SK282424B6 - "S" a "T" kryštalické formy 1-[5-metánsulfónamidoindolyl-2- karbonyl]-4-[3-(1-metyl-etylamino)-2-pyridinyl] piperazínu - Google Patents

"S" a "T" kryštalické formy 1-[5-metánsulfónamidoindolyl-2- karbonyl]-4-[3-(1-metyl-etylamino)-2-pyridinyl] piperazínu Download PDF

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Publication number
SK282424B6
SK282424B6 SK1229-96A SK122996A SK282424B6 SK 282424 B6 SK282424 B6 SK 282424B6 SK 122996 A SK122996 A SK 122996A SK 282424 B6 SK282424 B6 SK 282424B6
Authority
SK
Slovakia
Prior art keywords
pyridinyl
carbonyl
methanesulfonamidoindolyl
methylethylamino
piperazine
Prior art date
Application number
SK1229-96A
Other languages
English (en)
Slovak (sk)
Other versions
SK122996A3 (en
Inventor
Jeffrey L. Havens
Donald P. Smith
Michael S. Bergren
Mark A. Lyster
Original Assignee
Pharmacia + Upjohn Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia + Upjohn Company filed Critical Pharmacia + Upjohn Company
Publication of SK122996A3 publication Critical patent/SK122996A3/sk
Publication of SK282424B6 publication Critical patent/SK282424B6/sk

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Virology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Indole Compounds (AREA)
SK1229-96A 1994-04-15 1995-03-01 "S" a "T" kryštalické formy 1-[5-metánsulfónamidoindolyl-2- karbonyl]-4-[3-(1-metyl-etylamino)-2-pyridinyl] piperazínu SK282424B6 (sk)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22786094A 1994-04-15 1994-04-15
US31178094A 1994-09-23 1994-09-23
PCT/US1995/002166 WO1995028398A1 (en) 1994-04-15 1995-03-01 Novel crystal forms of 1-[5-methanesulfonamidoindolyl-2-carbonyl]-4-[3-(1-methylethylamino)-2-pyridinyl]piperazine

Publications (2)

Publication Number Publication Date
SK122996A3 SK122996A3 (en) 1997-05-07
SK282424B6 true SK282424B6 (sk) 2002-01-07

Family

ID=26921831

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1229-96A SK282424B6 (sk) 1994-04-15 1995-03-01 "S" a "T" kryštalické formy 1-[5-metánsulfónamidoindolyl-2- karbonyl]-4-[3-(1-metyl-etylamino)-2-pyridinyl] piperazínu

Country Status (26)

Country Link
US (1) US6452007B1 (zh)
EP (1) EP0755393B1 (zh)
JP (1) JP3817261B2 (zh)
KR (1) KR100364941B1 (zh)
CN (1) CN1147253A (zh)
AT (1) ATE207481T1 (zh)
AU (1) AU693939B2 (zh)
CA (1) CA2184598C (zh)
CZ (1) CZ287164B6 (zh)
DE (1) DE69523447T2 (zh)
DK (1) DK0755393T3 (zh)
ES (1) ES2164147T3 (zh)
FI (1) FI111364B (zh)
HU (1) HU226827B1 (zh)
IL (1) IL113162A (zh)
LV (1) LV12957B (zh)
MX (1) MX9604831A (zh)
MY (1) MY116830A (zh)
NO (1) NO310024B1 (zh)
NZ (1) NZ282211A (zh)
PL (1) PL180776B1 (zh)
PT (1) PT755393E (zh)
RU (1) RU2136677C1 (zh)
SK (1) SK282424B6 (zh)
TW (1) TW393478B (zh)
WO (1) WO1995028398A1 (zh)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4827296B2 (ja) 1998-06-11 2011-11-30 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー デラビルジン錠製剤
US6872811B1 (en) 1998-09-30 2005-03-29 Millennium Pharmaceuticals, Inc. HRPCa9 and HRPCa10 nucleic acids and polypeptides
DE102011113749A1 (de) * 2011-09-14 2013-03-14 Aicuris Gmbh & Co. Kg Sulfonsäuresalze Heterocyclylamid-substituiertr Imidazole

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3565924A (en) 1968-07-01 1971-02-23 Wisconsin Alumni Res Found 25-hydroxycholfcalciferol
US3833622A (en) 1969-03-17 1974-09-03 Upjohn Co Crystalline 25-hydroxycholecalciferol hydrate and structurally related compounds
GB1532682A (en) 1976-04-27 1978-11-22 Bristol Myers Co Process for the preparation of cephadroxil
IL63968A (en) 1980-10-01 1985-10-31 Glaxo Group Ltd Form 2 ranitidine hydrochloride,its preparation and pharmaceutical compositions containing it
AU654808B2 (en) * 1989-12-28 1994-11-24 Pharmacia & Upjohn Company Diaromatic substituted anti-aids compounds
US5563142A (en) * 1989-12-28 1996-10-08 The Upjohn Company Diaromatic substituted compounds as anti-HIV-1 agents
US5599930A (en) * 1991-07-03 1997-02-04 The Upjohn Company Substituted indoles as anti-AIDS pharmaceuticals

Also Published As

Publication number Publication date
JPH09512007A (ja) 1997-12-02
HUT76467A (en) 1997-09-29
CZ294296A3 (en) 1997-01-15
FI964114A (fi) 1996-10-14
DE69523447D1 (de) 2001-11-29
IL113162A0 (en) 1995-06-29
CZ287164B6 (en) 2000-10-11
HU9602857D0 (en) 1996-12-30
US6452007B1 (en) 2002-09-17
JP3817261B2 (ja) 2006-09-06
WO1995028398A1 (en) 1995-10-26
AU693939B2 (en) 1998-07-09
ATE207481T1 (de) 2001-11-15
EP0755393B1 (en) 2001-10-24
CA2184598C (en) 2005-05-03
PT755393E (pt) 2002-04-29
IL113162A (en) 1999-04-11
KR100364941B1 (ko) 2003-02-19
FI964114A0 (fi) 1996-10-14
DE69523447T2 (de) 2002-05-16
NZ282211A (en) 1997-10-24
MX9604831A (es) 1998-05-31
PL316688A1 (en) 1997-02-03
CN1147253A (zh) 1997-04-09
DK0755393T3 (da) 2001-12-17
KR970702275A (ko) 1997-05-13
MY116830A (en) 2004-04-30
LV12957B (en) 2003-04-20
RU2136677C1 (ru) 1999-09-10
SK122996A3 (en) 1997-05-07
NO964386L (no) 1996-10-15
CA2184598A1 (en) 1995-10-26
HU226827B1 (en) 2009-11-30
ES2164147T3 (es) 2002-02-16
FI111364B (fi) 2003-07-15
PL180776B1 (pl) 2001-04-30
TW393478B (en) 2000-06-11
AU3513695A (en) 1995-11-10
NO310024B1 (no) 2001-05-07
NO964386D0 (no) 1996-10-15
EP0755393A1 (en) 1997-01-29

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