SK282823B6 - Derivát tienopyrimidínu, spôsob jeho prípravy a farmaceutický prostriedok, ktorý ho obsahuje - Google Patents

Derivát tienopyrimidínu, spôsob jeho prípravy a farmaceutický prostriedok, ktorý ho obsahuje Download PDF

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Publication number
SK282823B6
SK282823B6 SK164-99A SK16499A SK282823B6 SK 282823 B6 SK282823 B6 SK 282823B6 SK 16499 A SK16499 A SK 16499A SK 282823 B6 SK282823 B6 SK 282823B6
Authority
SK
Slovakia
Prior art keywords
pyrimidine
chloro
pyridin
thieno
methyl
Prior art date
Application number
SK164-99A
Other languages
English (en)
Slovak (sk)
Other versions
SK16499A3 (en
Inventor
Jonas Rochus
Pierre Schelling
Franz-Werner Kluxen
Maria Christadler
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of SK16499A3 publication Critical patent/SK16499A3/sk
Publication of SK282823B6 publication Critical patent/SK282823B6/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Gynecology & Obstetrics (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SK164-99A 1996-08-12 1997-07-30 Derivát tienopyrimidínu, spôsob jeho prípravy a farmaceutický prostriedok, ktorý ho obsahuje SK282823B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19632423A DE19632423A1 (de) 1996-08-12 1996-08-12 Thienopyrimidine
PCT/EP1997/004139 WO1998006722A1 (de) 1996-08-12 1997-07-30 Thienopyrimidine

Publications (2)

Publication Number Publication Date
SK16499A3 SK16499A3 (en) 1999-06-11
SK282823B6 true SK282823B6 (sk) 2002-12-03

Family

ID=7802392

Family Applications (1)

Application Number Title Priority Date Filing Date
SK164-99A SK282823B6 (sk) 1996-08-12 1997-07-30 Derivát tienopyrimidínu, spôsob jeho prípravy a farmaceutický prostriedok, ktorý ho obsahuje

Country Status (29)

Country Link
US (1) US6110920A (ko)
EP (1) EP0920431B1 (ko)
JP (1) JP4405593B2 (ko)
KR (1) KR100502271B1 (ko)
CN (1) CN1081638C (ko)
AR (1) AR009052A1 (ko)
AT (1) ATE233265T1 (ko)
AU (1) AU725227B2 (ko)
BR (1) BR9711062A (ko)
CA (1) CA2263561C (ko)
CZ (1) CZ287772B6 (ko)
DE (2) DE19632423A1 (ko)
DK (1) DK0920431T3 (ko)
ES (1) ES2191192T3 (ko)
HK (1) HK1021731A1 (ko)
HU (1) HUP0001607A3 (ko)
IL (1) IL128504A (ko)
NO (1) NO990643D0 (ko)
NZ (1) NZ334600A (ko)
PL (1) PL190174B1 (ko)
PT (1) PT920431E (ko)
RU (1) RU2199541C2 (ko)
SI (1) SI0920431T1 (ko)
SK (1) SK282823B6 (ko)
TR (1) TR199900308T2 (ko)
TW (1) TW359672B (ko)
UA (1) UA55421C2 (ko)
WO (1) WO1998006722A1 (ko)
ZA (1) ZA977156B (ko)

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US6399826B1 (en) 1999-08-11 2002-06-04 Sepracor Inc. Salts of sibutramine metabolites, methods of making sibutramine metabolites and intermediates useful in the same, and methods of treating pain
DE10031585A1 (de) * 2000-06-29 2002-01-10 Merck Patent Gmbh 2-Aminoalkyl-thieno[2,3-d]pyrimidine
KR20030034232A (ko) * 2000-09-29 2003-05-01 닛뽕소다 가부시키가이샤 티에노피리미딘 화합물 및 그 염 및 제조방법
HUP0303005A3 (en) * 2001-02-02 2005-05-30 Merck Patent Gmbh Pharmaceutical compositions comprising pyrazolo[4,3-d]pyrimidines or thienopyrimidines and endothelin receptor antagonists
WO2002083631A1 (en) 2001-04-13 2002-10-24 Sepracor Inc. Methods of preparing didesmethylsibutramine and other sibutramine derivatives
CN100343258C (zh) * 2001-04-30 2007-10-17 美国拜尔公司 新的4－氨基－5,6－取代的噻吩并[2,3－d]嘧啶化合物
WO2003035653A1 (fr) * 2001-10-26 2003-05-01 Nippon Soda Co.,Ltd. Compose pyridothienopyrimidine et son sel
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US7893101B2 (en) 2002-03-20 2011-02-22 Celgene Corporation Solid forms comprising (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione, compositions thereof, and uses thereof
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BRPI0918055A2 (pt) 2008-09-02 2015-12-01 Addex Pharmaceuticals Sa derivados de 3-azabiciclo[3,1,0]hexila como moduladores de receptores metabotrópicos de glutamato.
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JP5690277B2 (ja) 2008-11-28 2015-03-25 ジャンセン ファーマシューティカルズ， インコーポレイテッド． 代謝型グルタミン酸受容体の調節因子としてのインドールおよびベンゾオキサジン誘導体
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Also Published As

Publication number Publication date
SI0920431T1 (en) 2003-08-31
CZ287772B6 (en) 2001-01-17
DE19632423A1 (de) 1998-02-19
KR100502271B1 (ko) 2005-07-22
ZA977156B (en) 1998-02-19
CZ44899A3 (cs) 1999-05-12
AU4203597A (en) 1998-03-06
AU725227B2 (en) 2000-10-12
DK0920431T3 (da) 2003-06-02
RU2199541C2 (ru) 2003-02-27
KR20000029932A (ko) 2000-05-25
NO990643L (no) 1999-02-11
IL128504A (en) 2003-01-12
HK1021731A1 (en) 2000-06-30
IL128504A0 (en) 2000-01-31
UA55421C2 (uk) 2003-04-15
EP0920431A1 (de) 1999-06-09
CA2263561A1 (en) 1998-02-19
SK16499A3 (en) 1999-06-11
CA2263561C (en) 2007-02-20
HUP0001607A3 (en) 2002-09-30
CN1227560A (zh) 1999-09-01
TW359672B (en) 1999-06-01
JP2000516223A (ja) 2000-12-05
ATE233265T1 (de) 2003-03-15
PL190174B1 (pl) 2005-11-30
PT920431E (pt) 2003-07-31
NO990643D0 (no) 1999-02-11
HUP0001607A2 (hu) 2000-10-28
DE59709404D1 (en) 2003-04-03
TR199900308T2 (xx) 1999-04-21
ES2191192T3 (es) 2003-09-01
JP4405593B2 (ja) 2010-01-27
WO1998006722A1 (de) 1998-02-19
US6110920A (en) 2000-08-29
BR9711062A (pt) 1999-08-17
AR009052A1 (es) 2000-03-08
CN1081638C (zh) 2002-03-27
NZ334600A (en) 2000-07-28
PL331538A1 (en) 1999-07-19
EP0920431B1 (de) 2003-02-26

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