SK283420B6 - Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny - Google Patents

Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny Download PDF

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Publication number
SK283420B6
SK283420B6 SK1337-94A SK133794A SK283420B6 SK 283420 B6 SK283420 B6 SK 283420B6 SK 133794 A SK133794 A SK 133794A SK 283420 B6 SK283420 B6 SK 283420B6
Authority
SK
Slovakia
Prior art keywords
methyl
oxo
oxazolidinyl
phenyl
alkyl
Prior art date
Application number
SK1337-94A
Other languages
English (en)
Slovak (sk)
Other versions
SK133794A3 (en
Inventor
Douglas K. Hutchinson
Steven Joseph Brickner
Michael Robert Barbachyn
Ronald B. Gammill
Mahest V. Patel
Original Assignee
Pharmacia & Upjohn Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Company filed Critical Pharmacia & Upjohn Company
Publication of SK133794A3 publication Critical patent/SK133794A3/sk
Publication of SK283420B6 publication Critical patent/SK283420B6/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
SK1337-94A 1992-05-08 1992-04-21 Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny SK283420B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88043292A 1992-05-08 1992-05-08
PCT/US1993/003570 WO1993023384A1 (en) 1992-05-08 1993-04-21 Oxazolidinones containing a substituted diazine moiety and their use as antimicrobials

Publications (2)

Publication Number Publication Date
SK133794A3 SK133794A3 (en) 1995-06-07
SK283420B6 true SK283420B6 (sk) 2003-07-01

Family

ID=25376270

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1337-94A SK283420B6 (sk) 1992-05-08 1992-04-21 Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny

Country Status (26)

Country Link
US (2) US5547950A (fi)
EP (1) EP0640077B1 (fi)
JP (1) JP3255920B2 (fi)
KR (1) KR100281775B1 (fi)
CN (1) CN1044236C (fi)
AT (1) ATE219770T1 (fi)
AU (1) AU668733B2 (fi)
CA (1) CA2133079C (fi)
CZ (1) CZ281884B6 (fi)
DE (1) DE69332061T2 (fi)
DK (1) DK0640077T3 (fi)
ES (1) ES2180545T3 (fi)
FI (1) FI945246A0 (fi)
HU (2) HUT72296A (fi)
IL (1) IL105555A (fi)
LV (1) LV13075B (fi)
MX (1) MX9302665A (fi)
MY (1) MY117338A (fi)
NO (1) NO306112B1 (fi)
PL (2) PL174850B1 (fi)
PT (1) PT640077E (fi)
RU (1) RU2105003C1 (fi)
SK (1) SK283420B6 (fi)
TW (1) TW274549B (fi)
WO (1) WO1993023384A1 (fi)
ZA (1) ZA932855B (fi)

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