerfont and methods of use and preparation thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3995039A (en) * 1975-05-27 1976-11-30 Merck & Co., Inc. Pyrazolo [1,5-a] [1,3,5] triazines
JPS6157587A (ja) * 1984-08-29 1986-03-24 Shionogi & Co Ltd 縮合複素環誘導体および抗潰瘍剤
US4824834A (en) * 1986-10-31 1989-04-25 Otsuka Pharmaceutical Company, Limited Pyrazolotriazine compounds
JP2691317B2 (ja) * 1989-08-25 1997-12-17 株式会社大塚製薬工場 4―ヒドロキシ―8―(3―低級アルコキシ―4―フェニルスルフィニルフェニル)ピラゾロ〔1,5―a〕―1,3,5―トリアジン光学活性体の塩類及びその製造方法
WO1992006096A1 (en) * 1990-10-09 1992-04-16 Otsuka Pharmaceutical Co., Ltd. Pyrimidine derivative, production thereof, and androgen inhibitor
ES2126573T3 (es) * 1991-04-22 1999-04-01 Otsuka Pharma Co Ltd Derivado de pirazol (1,5-a)pirimidina y agente antiinflamatorio que contiene este derivado.
US5356897A (en) * 1991-09-09 1994-10-18 Fujisawa Pharmaceutical Co., Ltd. 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines

Also Published As

Publication number Publication date
SI9720045B (sl) 2008-02-29
EA199900158A1 (ru) 1999-10-28
PL331523A1 (en) 1999-07-19
JP2005097257A (ja) 2005-04-14
IL127871A0 (en) 1999-10-28
JP4194539B2 (ja) 2008-12-10
IL127871A (en) 2010-04-29
SI9720045A (sl) 1999-10-31
PL195762B1 (pl) 2007-10-31
NO990264L (no) 1999-03-10
CN1104432C (zh) 2003-04-02
EE9900019A (et) 1999-08-16
NZ333777A (en) 2000-07-28
AR049583A2 (es) 2006-08-16
IL164513A0 (en) 2005-12-18
CN1250223C (zh) 2006-04-12
NO990264D0 (no) 1999-01-21
CN1388126A (zh) 2003-01-01
CN1225637A (zh) 1999-08-11
JP2002513382A (ja) 2002-05-08
CZ299451B6 (cs) 2008-07-30
CA2259583C (en) 2009-11-17
HRP970413A2 (en) 1998-10-31
SK9799A3 (sk) 2005-04-01
JP4704521B2 (ja) 2011-06-15
CZ18499A3 (cs) 1999-11-17
CA2259583A1 (en) 1998-01-29
NO315610B3 (no) 2003-09-29
NO315610B1 (no) 2003-09-29
IL150163A (en) 2010-12-30
EE04316B1 (et) 2004-06-15
IL164513A (en) 2010-04-29
EA004403B1 (ru) 2004-04-29
BR9710544A (pt) 1999-08-17
CN1327793A (zh) 2001-12-26

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MK4A Expiry of patent

Expiry date: 20170723